Controlled release of enhanced cross-hybrid IgGA Fc PD-L1 inhibitors using oncolytic adenoviruses.

Fc engineering IgA IgG PD-L1 therapy oncolytic adenoviruses

Journal

Molecular therapy oncolytics
ISSN: 2372-7705
Titre abrégé: Mol Ther Oncolytics
Pays: United States
ID NLM: 101666776

Informations de publication

Date de publication:
16 Mar 2023
Historique:
received: 31 08 2022
accepted: 31 01 2023
entrez: 13 3 2023
pubmed: 14 3 2023
medline: 14 3 2023
Statut: epublish

Résumé

Immune checkpoint inhibitors have clinical success in prolonging the life of many cancer patients. However, only a minority of patients benefit from such therapy, calling for further improvements. Currently, most PD-L1 checkpoint inhibitors in the clinic do not elicit Fc effector mechanisms that would substantially increase their efficacy. To gain potency and circumvent off-target effects, we previously designed an oncolytic adenovirus (Ad-Cab) expressing an Fc fusion peptide against PD-L1 on a cross-hybrid immunoglobulin GA (IgGA) Fc. Ad-Cab elicited antibody effector mechanisms of IgG1 and IgA, which led to higher tumor killing compared with each isotype alone and with clinically approved PD-L1 checkpoint inhibitors. In this study, we further improved the therapy to increase the IgG1 Fc effector mechanisms of the IgGA Fc fusion peptide (Ad-Cab FT) by adding four somatic mutations that increase natural killer (NK) cell activation. Ad-Cab FT was shown to work better at lower concentrations compared with Ad-Cab

Identifiants

pubmed: 36911070
doi: 10.1016/j.omto.2023.01.006
pii: S2372-7705(23)00008-6
pmc: PMC9995465
doi:

Types de publication

Journal Article

Langues

eng

Pagination

264-276

Informations de copyright

© 2023.

Déclaration de conflit d'intérêts

V.C. is a co-founder and shareholder of Valo Therapeutics LTD (not related to this study).

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Auteurs

Firas Hamdan (F)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Michaela Feodoroff (M)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Institute for Molecular Medicine Finland (FIMM), Helsinki Institute of Life Science (HiLIFE), University of Helsinki, Helsinki, Finland.
iCAN Digital Precision Cancer Medicine Flagship, University of Helsinki, Helsinki, Finland.

Salvatore Russo (S)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Manlio Fusciello (M)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Sara Feola (S)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Jacopo Chiaro (J)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Gabriella Antignani (G)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Francesca Greco (F)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Jeanette Leusen (J)

Center for Translational Immunology, University Medical Center Utrecht, Utrecht, the Netherlands.

Erkko Ylösmäki (E)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.

Mikaela Grönholm (M)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
iCAN Digital Precision Cancer Medicine Flagship, University of Helsinki, Helsinki, Finland.

Vincenzo Cerullo (V)

Laboratory of Immunovirotherapy, Drug Research Program, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
Translational Immunology Research Program (TRIMM), University of Helsinki, Helsinki, Finland.
Drug Delivery, Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, Helsinki, Finland.
iCAN Digital Precision Cancer Medicine Flagship, University of Helsinki, Helsinki, Finland.
Department of Molecular Medicine and Medical Biotechnology and CEINGE, Naples University Federico II, Naples, Italy.

Classifications MeSH