Exploration of Anti-HIV Phytocompounds against SARS-CoV-2 Main Protease: Structure-Based Screening, Molecular Simulation, ADME Analysis and Conceptual DFT Studies.


Journal

Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009

Informations de publication

Date de publication:
28 Nov 2022
Historique:
received: 11 09 2022
revised: 21 10 2022
accepted: 14 11 2022
entrez: 11 12 2022
pubmed: 12 12 2022
medline: 15 12 2022
Statut: epublish

Résumé

The ever-expanding pandemic severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) infection has gained attention as COVID-19 and caused an emergency in public health to an unmatched level to date. However, the treatments used are the only options; currently, no effective and licensed medications are available to combat disease transmission, necessitating further research. In the present study, an in silico-based virtual screening of anti-HIV bioactive compounds from medicinal plants was carried out through molecular docking against the main protease (M

Identifiants

pubmed: 36500380
pii: molecules27238288
doi: 10.3390/molecules27238288
pmc: PMC9736867
pii:
doi:

Substances chimiques

3C-like proteinase, SARS-CoV-2 EC 3.4.22.-
Coronavirus 3C Proteases EC 3.4.22.28
hypericin 7V2F1075HD
pseudohypericin MQ0U4663ZO
Protease Inhibitors 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : King Khalid University
ID : R.G.P. 2/ 78/ 43

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Auteurs

Mahadevamurthy Murali (M)

Department of Studies in Botany, University of Mysore, Mysore 570006, India.

Hittanahallikoppal Gajendramurthy Gowtham (HG)

Department of PG Studies in Biotechnology, Nrupathunga University, Nrupathunga Road, Bangalore 560001, India.

Natarajamurthy Shilpa (N)

Department of Studies in Microbiology, University of Mysore, Mysore 570006, India.

Hemanth Kumar Naguvanahalli Krishnappa (HKN)

Post Graduate Department of Botany, Maharani's Science College for Women, JLB Road, Mysuru 570005, India.

Ana E Ledesma (AE)

Centro de InvestigaciónenBiofísicaAplicada y Alimentos, Facultad de Ciencias Exactas y Tecnologías (FCEyN), Universidad Nacional de Santiago del Estero (CIBAAL-UNSE-CONICET), Santiago del Estero 4206, Argentina.

Anisha S Jain (AS)

Department of Microbiology, JSS Academy of Higher Education and Research, Mysuru 570015, India.

Ali A Shati (AA)

Biology Department, Faculty of Science, King Khalid University, Abha 9004, Saudi Arabia.

Mohammad Y Alfaifi (MY)

Biology Department, Faculty of Science, King Khalid University, Abha 9004, Saudi Arabia.

Serag Eldin I Elbehairi (SEI)

Biology Department, Faculty of Science, King Khalid University, Abha 9004, Saudi Arabia.
Cell Culture Lab, Egyptian Organization for Biological Products and Vaccines (VACSERA Holding Company), 51 Wezaret El-Zeraa St., Giza 12511, Egypt.

Raghu Ram Achar (RR)

Division of Biochemistry, School of Life Sciences, JSS Academy of Higher Education and Research, Mysuru 570015, India.

Ekaterina Silina (E)

Department of Hospital Surgery, N.I. Pirogov Russian National Research Medical University, Moscow 117997, Russia.

Victor Stupin (V)

Department of Hospital Surgery, N.I. Pirogov Russian National Research Medical University, Moscow 117997, Russia.

Joaquín Ortega-Castro (J)

Departament de Química, Facultat de Ciences, Universitat de les IllesBalears, E-07122 Palma de Malllorca, Spain.

Juan Frau (J)

Departament de Química, Facultat de Ciences, Universitat de les IllesBalears, E-07122 Palma de Malllorca, Spain.

Norma Flores-Holguín (N)

Laboratorio Virtual NANOCOSMOS, Departamento de Medio Ambiente y Energía, Centro de Investigaciónen Materiales Avanzados, Chihuahua 31136, Mexico.

Kestur Nagaraj Amruthesh (KN)

Department of Studies in Botany, University of Mysore, Mysore 570006, India.

Chandan Shivamallu (C)

Department of Biotechnology and Bioinformatics, JSS Academy of Higher Education and Research, Mysuru 570015, India.

Shiva Prasad Kollur (SP)

School of Physical Sciences, Amrita Vishwa Vidyapeetham, Mysuru Campus, Mysuru 570026, India.

Daniel Glossman-Mitnik (D)

Laboratorio Virtual NANOCOSMOS, Departamento de Medio Ambiente y Energía, Centro de Investigaciónen Materiales Avanzados, Chihuahua 31136, Mexico.

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Classifications MeSH