Therapeutic targeting of eukaryotic initiation factor (eIF) 4E.


Journal

Biochemical Society transactions
ISSN: 1470-8752
Titre abrégé: Biochem Soc Trans
Pays: England
ID NLM: 7506897

Informations de publication

Date de publication:
27 02 2023
Historique:
received: 06 12 2022
revised: 06 01 2023
accepted: 10 01 2023
pubmed: 21 1 2023
medline: 3 3 2023
entrez: 20 1 2023
Statut: ppublish

Résumé

Fundamental studies unraveled the role of eukaryotic initiation factor (eIF) 4E in mRNA translation and its control. Under physiological conditions, regulation of translation by eIF4E is essential to cellular homeostasis. Under stress, gene flow information is parsed by eIF4E to support adaptive mechanisms that favor cell survival. Dysregulated eIF4E activity fuels tumor formation and progression and modulates response to therapy. Thus, there has been heightened interest in understanding eIF4E function in controlling gene expression as well as developing strategies to block its activity to treat disease.

Identifiants

pubmed: 36661272
pii: 232479
doi: 10.1042/BST20220285
doi:

Substances chimiques

Eukaryotic Initiation Factor-4E 0
Peptide Initiation Factors 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

113-124

Subventions

Organisme : CIHR
Pays : Canada

Informations de copyright

© 2023 The Author(s). Published by Portland Press Limited on behalf of the Biochemical Society.

Auteurs

Jerry Pelletier (J)

Department of Biochemistry, McGill University, Montreal, QC, Canada.
Rosalind & Morris Goodman Cancer Research Institute, McGill University, Montreal, QC, Canada.
Centre de Recherche en Biologie Structurale (CRBS), McGill University, Montreal, QC, Canada.
Department of Oncology, McGill University, Montreal, QC, Canada.
McGill Research Center on Complex Traits, McGill University, Montreal, QC, Canada.

Nahum Sonenberg (N)

Department of Biochemistry, McGill University, Montreal, QC, Canada.
Rosalind & Morris Goodman Cancer Research Institute, McGill University, Montreal, QC, Canada.
Centre de Recherche en Biologie Structurale (CRBS), McGill University, Montreal, QC, Canada.

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Classifications MeSH