Piperacillin Population Pharmacokinetics and Dosing Regimen Optimization in Critically Ill Children Receiving Continuous Renal Replacement Therapy.

children critical care intensive care pediatric drug therapy pediatric infectious disease pharmacology piperacillin population pharmacokinetics renal failure renal replacement therapy

Journal

Antimicrobial agents and chemotherapy
ISSN: 1098-6596
Titre abrégé: Antimicrob Agents Chemother
Pays: United States
ID NLM: 0315061

Informations de publication

Date de publication:
20 12 2022
Historique:
pubmed: 8 11 2022
medline: 23 12 2022
entrez: 7 11 2022
Statut: ppublish

Résumé

We aimed to develop a piperacillin population pharmacokinetic (PK) model in critically ill children receiving continuous renal replacement therapy (CRRT) and to optimize dosing regimens. The piperacillin plasma concentration was quantified by high-performance liquid chromatography. Piperacillin PK was investigated using a nonlinear mixed-effect modeling approach. Monte Carlo simulations were performed to compute the optimal scheme of administration according to the target of 100% interdose interval time in which concentration is one to four times above the MIC (100% fT > 1 to 4× MIC). A total of 32 children with a median (interquartile range [IQR]) postnatal age of 2 years (0 to 11), body weight (BW) of 15 kg (6 to 38), and receiving CRRT were included. Concentration-time courses were best described by a one-compartment model with first-order elimination. BW and residual diuresis (

Identifiants

pubmed: 36342152
doi: 10.1128/aac.01135-22
pmc: PMC9764994
doi:

Substances chimiques

Piperacillin X00B0D5O0E
Anti-Bacterial Agents 0
Piperacillin, Tazobactam Drug Combination 157044-21-8

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

e0113522

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Auteurs

Michael Thy (M)

Service de Maladies Infectieuses et Tropicales, Hôpital Bichat Claude Bernard, AP-HP, Université Paris Cité, Paris, France.
EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.

Saïk Urien (S)

Unité de recherche Clinique-Centre d'Investigation Clinique, Hôpital Cochin-Necker, AP-HP, Paris, France.

Frantz Foissac (F)

EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.
Unité de recherche Clinique-Centre d'Investigation Clinique, Hôpital Cochin-Necker, AP-HP, Paris, France.

Naïm Bouazza (N)

EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.
Unité de recherche Clinique-Centre d'Investigation Clinique, Hôpital Cochin-Necker, AP-HP, Paris, France.

Inès Gana (I)

Unité de recherche Clinique-Centre d'Investigation Clinique, Hôpital Cochin-Necker, AP-HP, Paris, France.

Emmanuelle Bille (E)

Service de microbiologie, Hôpital Necker Enfants-Malades, AP-HP, Université Paris Cité, Paris, France.

Agathe Béranger (A)

EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.
Service de Réanimation chirurgicale cardiaque pédiatrique, Hôpital Necker Enfants-Malades, AP-HP, Université Paris Cité, Paris, France.

Julie Toubiana (J)

Service de Pédiatrie Générale et Infectieuse, Assistance Publique-Hôpitaux de Paris, Hôpital Necker-Enfants Malades, AP-HP, Université Paris Cité, Paris, France.

Romain Berthaud (R)

Service de Néphrologie Pédiatrique, Centre de Référence MARHEA, Hôpital Necker-Enfants Malades, AP-HP, Université Paris Cité, Paris, France.

Fabrice Lesage (F)

Service de réanimation et surveillance continue médicochirurgicales, Hôpital Necker Enfants-Malades, AP-HP, Université Paris Cité, Paris, France.

Sylvain Renolleau (S)

Service de réanimation et surveillance continue médicochirurgicales, Hôpital Necker Enfants-Malades, AP-HP, Université Paris Cité, Paris, France.

Jean-Marc Tréluyer (JM)

EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.
Service de microbiologie, Hôpital Necker Enfants-Malades, AP-HP, Université Paris Cité, Paris, France.
Service de pharmacologie clinique, Hôpital Cochin, AP-HP, Université Paris Cité, Paris, France.

Sihem Benaboud (S)

EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.
Service de pharmacologie clinique, Hôpital Cochin, AP-HP, Université Paris Cité, Paris, France.

Mehdi Oualha (M)

EA7323, Evaluation des thérapeutiques et pharmacologie périnatale et pédiatrique, Université Paris Cité, Paris, France.
Service de réanimation et surveillance continue médicochirurgicales, Hôpital Necker Enfants-Malades, AP-HP, Université Paris Cité, Paris, France.

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Classifications MeSH