225Ac–DOTATATE
actinium-225
neuroendocrine tumors
radiobiology
radiolabeling
radionuclide production
radiopharmaceuticals
targeted alpha-therapy
targeted radionuclide therapy
Journal
Pharmaceutics
ISSN: 1999-4923
Titre abrégé: Pharmaceutics
Pays: Switzerland
ID NLM: 101534003
Informations de publication
Date de publication:
24 Mar 2023
24 Mar 2023
Historique:
received:
14
02
2023
revised:
18
03
2023
accepted:
22
03
2023
medline:
28
4
2023
pubmed:
28
4
2023
entrez:
28
4
2023
Statut:
epublish
Résumé
The widespread use of peptide receptor radionuclide therapy (PRRT) represents a major therapeutic breakthrough in nuclear medicine, particularly since the introduction of
Identifiants
pubmed: 37111537
pii: pharmaceutics15041051
doi: 10.3390/pharmaceutics15041051
pmc: PMC10146019
pii:
doi:
Types de publication
Journal Article
Review
Langues
eng
Références
Mol Pharm. 2018 Apr 2;15(4):1457-1466
pubmed: 29502411
Pharmaceuticals (Basel). 2021 Jul 06;14(7):
pubmed: 34358076
J Nucl Med. 2004 Jan;45(1):129-37
pubmed: 14734685
Nucl Med Biol. 2022 Sep-Oct;112-113:35-43
pubmed: 35797877
J Clin Endocrinol Metab. 2019 Apr 1;104(4):1336-1344
pubmed: 30566620
Lancet Reg Health Eur. 2022 Sep 23;23:100510
pubmed: 36176500
Clin Nucl Med. 2017 Jun;42(6):436-443
pubmed: 28263217
Cancer Biother Radiopharm. 2022 Jun;37(5):355-363
pubmed: 35695807
Eur J Nucl Med Mol Imaging. 2014 Feb;41(2):205-10
pubmed: 24030668
Theranostics. 2016 Mar 01;6(5):698-709
pubmed: 27022417
Eur J Nucl Med Mol Imaging. 2016 Jun;43(6):1040-6
pubmed: 26611427
Anticancer Res. 2004 Jan-Feb;24(1):101-5
pubmed: 15015582
Dev Neurobiol. 2012 Sep;72(9):1181-95
pubmed: 21976424
J Nucl Med. 2005 Jan;46 Suppl 1:99S-106S
pubmed: 15653658
J Clin Oncol. 2018 Sep 1;36(25):2578-2584
pubmed: 29878866
N Engl J Med. 2013 Jul 18;369(3):213-23
pubmed: 23863050
EJNMMI Phys. 2021 Aug 18;8(1):60
pubmed: 34406515
J Nucl Med. 2011 Jul;52(7):1041-7
pubmed: 21680680
Digestion. 1996;57 Suppl 1:57-61
pubmed: 8813472
J Nucl Med. 2011 Sep;52(9):1361-8
pubmed: 21795361
Eur J Nucl Med Mol Imaging. 2014 Nov;41(11):2106-19
pubmed: 25070685
Bioconjug Chem. 2021 Jul 21;32(7):1348-1363
pubmed: 32216377
J Clin Oncol. 2008 Jun 20;26(18):3063-72
pubmed: 18565894
Eur J Nucl Med Mol Imaging. 2021 Oct;48(11):3408-3421
pubmed: 33772332
Clin Gastroenterol Hepatol. 2019 Oct;17(11):2212-2217.e1
pubmed: 30580091
Curr Radiopharm. 2018;11(3):200-208
pubmed: 29732998
Eur J Nucl Med Mol Imaging. 2020 Apr;47(4):934-946
