Molecular Insight into
mycobacterium tuberculosis
nitrofuranyl amides
spontaneous mutagenesis
whole-genome sequencing
Journal
Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453
Informations de publication
Date de publication:
12 Sep 2022
12 Sep 2022
Historique:
received:
12
08
2022
revised:
04
09
2022
accepted:
08
09
2022
entrez:
23
9
2022
pubmed:
24
9
2022
medline:
24
9
2022
Statut:
epublish
Résumé
We performed synthesis of new nitrofuranyl amides and investigated their anti-TB activity and primary genetic response of mycobacteria through whole-genome sequencing (WGS) of spontaneous resistant mutants. The in vitro activity was assessed on reference strain
Identifiants
pubmed: 36145357
pii: ph15091136
doi: 10.3390/ph15091136
pmc: PMC9504009
pii:
doi:
Types de publication
Journal Article
Langues
eng
Subventions
Organisme : Russian Science Foundation
ID : 19-15-00028
Organisme : Federal Service for Surveillance on Consumer Rights Protection and Human Wellbeing
ID : АААА-А21-121021600206-5
Organisme : Bulgarian Science Fund
ID : KP-06-N39/7
Organisme : Bulgarian Science Fund
ID : KP-06-N41/3
Organisme : Fundação para a Ciência e Tecnologia
ID : UID/DTP/04138/2019
Organisme : Fundação para a Ciência e Tecnologia
ID : CEECIND/00394/2017
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