High Affinity Decynium-22 Binding to Brain Membrane Homogenates and Reduced Dorsal Camouflaging after Acute Exposure to it in Zebrafish.
Danio rerio (zebrafish)
SLC22A
anxiety
black–white plus maze
dive tank
predator avoidance
pseudoisocyanine
uptake 2 transporters
Journal
Frontiers in pharmacology
ISSN: 1663-9812
Titre abrégé: Front Pharmacol
Pays: Switzerland
ID NLM: 101548923
Informations de publication
Date de publication:
2022
2022
Historique:
received:
22
12
2021
accepted:
29
03
2022
entrez:
27
6
2022
pubmed:
28
6
2022
medline:
28
6
2022
Statut:
epublish
Résumé
Organic cation transporters (OCTs) are expressed in the mammalian brain, kidney, liver, placenta, and intestines, where they facilitate the transport of cations and other substrates between extracellular fluids and cells. Despite increasing reliance on ectothermic vertebrates as alternative toxicology models, properties of their OCT homologs transporting many drugs and toxins remain poorly characterized. Recently, in zebrafish (
Identifiants
pubmed: 35754508
doi: 10.3389/fphar.2022.841423
pii: 841423
pmc: PMC9218599
doi:
Types de publication
Journal Article
Langues
eng
Pagination
841423Informations de copyright
Copyright © 2022 Gould, Barba-Escobedo, Horton and Daws.
Déclaration de conflit d'intérêts
The authors declare that the research was conducted in the absence of any commercial or financial relationships that could be construed as a potential conflict of interest.
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