Enantioselective Au-Catalyzed Synthesis of Thia[5]- and Thia[6]helicenes and Their Transformation into Bowl-shaped Pleiadenes.

Au-catalysis alkyne hydroarylation asymmetric catalysis bowl-shaped molecules thiahelicenes

Journal

Advanced materials (Deerfield Beach, Fla.)
ISSN: 1521-4095
Titre abrégé: Adv Mater
Pays: Germany
ID NLM: 9885358

Informations de publication

Date de publication:
Apr 2023
Historique:
revised: 17 01 2023
received: 02 12 2022
medline: 8 2 2023
pubmed: 8 2 2023
entrez: 7 2 2023
Statut: ppublish

Résumé

A series of helically shaped benzo[b]chryseno[4,3-d]thiophenes, naphtho[1,2-b]phenanthro[4,3-d]thiophenes, and chryseno[3,4-b]naphtho[1,2-d]thiophenes is synthesized via a highly enantioselective Au-catalyzed intramolecular alkyne hydroarylation reaction. The inversion barriers of the structures obtained are determined both theoretically and experimentally, and their chiroptical properties are reported. Preliminary studies on the post-synthetic functionalization of these thiahelicenes and their transformation into azahelicenes are also presented. In addition, a straightforward one-step protocol is developed, which wraps the initially obtained chryseno[3,4-b]naphtho[1,2-d]thiophenes into bowl-shaped pleiadene derivatives without erosion of the enantiopurity. The number of structurally related products that are obtained with high enantioselectivity enables the establishment of comprehensive correlations between the structure and conformational stability or (chir)optical properties.

Identifiants

pubmed: 36747350
doi: 10.1002/adma.202211279
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

e2211279

Subventions

Organisme : Deutsche Forschungsgemeinschaft
ID : INST 186/1352-1
Organisme : Deutsche Forschungsgemeinschaft
ID : INST 186/1237-1
Organisme : China Scholarship Council

Informations de copyright

© 2023 The Authors. Advanced Materials published by Wiley-VCH GmbH.

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Auteurs

Wei Fu (W)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Valentina Pelliccioli (V)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Moritz von Geyso (M)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Pablo Redero (P)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Christian Böhmer (C)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Martin Simon (M)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Christopher Golz (C)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Manuel Alcarazo (M)

Institut für Organische und Biomolekulare Chemie, Georg-August-Universität Göttingen, Tammannstr 2, 37077, Göttingen, Germany.

Classifications MeSH