Biological evaluation of integrin α


Journal

European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences
ISSN: 1879-0720
Titre abrégé: Eur J Pharm Sci
Pays: Netherlands
ID NLM: 9317982

Informations de publication

Date de publication:
01 Jan 2023
Historique:
received: 11 08 2022
revised: 10 11 2022
accepted: 16 11 2022
pubmed: 21 11 2022
medline: 15 12 2022
entrez: 20 11 2022
Statut: ppublish

Résumé

Integrins are cell surface receptors involved in multiple functions vital for cellular proliferation. Various tumor cells overexpress αβ-integrins, making them ideal biomarkers for diagnostic imaging and tumor-targeted drug delivery. LXY30 is a peptide that can specifically recognize and interact with the integrin α

Identifiants

pubmed: 36403717
pii: S0928-0987(22)00221-4
doi: 10.1016/j.ejps.2022.106336
pii:
doi:

Substances chimiques

Gallium Radioisotopes 0
Integrin alpha3beta1 0
Peptides 0
Radiopharmaceuticals 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

106336

Informations de copyright

Copyright © 2022 The Authors. Published by Elsevier B.V. All rights reserved.

Auteurs

Elisavet Lambidis (E)

Department of Chemistry, Radiochemistry, University of Helsinki, Helsinki FI-00014, Finland.

Chun-Chieh Chen (CC)

Department of Molecular and Cellular Biology, University of California, Davis, CA 95616, U.S.A.

Dave Lumen (D)

Department of Chemistry, Radiochemistry, University of Helsinki, Helsinki FI-00014, Finland.

Ana Isabel Fraguas Sánchez (AIF)

Department of Chemistry, Radiochemistry, University of Helsinki, Helsinki FI-00014, Finland.

Mirkka Sarparanta (M)

Department of Chemistry, Radiochemistry, University of Helsinki, Helsinki FI-00014, Finland.

R Holland Cheng (RH)

Department of Molecular and Cellular Biology, University of California, Davis, CA 95616, U.S.A.. Electronic address: rhch@ucdavis.edu.

Anu J Airaksinen (AJ)

Department of Chemistry, Radiochemistry, University of Helsinki, Helsinki FI-00014, Finland; Turku PET Centre, Department of Chemistry, University of Turku, Turku FI-20520, Finland. Electronic address: anu.airaksinen@utu.fi.

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Classifications MeSH