The Selective Agonist for Sphingosine-1-Phosphate Receptors Siponimod Increases the Expression Level of

CNS resident cells NR4A NURR1 fingolimod multiple sclerosis siponimod sphingosine-1-phosphate (S1P) receptors

Journal

Current issues in molecular biology
ISSN: 1467-3045
Titre abrégé: Curr Issues Mol Biol
Pays: Switzerland
ID NLM: 100931761

Informations de publication

Date de publication:
07 Mar 2022
Historique:
received: 28 01 2022
revised: 23 02 2022
accepted: 01 03 2022
entrez: 20 6 2022
pubmed: 21 6 2022
medline: 21 6 2022
Statut: epublish

Résumé

Fingolimod (FTY720) and siponimod (BAF312) are selective agonists for sphingosine-1-phosphate (S1P) receptors approved for the treatment of relapsing-remitting (RR) and secondary progressive (SP) multiple sclerosis (MS), respectively. BAF312 exerts pro-myelination and neuro-protective functions on CNS resident cells, although the underlying molecular mechanism is not yet fully understood.

Identifiants

pubmed: 35723306
pii: cimb44030083
doi: 10.3390/cimb44030083
pmc: PMC8947415
doi:

Types de publication

Journal Article

Langues

eng

Pagination

1247-1256

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Auteurs

Francesca Montarolo (F)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.
Neurology Department and Regional Referring Center of Multiple Sclerosis (CReSM), University Hospital San Luigi Gonzaga, 10043 Orbassano, Italy.
Department of Molecular Biotechnology and Health Sciences, University of Turin, 10126 Turin, Italy.

Serena Martire (S)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.
Neurology Department and Regional Referring Center of Multiple Sclerosis (CReSM), University Hospital San Luigi Gonzaga, 10043 Orbassano, Italy.
Department of Neuroscience "Rita Levi Montalcini", University of Turin, 10126 Turin, Italy.

Fabiana Marnetto (F)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.
Neurology Department and Regional Referring Center of Multiple Sclerosis (CReSM), University Hospital San Luigi Gonzaga, 10043 Orbassano, Italy.

Paola Valentino (P)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.
Neurology Department and Regional Referring Center of Multiple Sclerosis (CReSM), University Hospital San Luigi Gonzaga, 10043 Orbassano, Italy.
Department of Neuroscience "Rita Levi Montalcini", University of Turin, 10126 Turin, Italy.

Sabdi Valverde (S)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.
Neurology Department and Regional Referring Center of Multiple Sclerosis (CReSM), University Hospital San Luigi Gonzaga, 10043 Orbassano, Italy.

Marco Alfonso Capobianco (MA)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.
Neurology Department and Regional Referring Center of Multiple Sclerosis (CReSM), University Hospital San Luigi Gonzaga, 10043 Orbassano, Italy.

Antonio Bertolotto (A)

Neuroscience Institute Cavalieri Ottolenghi (NICO), 10043 Orbassano, Italy.

Classifications MeSH