Preparation and Characterization of Lidocaine-Loaded, Microemulsion-Based Topical Gels.
Lidocaine
Local Anesthesia
Microemulsion
Microemulsion-Based Gel
Phase Diagrams
Skin Permeation
Journal
Iranian journal of pharmaceutical research : IJPR
ISSN: 1726-6890
Titre abrégé: Iran J Pharm Res
Pays: Netherlands
ID NLM: 101208407
Informations de publication
Date de publication:
Dec 2022
Dec 2022
Historique:
received:
14
03
2021
revised:
07
06
2021
accepted:
07
06
2021
entrez:
29
6
2022
pubmed:
30
6
2022
medline:
30
6
2022
Statut:
epublish
Résumé
Microemulsion-based gels (MBGs) were prepared for transdermal delivery of lidocaine and evaluated for their potential for local anesthesia. Lidocaine solubility was measured in various oils, and phase diagrams were constructed to map the concentration range of oil, surfactant, cosurfactant, and water for oil-in-water (o/w) microemulsion (ME) domains, employing the water titration method at different surfactant/cosurfactant weight ratios. Refractive index, electrical conductivity, droplet size, zeta potential, pH, viscosity, and stability of fluid o/w MEs were evaluated. Carbomer
Identifiants
pubmed: 35765506
doi: 10.5812/ijpr.123787
pmc: PMC9191217
doi:
Types de publication
Journal Article
Langues
eng
Pagination
e123787Informations de copyright
Copyright © 2022, Author(s).
Déclaration de conflit d'intérêts
Conflict of Interests: The authors declared that there is no conflict of interest.
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