Molecular Structure-Based Screening of the Constituents of
Calotropis procera
alpha glucosidase
cheminformatics
diabetes
molecular docking
molecular dynamics simulations
Journal
Current issues in molecular biology
ISSN: 1467-3045
Titre abrégé: Curr Issues Mol Biol
Pays: Switzerland
ID NLM: 100931761
Informations de publication
Date de publication:
21 Feb 2022
21 Feb 2022
Historique:
received:
25
12
2021
revised:
07
01
2022
accepted:
09
01
2022
entrez:
20
6
2022
pubmed:
21
6
2022
medline:
21
6
2022
Statut:
epublish
Résumé
Diabetes mellitus is a disorder characterized by higher levels of blood glucose due to impaired insulin mechanisms. Alpha glucosidase is a critical drug target implicated in the mechanisms of diabetes mellitus and its inhibition controls hyperglycemia. Since the existing standard synthetic drugs have therapeutic limitations, it is imperative to identify new potent inhibitors of natural product origin which may slow carbohydrate digestion and absorption via alpha glucosidase. Since plant extracts from
Identifiants
pubmed: 35723349
pii: cimb44020064
doi: 10.3390/cimb44020064
pmc: PMC8928985
doi:
Types de publication
Journal Article
Langues
eng
Pagination
963-987Références
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