Digoxin Derivatives Sensitize a

Pdr5p Saccharomyces cerevisiae digoxin efflux pump fluconazole yeast

Journal

Journal of fungi (Basel, Switzerland)
ISSN: 2309-608X
Titre abrégé: J Fungi (Basel)
Pays: Switzerland
ID NLM: 101671827

Informations de publication

Date de publication:
25 Jul 2022
Historique:
received: 28 06 2022
revised: 21 07 2022
accepted: 21 07 2022
entrez: 27 7 2022
pubmed: 28 7 2022
medline: 28 7 2022
Statut: epublish

Résumé

The poor outcome of treatments for fungal infections is a consequence of the increasing incidence of resistance to antifungal agents, mainly due to the overexpression of efflux pumps. To surpass this mechanism of resistance, a substance able to inhibit these pumps could be administered in association with antifungals.

Identifiants

pubmed: 35893137
pii: jof8080769
doi: 10.3390/jof8080769
pmc: PMC9330353
pii:
doi:

Types de publication

Journal Article

Langues

eng

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Auteurs

Daniel Clemente de Moraes (DC)

Departamento de Microbiologia Geral, Instituto de Microbiologia Paulo de Góes, Centro de Ciências da Saúde, Universidade Federal do Rio de Janeiro, Cidade Universitária, Avenida Carlos Chagas Filho 373, Rio de Janeiro 21941-590, Brazil.

Ana Claudia Tessis (AC)

Instituto Federal do Rio de Janeiro, Rua Senador Furtado 121, Rio de Janeiro 20270-021, Brazil.

Rodrigo Rollin-Pinheiro (R)

Departamento de Microbiologia Geral, Instituto de Microbiologia Paulo de Góes, Centro de Ciências da Saúde, Universidade Federal do Rio de Janeiro, Cidade Universitária, Avenida Carlos Chagas Filho 373, Rio de Janeiro 21941-590, Brazil.

Jefferson Luiz Princival (JL)

Laboratory of Cell Biochemistry, Universidade Federal de São João del Rei, Campus Centro-Oeste Dona Lindu, Avenida Sebastião Gonçalves Coelho 400, Divinópolis 35501-296, Brazil.

José Augusto Ferreira Perez Villar (JAFP)

Laboratory of Cell Biochemistry, Universidade Federal de São João del Rei, Campus Centro-Oeste Dona Lindu, Avenida Sebastião Gonçalves Coelho 400, Divinópolis 35501-296, Brazil.

Leandro Augusto Barbosa (LA)

Laboratory of Cell Biochemistry, Universidade Federal de São João del Rei, Campus Centro-Oeste Dona Lindu, Avenida Sebastião Gonçalves Coelho 400, Divinópolis 35501-296, Brazil.

Eliana Barreto-Bergter (E)

Departamento de Microbiologia Geral, Instituto de Microbiologia Paulo de Góes, Centro de Ciências da Saúde, Universidade Federal do Rio de Janeiro, Cidade Universitária, Avenida Carlos Chagas Filho 373, Rio de Janeiro 21941-590, Brazil.

Antônio Ferreira-Pereira (A)

Departamento de Microbiologia Geral, Instituto de Microbiologia Paulo de Góes, Centro de Ciências da Saúde, Universidade Federal do Rio de Janeiro, Cidade Universitária, Avenida Carlos Chagas Filho 373, Rio de Janeiro 21941-590, Brazil.

Classifications MeSH