pubmed: 31707430
Nucl Med Biol. 2007 Feb;34(2):185-93
pubmed: 17307126
Eur J Nucl Med Mol Imaging. 2022 Apr;49(5):1595-1606
pubmed: 34837103
Eur J Nucl Med Mol Imaging. 2017 Mar;44(3):490-499
pubmed: 27704193
Pharmaceuticals (Basel). 2014 Mar 13;7(3):353-65
pubmed: 24633429
Phys Med Biol. 2021 Jan 29;66(3):035016
pubmed: 33321484
PLoS One. 2013 Apr 22;8(4):e62487
pubmed: 23614051
J Clin Oncol. 2010 Apr 1;28(10):1652-9
pubmed: 20194865
Nucl Med Rev Cent East Eur. 2016;19(2):111-7
pubmed: 27479788
J Clin Oncol. 2008 May 1;26(13):2124-30
pubmed: 18445841
Angew Chem Int Ed Engl. 2017 Nov 13;56(46):14712-14717
pubmed: 28963750
Cancer Discov. 2018 Apr;8(4):OF2
pubmed: 29487054
Bioconjug Chem. 2022 Dec 21;33(12):2381-2397
pubmed: 36378809
Eur J Nucl Med Mol Imaging. 2022 Feb;49(3):871-880
pubmed: 34537893
J Clin Oncol. 2011 Jun 10;29(17):2416-23
pubmed: 21555692
Eur J Nucl Med Mol Imaging. 2007 Feb;34(2):219-27
pubmed: 17021812
Br J Radiol. 2018 Nov;91(1091):20180041
pubmed: 29513039
Eur J Nucl Med. 2000 Mar;27(3):273-82
pubmed: 10774879
Pol Arch Intern Med. 2022 Aug 22;132(7-8):
pubmed: 35699734
J Chromatogr A. 2015 Feb 6;1380:55-63
pubmed: 25596759
Cancer Biother Radiopharm. 2000 Jun;15(3):235-44
pubmed: 10941530
Clin Cancer Res. 2008 Jun 1;14(11):3555-61
pubmed: 18519789
Ann N Y Acad Sci. 1994 Sep 15;733:496-506
pubmed: 7978900
Life Sci. 1982 Sep 13;31(11):1133-40
pubmed: 6128648
Q J Nucl Med Mol Imaging. 2020 Sep;64(3):265-277
pubmed: 32441067
Bioconjug Chem. 2022 Oct 19;33(10):1900-1921
pubmed: 36126334
Front Med (Lausanne). 2022 Dec 07;9:1034315
pubmed: 36569154
Chem Biol Drug Des. 2018 Jul;92(1):1344-1356
pubmed: 29611298
Sci Rep. 2017 Aug 15;7(1):8216
pubmed: 28811573
Oncoimmunology. 2019 May 1;8(8):1607673
pubmed: 31413916
Mol Pharm. 2019 Dec 2;16(12):4807-4816
pubmed: 31518138
Eur J Nucl Med Mol Imaging. 2011 Dec;38(12):2125-35
pubmed: 21892623
Front Med (Lausanne). 2015 Mar 17;2:12
pubmed: 25853132
Appl Radiat Isot. 2002 Dec;57(6):841-7
pubmed: 12406626
Appl Radiat Isot. 2005 Mar;62(3):383-7
pubmed: 15607913
Pharmaceutics. 2021 Jun 18;13(6):
pubmed: 34207408
Nucl Med Biol. 2022 Jul-Aug;110-111:28-36
pubmed: 35512517
Neuroendocrinology. 2019;108(3):256-264
pubmed: 30352433
Molecules. 2019 Sep 19;24(18):
pubmed: 31546752
Eur J Nucl Med Mol Imaging. 2021 Jan;48(1):152-160
pubmed: 32472437
Ann N Y Acad Sci. 2004 Apr;1014:234-45
pubmed: 15153440
Appl Radiat Isot. 2018 Oct;140:18-23
