Identification of RAD51-BRCA2 Inhibitors Using


Journal

ACS medicinal chemistry letters
ISSN: 1948-5875
Titre abrégé: ACS Med Chem Lett
Pays: United States
ID NLM: 101521073

Informations de publication

Date de publication:
11 Aug 2022
Historique:
received: 15 02 2022
accepted: 22 07 2022
entrez: 18 8 2022
pubmed: 19 8 2022
medline: 19 8 2022
Statut: epublish

Résumé

RAD51 is an ATP-dependent recombinase, recruited by BRCA2 to mediate DNA double-strand breaks repair through homologous recombination and represents an attractive cancer drug target. Herein, we applied for the first-time protein-templated dynamic combinatorial chemistry on RAD51 as a hit identification strategy. Upon design of

Identifiants

pubmed: 35978685
doi: 10.1021/acsmedchemlett.2c00063
pmc: PMC9377020
doi:

Types de publication

Journal Article

Langues

eng

Pagination

1262-1269

Informations de copyright

© 2022 The Authors. Published by American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

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Auteurs

Greta Bagnolini (G)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.
Department of Pharmacy and Biotechnology (FaBiT), University of Bologna, 40126 Bologna, Italy.
Helmholtz Centre for Infection Research (HZI), Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), 66123 Saarbrücken, Germany.

Beatrice Balboni (B)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.
Department of Pharmacy and Biotechnology (FaBiT), University of Bologna, 40126 Bologna, Italy.

Fabrizio Schipani (F)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.

Dario Gioia (D)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.

Marina Veronesi (M)

Structural Biophysics and Translational Pharmacology, Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.
D3-PharmaChemistry, Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.

Francesca De Franco (F)

TES Pharma Srl, I-06073 Corciano, Perugia Italy.

Cansu Kaya (C)

Helmholtz Centre for Infection Research (HZI), Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), 66123 Saarbrücken, Germany.
Department of Pharmacy, Saarland University, 66123 Saarbrücken, Germany.

Ravindra P Jumde (RP)

Helmholtz Centre for Infection Research (HZI), Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), 66123 Saarbrücken, Germany.

Jose Antonio Ortega (JA)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.

Stefania Girotto (S)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.

Anna K H Hirsch (AKH)

Helmholtz Centre for Infection Research (HZI), Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), 66123 Saarbrücken, Germany.
Department of Pharmacy, Saarland University, 66123 Saarbrücken, Germany.

Marinella Roberti (M)

Department of Pharmacy and Biotechnology (FaBiT), University of Bologna, 40126 Bologna, Italy.

Andrea Cavalli (A)

Computational & Chemical Biology (CCB), Istituto Italiano di Tecnologia (IIT), 16163 Genova, Italy.
Department of Pharmacy and Biotechnology (FaBiT), University of Bologna, 40126 Bologna, Italy.

Classifications MeSH