Genetic Study of SARS-CoV-2 Non Structural Protein 12 in COVID-19 Patients Non Responders to Remdesivir.


Journal

Microbiology spectrum
ISSN: 2165-0497
Titre abrégé: Microbiol Spectr
Pays: United States
ID NLM: 101634614

Informations de publication

Date de publication:
21 12 2022
Historique:
pubmed: 11 11 2022
medline: 28 12 2022
entrez: 10 11 2022
Statut: ppublish

Résumé

Remdesivir (RDV) was the first antiviral drug approved by the FDA to treat severe coronavirus disease-2019 (COVID-19) patients. RDV inhibits SARS-CoV-2 replication by stalling the non structural protein 12 (nsp12) subunit of the RNA-dependent RNA polymerase (RdRp). No evidence of global widespread RDV-resistance mutations has been reported, however, defining genetic pathways to RDV resistance and determining emergent mutations prior and subsequent antiviral therapy in clinical settings is necessary. This study identified 57/149 (38.3%) patients who did not respond to one course (5-days) (

Identifiants

pubmed: 36354320
doi: 10.1128/spectrum.02448-22
pmc: PMC9769853
doi:

Substances chimiques

remdesivir 3QKI37EEHE
Adenosine Monophosphate 415SHH325A
Antiviral Agents 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

e0244822

Auteurs

Marta Santos Bravo (M)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.
Institut of Global Health of Barcelona (ISGlobal), Barcelona, Spain.

Rodrigo Alonso (R)

Department of Infectious Diseases, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Dafne Soria (D)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Sonsoles Sánchez Palomino (S)

AIDS Research Group, Institut de Recerca Biomèdica August Pi i Sunyer (IDIBAPS), Barcelona, Spain.

Ángela Sanzo Machuca (Á)

Universitat Autónoma de Barcelona, Barcelona, Spain.

Cristina Rodríguez (C)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

José Alcamí (J)

AIDS Research Group, Institut de Recerca Biomèdica August Pi i Sunyer (IDIBAPS), Barcelona, Spain.
AIDS Immunopathogenesis Unit, Instituto de Salud Carlos III, Madrid, Spain.
CIBER de Enfermedades Infecciosas (CIBERINFEC), Instituto de Salud Carlos III, Madrid, Spain.

Francisco Díez-Fuertes (F)

AIDS Immunopathogenesis Unit, Instituto de Salud Carlos III, Madrid, Spain.
CIBER de Enfermedades Infecciosas (CIBERINFEC), Instituto de Salud Carlos III, Madrid, Spain.

Àlvar Simarro Redon (À)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Juan Carlos Hurtado (JC)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.
Institut of Global Health of Barcelona (ISGlobal), Barcelona, Spain.

Francesc Fernández Avilés (F)

Hematological Unit, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Marta Bodro (M)

Transplant Unit, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Elisa Rubio (E)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Jose Luis Villanueva (JL)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Andrea Vergara (A)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Pedro Castro (P)

Intensive Care Unit, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Montserrat Tuset (M)

Pharmacology Unit, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Genoveva Cuesta (G)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Pedro Puerta (P)

Department of Infectious Diseases, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Carolina García (C)

Department of Infectious Diseases, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

María Del Mar Mosquera Gutiérrez (MDM)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Miguel J Martínez (MJ)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.
Institut of Global Health of Barcelona (ISGlobal), Barcelona, Spain.
CIBER de Enfermedades Infecciosas (CIBERINFEC), Instituto de Salud Carlos III, Madrid, Spain.

Jordi Vila (J)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

Alex Soriano (A)

Department of Infectious Diseases, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.

María Ángeles Marcos (MÁ)

Department of Microbiology, Hospital Clinic of Barcelonagrid.410458.c, Barcelona, Spain.
Institut of Global Health of Barcelona (ISGlobal), Barcelona, Spain.

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