pubmed: 29936271
Clin Cancer Res. 2006 Feb 1;12(3 Pt 1):897-903
pubmed: 16467104
Cancer Res. 2005 Jun 1;65(11):4888-95
pubmed: 15930310
J Nucl Med. 2020 Apr;61(4):563-569
pubmed: 31586001
J Nucl Med. 2020 Jan;61(1):62-69
pubmed: 31101746
Pharmaceuticals (Basel). 2022 Sep 21;15(10):
pubmed: 36297279
EJNMMI Radiopharm Chem. 2022 Oct 23;7(1):28
pubmed: 36274098
Pharmacol Ther. 2015 Aug;152:98-110
pubmed: 25956467
Eur J Nucl Med Mol Imaging. 2014 Jun;41(6):1141-57
pubmed: 24668274
Pharmaceutics. 2021 May 13;13(5):
pubmed: 34068206
Endocrinol Metab Clin North Am. 2018 Sep;47(3):615-625
pubmed: 30098719
Front Oncol. 2022 Nov 24;12:993182
pubmed: 36505778
Front Oncol. 2020 Nov 05;10:531660
pubmed: 33251129
Clin Cancer Res. 2017 Aug 15;23(16):4617-4624
pubmed: 28428192
Eur J Nucl Med Mol Imaging. 2015 Jul;42(8):1238-46
pubmed: 25808630
Appl Radiat Isot. 2019 Nov;153:108816
pubmed: 31344650
Nucl Med Biol. 1999 Jul;26(5):581-9
pubmed: 10473198
Curr Radiopharm. 2018;11(3):180-191
pubmed: 29766832
Neuroendocrinology. 2012;95(2):157-76
pubmed: 22262022
Inorg Chem. 2022 Aug 15;61(32):12847-12855
pubmed: 35914099
Eur J Nucl Med Mol Imaging. 2018 Jun;45(6):970-988
pubmed: 29497803
Lancet Oncol. 2021 Dec;22(12):1752-1763
pubmed: 34793718
J Am Chem Soc. 2021 Jul 14;143(27):10429-10440
pubmed: 34190542
Neuroendocrinology. 2016;103(2):172-85
pubmed: 26731013
Eur J Nucl Med Mol Imaging. 2012 Feb;39 Suppl 1:S103-12
pubmed: 22388631
Inorg Chem. 2020 Sep 8;59(17):12156-12165
pubmed: 32677829
Neuroendocrinology. 2004;80 Suppl 1:3-7
pubmed: 15477707
Clin Nucl Med. 2020 Mar;45(3):241-243
pubmed: 31977472
Eur J Nucl Med. 2001 Sep;28(9):1319-25
pubmed: 11585290
J Pediatr Hematol Oncol. 2016 Mar;38(2):87-96
pubmed: 26296147
EJNMMI Res. 2016 Dec;6(1):83
pubmed: 27873240
Int J Cancer. 1997 Mar 4;70(5):530-7
pubmed: 9052751
J Nucl Med. 2017 Oct;58(10):1624-1631
pubmed: 28408529
Eur J Nucl Med. 2001 Jul;28(7):836-46
pubmed: 11504080
Pharmaceutics. 2021 Oct 16;13(10):
pubmed: 34683999
J Nucl Med. 2012 Dec;53(12):1951-9
pubmed: 23139086
EJNMMI Radiopharm Chem. 2022 Sep 6;7(1):23
pubmed: 36068452
ACS Omega. 2020 Oct 06;5(41):26431-26440
pubmed: 33110971
Eur J Nucl Med Mol Imaging. 2019 Jan;46(1):129-138
pubmed: 30232539
BMC Cancer. 2019 Aug 8;19(1):788
pubmed: 31395036
Semin Nucl Med. 2006 Apr;36(2):147-56
pubmed: 16517236
J Nucl Med. 2021 Jul 1;62(7):1012-1015
pubmed: 33127622
J Nucl Med. 2023 Feb;64(2):219-220
