Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors.
Journal
Journal of medicinal chemistry
ISSN: 1520-4804
Titre abrégé: J Med Chem
Pays: United States
ID NLM: 9716531
Informations de publication
Date de publication:
14 07 2022
14 07 2022
Historique:
pubmed:
22
6
2022
medline:
16
7
2022
entrez:
21
6
2022
Statut:
ppublish
Résumé
With over 200 million cases and close to half a million deaths each year, malaria is a threat to global health, particularly in developing countries.
Identifiants
pubmed: 35727231
doi: 10.1021/acs.jmedchem.2c00611
pmc: PMC10152543
mid: NIHMS1892919
doi:
Substances chimiques
Antimalarials
0
Artemisinins
0
Peptides
0
Proteasome Inhibitors
0
Protozoan Proteins
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Research Support, N.I.H., Extramural
Langues
eng
Sous-ensembles de citation
IM
Pagination
9350-9375Subventions
Organisme : NIAID NIH HHS
ID : R01 AI143714
Pays : United States
Organisme : NIAID NIH HHS
ID : R21 AI123794
Pays : United States
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