Novel Coumarin-Pyridine Hybrids as Potent Multi-Target Directed Ligands Aiming at Symptoms of Alzheimer's Disease.

Alzheimer’s disease cholinesterase inhibitors coumarin derivatives docking study neurodegenerative diseases

Journal

Frontiers in chemistry
ISSN: 2296-2646
Titre abrégé: Front Chem
Pays: Switzerland
ID NLM: 101627988

Informations de publication

Date de publication:
2022
Historique:
received: 13 03 2022
accepted: 16 05 2022
entrez: 18 7 2022
pubmed: 19 7 2022
medline: 19 7 2022
Statut: epublish

Résumé

In this research, a series of coumarin-based scaffolds linked to pyridine derivatives

Identifiants

pubmed: 35844650
doi: 10.3389/fchem.2022.895483
pii: 895483
pmc: PMC9280334
doi:

Types de publication

Journal Article

Langues

eng

Pagination

895483

Informations de copyright

Copyright © 2022 Babaei, Küçükkılınç, Jalili-Baleh, Nadri, Öz, Forootanfar, Hosseinzadeh, Akbari, Ardestani, Firoozpour, Foroumadi, Sharifzadeh, Mirjalili and Khoobi.

Déclaration de conflit d'intérêts

The authors declare that the research was conducted in the absence of any commercial or financial relationships that could be construed as a potential conflict of interest. The handling editor MS declared a shared affiliation with the authors EH, SM, MS, MK at the time of review.

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Auteurs

Elaheh Babaei (E)

Department of Chemistry, Faculty of Science, Yazd University, Yazd, Iran.

Tuba Tüylü Küçükkılınç (TT)

Department of Biochemistry, Faculty of Pharmacy, Hacettepe University, Ankara, Turkey.

Leili Jalili-Baleh (L)

Department of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences, Tehran University of Medical Science, Tehran, Iran.

Hamid Nadri (H)

Faculty of Pharmacy, Shahid Sadoughi University of Medical Sciences, Yazd, Iran.

Esin Öz (E)

Department of Biochemistry, Faculty of Pharmacy, Hacettepe University, Ankara, Turkey.

Hamid Forootanfar (H)

Department of Pharmaceutical Biotechnology, Faculty of Pharmacy, Kerman University of Medical Sciences, Kerman, Iran.

Elaheh Hosseinzadeh (E)

The Institute of Pharmaceutical Sciences (TIPS), Tehran University of Medical Sciences, Tehran, Iran.

Tayebeh Akbari (T)

Department of Microbiology, Islamic Azad University, North Tehran Branch, Tehran, Iran.

Mehdi Shafiee Ardestani (MS)

Department of Radiopharmacy, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Iran.

Loghman Firoozpour (L)

Department of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences, Tehran University of Medical Science, Tehran, Iran.

Alireza Foroumadi (A)

Department of Medicinal Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences, Tehran University of Medical Science, Tehran, Iran.

Mohammad Sharifzadeh (M)

Department of Toxicology and Pharmacology, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Iran.

Bi Bi Fatemeh Mirjalili (BBF)

Department of Chemistry, Faculty of Science, Yazd University, Yazd, Iran.

Mehdi Khoobi (M)

The Institute of Pharmaceutical Sciences (TIPS), Tehran University of Medical Sciences, Tehran, Iran.
Department of Radiopharmacy, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Iran.

Classifications MeSH