Protocetraric and Salazinic Acids as Potential Inhibitors of SARS-CoV-2 3CL Protease: Biochemical, Cytotoxic, and Computational Characterization of Depsidones as Slow-Binding Inactivators.
SARS-CoV-2 3CL protease
cysteine enzyme
inactivator
inhibition assay
lichen secondary metabolites
slow binding inhibitor
Journal
Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453
Informations de publication
Date de publication:
04 Jun 2022
04 Jun 2022
Historique:
received:
16
05
2022
revised:
01
06
2022
accepted:
02
06
2022
entrez:
24
6
2022
pubmed:
25
6
2022
medline:
25
6
2022
Statut:
epublish
Résumé
The study investigated the inhibitory activity of protocetraric and salazinic acids against SARS-CoV-2 3CL
Identifiants
pubmed: 35745633
pii: ph15060714
doi: 10.3390/ph15060714
pmc: PMC9227325
pii:
doi:
Types de publication
Journal Article
Langues
eng
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