The impact of enteric coating of aspirin on aspirin responsiveness in patients with suspected or newly diagnosed ischemic stroke: prospective cohort study: results from the (ECASIS) study.


Journal

European journal of clinical pharmacology
ISSN: 1432-1041
Titre abrégé: Eur J Clin Pharmacol
Pays: Germany
ID NLM: 1256165

Informations de publication

Date de publication:
Nov 2022
Historique:
received: 13 12 2021
accepted: 22 08 2022
pubmed: 20 9 2022
medline: 12 10 2022
entrez: 19 9 2022
Statut: ppublish

Résumé

Uncertainty remains regarding the impact of enteric-coated aspirin (EC-ASA) on secondary prevention of ischemic stroke compared to plain aspirin (P-ASA). Hence, this study was designed to investigate the effect of EC formulation on ASA response via evaluating thromboxane B2 (TXB2) levels in patients with suspected or newly diagnosed stroke. A prospective cohort study on suspected or newly diagnosed ischemic stroke patients who are aspirin-naive was conducted. Patients were received either EC aspirin or plain aspirin for at least 3 days. The primary outcome was the proportion of aspirin non-responsiveness between two groups (level of residual serum TXB2 associated with elevated thrombotic risk (< 99.0% inhibition or TXB2 > 3.1 ng/ml) within 72 h after three daily aspirin doses, while secondary outcomes were the incidence of early gastrointestinal tract (GIT) bleeding with the various aspirin preparations. (Trial registration: Clinicaltrials.gov NCT04330872 registered on 02 April 2020). Of 42 patients, ischemic strokes were confirmed in both P-ASA (81%) and EC-ASA (67%) arms. ASA non-responsiveness showed no significant difference between the two formulations (P-ASA vs. EC-ASA; 28.6% vs 23.8%; P = 0.726). Univariate and multivariate logistic regression analysis showed that patients treated with EC-ASA were more likely to have a lower rate of non-responders compared to P-ASA (unadjusted OR 0.78; 95% CI 0.20, 3.11); with the risk highest in type 2 diabetic patients with HBA1c > 6.5% (adjusted OR 6; 95% CI 1.02, 35.27; P = 0.047). No incidence of GIT bleeding observed throughout the study. A significant proportion of ASA non-responsiveness was recorded regardless of ASA formulation administered. The increased risk of ASA non-responsiveness in diabetic patients needs further exploration by larger prospective studies.

Sections du résumé

BACKGROUND AND PURPOSE OBJECTIVE
Uncertainty remains regarding the impact of enteric-coated aspirin (EC-ASA) on secondary prevention of ischemic stroke compared to plain aspirin (P-ASA). Hence, this study was designed to investigate the effect of EC formulation on ASA response via evaluating thromboxane B2 (TXB2) levels in patients with suspected or newly diagnosed stroke.
METHODS METHODS
A prospective cohort study on suspected or newly diagnosed ischemic stroke patients who are aspirin-naive was conducted. Patients were received either EC aspirin or plain aspirin for at least 3 days. The primary outcome was the proportion of aspirin non-responsiveness between two groups (level of residual serum TXB2 associated with elevated thrombotic risk (< 99.0% inhibition or TXB2 > 3.1 ng/ml) within 72 h after three daily aspirin doses, while secondary outcomes were the incidence of early gastrointestinal tract (GIT) bleeding with the various aspirin preparations. (Trial registration: Clinicaltrials.gov NCT04330872 registered on 02 April 2020).
RESULTS RESULTS
Of 42 patients, ischemic strokes were confirmed in both P-ASA (81%) and EC-ASA (67%) arms. ASA non-responsiveness showed no significant difference between the two formulations (P-ASA vs. EC-ASA; 28.6% vs 23.8%; P = 0.726). Univariate and multivariate logistic regression analysis showed that patients treated with EC-ASA were more likely to have a lower rate of non-responders compared to P-ASA (unadjusted OR 0.78; 95% CI 0.20, 3.11); with the risk highest in type 2 diabetic patients with HBA1c > 6.5% (adjusted OR 6; 95% CI 1.02, 35.27; P = 0.047). No incidence of GIT bleeding observed throughout the study.
CONCLUSION CONCLUSIONS
A significant proportion of ASA non-responsiveness was recorded regardless of ASA formulation administered. The increased risk of ASA non-responsiveness in diabetic patients needs further exploration by larger prospective studies.

Identifiants

pubmed: 36121499
doi: 10.1007/s00228-022-03391-2
pii: 10.1007/s00228-022-03391-2
pmc: PMC9546947
doi:

Substances chimiques

Glycated Hemoglobin A 0
Platelet Aggregation Inhibitors 0
Thromboxane B2 54397-85-2
Aspirin R16CO5Y76E

Banques de données

ClinicalTrials.gov
['NCT04330872']

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

1801-1811

Informations de copyright

© 2022. The Author(s).

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Auteurs

Mohamed Nabil Elshafei (MN)

Clinical Pharmacy Department, Hamad General Hospital, Hamad Medical Corporation, P.O. 3050, Doha, Qatar. mohnabil2010@yahoo.com.

Yahia Imam (Y)

Neurology Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.
Weill Cornell Medicine-Qatar, Doha, Qatar.

Arwa Ebrahim Alsaud (AE)

Internal Medicine Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.

Prem Chandra (P)

Biostatstics Section, Medical Research Center, Hamad Medical Corporation, Doha, Qatar.

Aijaz Parray (A)

The Neuroscience Institute, Academic Health Systems, Hamad Medical Corporation, Doha, Qatar.

Mohamed S Abdelmoneim (MS)

Neurology Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.
The Neuroscience Institute, Academic Health Systems, Hamad Medical Corporation, Doha, Qatar.

Khaldun Obeidat (K)

Internal Medicine Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.

Razan Saeid (R)

Internal Medicine Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.

Mohammad Ali (M)

Internal Medicine Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.

Raheem Ayadathil (R)

The Neuroscience Institute, Academic Health Systems, Hamad Medical Corporation, Doha, Qatar.

Mouhand F H Mohamed (MFH)

Internal Medicine Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.

Ibtihal M Abdallah (IM)

Clinical Pharmacy Department, Hamad General Hospital, Hamad Medical Corporation, P.O. 3050, Doha, Qatar.

Shaban Mohammed (S)

Department of Pharmacy, Hamad Medical Corporation, Doha, Qatar.

Naveed Akhtar (N)

Neurology Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.
Weill Cornell Medicine-Qatar, Doha, Qatar.

Mohammed Ibn-Masoud Danjuma (MI)

Internal Medicine Department, Hamad General Hospital, Hamad Medical Corporation, Doha, Qatar.
College of Medicine, Qatar University, Doha, Qatar.

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