pubmed: 36265909
Eur J Nucl Med Mol Imaging. 2019 Mar;46(3):728-742
pubmed: 30506283
Neuroendocrinology. 2021;111(4):330-343
pubmed: 32097917
Anal Chem. 2005 Oct 1;77(19):6288-91
pubmed: 16194090
J Nucl Med. 2014 Feb;55(2):183-90
pubmed: 24434296
Bioconjug Chem. 2000 Jul-Aug;11(4):510-9
pubmed: 10898572
EJNMMI Radiopharm Chem. 2021 Dec 20;6(1):38
pubmed: 34928478
Indian J Nucl Med. 2020 Jul-Sep;35(3):226-228
pubmed: 33082679
Cancer Biother Radiopharm. 2018 Oct;33(8):336-348
pubmed: 29889562
Pharmaceutics. 2021 Sep 13;13(9):
pubmed: 34575538
Crit Rev Oncol Hematol. 2018 Mar;123:7-20
pubmed: 29482781
Nucleosides Nucleotides Nucleic Acids. 2020;39(1-3):439-452
pubmed: 31560250
Curr Radiopharm. 2018;11(3):156-172
pubmed: 29658444
J Nucl Med. 2023 Apr;64(4):549-554
pubmed: 36396453
Eur J Nucl Med Mol Imaging. 2017 Jul;44(7):1207-1214
pubmed: 28246882
Semin Nucl Med. 2019 Sep;49(5):422-437
pubmed: 31470935
Eur J Nucl Med Mol Imaging. 2021 Dec;49(1):54-63
pubmed: 34448031
N Engl J Med. 2017 Jan 12;376(2):125-135
pubmed: 28076709
Nature. 1979 Aug 9;280(5722):512-4
pubmed: 460433
EJNMMI Phys. 2021 Jan 12;8(1):4
pubmed: 33432383
Eur J Nucl Med Mol Imaging. 2019 Mar;46(3):704-717
pubmed: 30267116
J Nucl Med. 2011 Dec;52 Suppl 2:56S-63S
pubmed: 22144556
Eur J Nucl Med Mol Imaging. 2021 Dec;49(1):279-289
pubmed: 34196752
Theranostics. 2016 Feb 13;6(4):501-10
pubmed: 26941843
Curr Radiopharm. 2018;11(3):173-179
pubmed: 29669509
Proc Natl Acad Sci U S A. 1982 Aug;79(15):4575-9
pubmed: 6126875
Cancer Biother Radiopharm. 2002 Apr;17(2):219-31
pubmed: 12030116
Clin Cancer Res. 2022 May 13;28(10):2030-2037
pubmed: 35247915
Semin Nucl Med. 2002 Apr;32(2):110-22
pubmed: 11965606
J Nucl Med. 2014 Sep;55(9):1492-8
pubmed: 24982438
Cancer Med. 2021 Feb;10(3):1128-1140
pubmed: 33347715
Eur J Nucl Med Mol Imaging. 2020 Mar;47(3):721-728
pubmed: 31758224
Clin Cancer Res. 2019 Jan 15;25(2):868-880
pubmed: 30352909
Endocr Relat Cancer. 2010 Jan 29;17(1):R75-90
pubmed: 20008097
Bioconjug Chem. 2022 Jun 15;33(6):1222-1231
pubmed: 35670495
Eur J Nucl Med Mol Imaging. 2020 Oct;47(11):2711-2712
pubmed: 32123970
EJNMMI Res. 2016 Dec;6(1):6
pubmed: 26791386
Appl Radiat Isot. 2021 Jun;172:109676
pubmed: 33725503
J Nucl Med. 2022 Apr;63(4):584-590
pubmed: 34385334
Endocr Rev. 2003 Aug;24(4):389-427
pubmed: 12920149
Appl Radiat Isot. 2005 May;62(5):667-79
pubmed: 15763472
Endocr Rev. 2004 Jun;25(3):458-511
pubmed: 15180952
