Unraveling the Reaction Mechanism of Russell's Viper Venom Factor X Activator: A Paradigm for the Reactivity of Zinc Metalloproteinases?


Journal

Journal of chemical information and modeling
ISSN: 1549-960X
Titre abrégé: J Chem Inf Model
Pays: United States
ID NLM: 101230060

Informations de publication

Date de publication:
10 07 2023
Historique:
medline: 11 7 2023
pubmed: 24 4 2023
entrez: 24 04 2023
Statut: ppublish

Résumé

Snake venom metalloproteinases (SVMPs) are important drug targets against snakebite envenoming, the neglected tropical disease with the highest mortality worldwide. Here, we focus on Russell's viper (

Identifiants

pubmed: 37092784
doi: 10.1021/acs.jcim.2c01156
pmc: PMC10336966
doi:

Substances chimiques

russellysin EC 3.4.24.58
Antivenins 0
Zinc J41CSQ7QDS
cancer procoagulant EC 3.4.22.26
Viper Venoms 0
Metalloproteases EC 3.4.-

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

4056-4069

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Auteurs

Juliana Castro-Amorim (J)

LAQV, REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, Rua do Campo Alegre, s/n, Porto 4169-007, Portugal.

Ana Oliveira (A)

LAQV, REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, Rua do Campo Alegre, s/n, Porto 4169-007, Portugal.

Ashis K Mukherjee (AK)

Institute of Advanced Study in Science and Technology, Vigyan Path Garchuk, Paschim Boragaon, Guwahati 781035, Assam, India.

Maria J Ramos (MJ)

LAQV, REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, Rua do Campo Alegre, s/n, Porto 4169-007, Portugal.

Pedro A Fernandes (PA)

LAQV, REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, Rua do Campo Alegre, s/n, Porto 4169-007, Portugal.

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Classifications MeSH