Inhibitors of Mitochondrial Human Carbonic Anhydrases VA and VB as a Therapeutic Strategy against Paclitaxel-Induced Neuropathic Pain in Mice.
CA VA and VB
Taxus brevifolia
carbonic anhydrase
glial cells
mitochondria
neuropathic pain
neuroprotection
Journal
International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791
Informations de publication
Date de publication:
02 Jun 2022
02 Jun 2022
Historique:
received:
21
04
2022
revised:
26
05
2022
accepted:
30
05
2022
entrez:
10
6
2022
pubmed:
11
6
2022
medline:
14
6
2022
Statut:
epublish
Résumé
Neuropathy development is a major dose-limiting side effect of anticancer treatments that significantly reduces patient's quality of life. The inadequate pharmacological approaches for neuropathic pain management warrant the identification of novel therapeutic targets. Mitochondrial dysfunctions that lead to reactive oxygen species (ROS) increase, cytosolic Ca
Identifiants
pubmed: 35682907
pii: ijms23116229
doi: 10.3390/ijms23116229
pmc: PMC9181376
pii:
doi:
Substances chimiques
Carbonic Anhydrase Inhibitors
0
Carbonic Anhydrases
EC 4.2.1.1
Paclitaxel
P88XT4IS4D
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : Italian Ministry of University and Research
ID : not available
Organisme : University of Florence
ID : not available
Organisme : NeuroDeRisk
ID : 821528
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