The Influence of the Polymer Type on the Quality of Newly Developed Oral Immediate-Release Tablets Containing Amiodarone Solid Dispersions Obtained by Hot-Melt Extrusion.
amiodarone hydrochloride
hot-melt extrusion
oral immediate release tablets
solid dispersions
Journal
Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009
Informations de publication
Date de publication:
05 Oct 2022
05 Oct 2022
Historique:
received:
13
09
2022
revised:
02
10
2022
accepted:
03
10
2022
entrez:
14
10
2022
pubmed:
15
10
2022
medline:
18
10
2022
Statut:
epublish
Résumé
The present study aims to demonstrate the influence of the polymer-carrier type and proportion on the quality performance of newly developed oral immediate-release tablets containing amiodarone solid dispersions obtained by hot-melt extrusion. Twelve solid dispersions including amiodarone and different polymers (PEG 1500, PEG 4000; PEG 8000, Soluplus
Identifiants
pubmed: 36235137
pii: molecules27196600
doi: 10.3390/molecules27196600
pmc: PMC9573735
pii:
doi:
Substances chimiques
Biological Products
0
Excipients
0
Polymers
0
Polyvinyls
0
Powders
0
Tablets
0
polyvinyl caprolactam-polyvinyl acetate-polyethylene glycol graft copolymer
0
Poloxamer
106392-12-5
Polyethylene Glycols
3WJQ0SDW1A
polyethylene glycol 4000
4R4HFI6D95
Amiodarone
N3RQ532IUT
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
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