Improved Subcutaneous Delivery of Ketoconazole Using EpiDerm and HSPiP Software-Based Simulations as Assessed by Cell Viability, Cellular Uptake, Permeation, and Hemolysis
Journal
ACS omega
ISSN: 2470-1343
Titre abrégé: ACS Omega
Pays: United States
ID NLM: 101691658
Informations de publication
Date de publication:
22 Nov 2022
22 Nov 2022
Historique:
received:
21
09
2022
accepted:
28
10
2022
entrez:
28
11
2022
pubmed:
29
11
2022
medline:
29
11
2022
Statut:
epublish
Résumé
Ketoconazole (KETO) is the drug of choice to control local, systemic, and resistant types of fungal infections. Subcutaneous (sub-Q) delivery offers several benefits. The present study investigated the sub-Q delivery of KETO using HSPiP software based on optimized concentrations of dimethylacetamide (DMA) in binary solvents (DMA + water),
Identifiants
pubmed: 36440147
doi: 10.1021/acsomega.2c06001
pmc: PMC9685774
doi:
Types de publication
Journal Article
Langues
eng
Pagination
42593-42606Informations de copyright
© 2022 The Authors. Published by American Chemical Society.
Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
Références
Int J Dermatol. 1995 Feb;34(2):145-6
pubmed: 7737778
Arch Drug Inf. 2011 Mar;4(1):10-21
pubmed: 21572515
Am J Hosp Pharm. 1983 Aug;40(8):1334-6
pubmed: 6310994
Mycopathologia. 2020 Aug;185(4):599-606
pubmed: 32737747
PLoS One. 2016 Mar 22;11(3):e0152074
pubmed: 27003833
Iran J Pharm Res. 2020 Summer;19(3):572-578
pubmed: 33680052
J Fungi (Basel). 2019 Mar 21;5(1):
pubmed: 30901907
J Fungi (Basel). 2018 Apr 06;4(2):
pubmed: 29642408
Adv Drug Deliv Rev. 2013 Feb;65(2):251-64
pubmed: 22626979
Int J Pharm. 2015 Jul 25;490(1-2):308-15
pubmed: 26027488
J Fungi (Basel). 2020 Nov 02;6(4):
pubmed: 33147877
Photodermatol Photoimmunol Photomed. 2011 Feb;27(1):2-9
pubmed: 21198876
Biophys J. 2009 Jan;96(1):248-54
pubmed: 18835898
Sci Rep. 2020 Jul 22;10(1):12243
pubmed: 32699361
Int J Pharm. 2011 Sep 15;416(1):202-9
pubmed: 21745557
Biomed Pap Med Fac Univ Palacky Olomouc Czech Repub. 2016 Mar;160(1):54-63
pubmed: 26006090
Drug Deliv. 2016;23(2):631-41
pubmed: 25005585
Biol Pharm Bull. 1993 Feb;16(2):188-94
pubmed: 8395931
PDA J Pharm Sci Technol. 2000 Nov-Dec;54(6):456-69
pubmed: 11107838
J Pharm Pharm Sci. 2018;21(1s):242s-253s
pubmed: 30348250
ACS Omega. 2021 Feb 11;6(7):5033-5045
pubmed: 33644612
Pharmazie. 1997 Feb;52(2):149-51
pubmed: 9122274
Acta Trop. 2018 Sep;185:69-76
pubmed: 29733808
PLoS Genet. 2014 Dec 04;10(12):e1004824
pubmed: 25474009
Am Ind Hyg Assoc J. 1988 Jun;49(6):301-8
pubmed: 2456684
Int J Pharm. 2000 Mar 30;198(1):1-6
pubmed: 10722946
Emerg Infect Dis. 2021;27(5):1266-1273
pubmed: 33755007
mBio. 2018 Oct 23;9(5):
pubmed: 30352939