Traceless Staudinger Ligation to Access Stable Aminoacyl- or Peptidyl-Dinucleotide.


Journal

ACS omega
ISSN: 2470-1343
Titre abrégé: ACS Omega
Pays: United States
ID NLM: 101691658

Informations de publication

Date de publication:
31 Jan 2023
Historique:
received: 22 09 2022
accepted: 26 10 2022
entrez: 6 2 2023
pubmed: 7 2 2023
medline: 7 2 2023
Statut: epublish

Résumé

Aminoacyl- and peptidyl-tRNA are specific biomolecules involved in many biological processes, from ribosomal protein synthesis to the synthesis of peptidoglycan precursors. Here, we report a post-synthetic approach based on traceless Staudinger ligation for the synthesis of a stable amide bond to access aminoacyl- or peptidyl-di-nucleotide. A series of amino-acid and peptide ester phenyl phosphines were synthetized, and their reactivity was studied on a 2'-N

Identifiants

pubmed: 36743074
doi: 10.1021/acsomega.2c06135
pmc: PMC9893454
doi:

Types de publication

Journal Article

Langues

eng

Pagination

3850-3860

Informations de copyright

© 2023 The Authors. Published by American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

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Auteurs

Camélia Kitoun (C)

Université Paris Cité, CNRS, Laboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques, Paris F-75006, France.

Saidbakhrom Saidjalolov (S)

Université Paris Cité, CNRS, Laboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques, Paris F-75006, France.

Delphine Bouquet (D)

Université Paris Cité, CNRS, Laboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques, Paris F-75006, France.

Fabiola Djago (F)

Institut de Chimie des Milieux et Matériaux de Poitiers IC2MP, Université de Poitiers, UMR 7285, Poitiers 86073, France.

Quentin Blancart Remaury (QB)

Institut de Chimie des Milieux et Matériaux de Poitiers IC2MP, Université de Poitiers, UMR 7285, Poitiers 86073, France.

Bruno Sargueil (B)

Université Paris Cité, CNRS, UMR 8038/CiTCoM, Paris F-75006, France.

Pauline Poinot (P)

Institut de Chimie des Milieux et Matériaux de Poitiers IC2MP, Université de Poitiers, UMR 7285, Poitiers 86073, France.

Mélanie Etheve-Quelquejeu (M)

Université Paris Cité, CNRS, Laboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques, Paris F-75006, France.

Laura Iannazzo (L)

Université Paris Cité, CNRS, Laboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques, Paris F-75006, France.

Classifications MeSH