Chem Commun (Camb). 2018 Mar 8;54(21):2599-2602
pubmed: 29388990
Chemistry. 2020 Sep 4;26(50):11435-11440
pubmed: 32588455
AJR Am J Roentgenol. 2018 Aug;211(2):278-285
pubmed: 29949416
J Nucl Med. 2018 May;59(5):795-802
pubmed: 29326358
Phys Med Biol. 2011 Feb 7;56(3):721-33
pubmed: 21220845
Appl Radiat Isot. 2012 Nov;70(11):2602-7
pubmed: 22940414
PLoS One. 2014 Feb 07;9(2):e88239
pubmed: 24516620
Theranostics. 2020 May 25;10(15):6946-6958
pubmed: 32550914
Eur J Nucl Med. 2001 Oct;28(10):1552-4
pubmed: 11685499
Theranostics. 2020 Jul 23;10(20):9364-9377
pubmed: 32802197
J Nucl Med. 2022 Jul 21;:
pubmed: 35863893
Biochem Biophys Res Commun. 1980 Sep 30;96(2):725-34
pubmed: 6107078
Molecules. 2018 Mar 05;23(3):
pubmed: 29510568
Eur J Nucl Med Mol Imaging. 2022 Aug;49(10):3596-3597
pubmed: 35522323
Bioconjug Chem. 2006 Nov-Dec;17(6):1551-60
pubmed: 17105236
Eur J Nucl Med Mol Imaging. 2010 Jul;37(7):1441-8
pubmed: 20461371
Sci Rep. 2019 Aug 12;9(1):11671
pubmed: 31406320
Cancer. 2015 Feb 15;121(4):589-97
pubmed: 25312765
Cancers (Basel). 2020 Apr 21;12(4):
pubmed: 32326199
Cancers (Basel). 2021 Apr 20;13(8):
pubmed: 33923965
Theranostics. 2020 Sep 14;10(25):11359-11375
pubmed: 33052220
Inorg Chem. 2021 Mar 15;60(6):4076-4092
pubmed: 33635057
Indian J Nucl Med. 2021 Apr-Jun;36(2):114-119
pubmed: 34385780
Front Oncol. 2022 Feb 03;12:796657
pubmed: 35186737
J Nucl Med. 2016 Dec;57(12):1941-1944
pubmed: 27390158
Mol Imaging Radionucl Ther. 2022 Jun 27;31(2):139-141
pubmed: 35771003
JAMA Oncol. 2017 Oct 01;3(10):1335-1342
pubmed: 28448665
Eur J Nucl Med Mol Imaging. 2014 May;41(5):925-33
pubmed: 24504504
J Nucl Med. 2005 Jan;46 Suppl 1:83S-91S
pubmed: 15653656
Cancer Med. 2017 Nov;6(11):2745-2756
pubmed: 28980417
Phys Med Biol. 2017 Jun 7;62(11):4406-4420
pubmed: 28362640
Appl Radiat Isot. 2012 Nov;70(11):2590-5
pubmed: 22944532
Nature. 1981 Jul 2;292(5818):55-8
pubmed: 6116194
Eur J Nucl Med Mol Imaging. 2014 Oct;41(10):1845-51
pubmed: 24615468
J Med Chem. 2002 Jan 17;45(2):469-77
pubmed: 11784151
J Med Chem. 1999 Jul 29;42(15):2988-92
pubmed: 10425108
Inorg Chem. 2022 Jan 17;61(2):801-806
pubmed: 34965102
BMC Cancer. 2022 Dec 22;22(1):1346
pubmed: 36550428
Appl Radiat Isot. 2013 Jun;76:38-45
pubmed: 23084477
J Nucl Med. 2022 Feb;63(2):218-225
pubmed: 34049983
Neuroendocrinology. 2013;97(4):347-54
pubmed: 23392072
EJNMMI Radiopharm Chem. 2019 Aug 6;4(1):21
pubmed: 31659557
Ann Oncol. 1999;10 Suppl 2:S23-9
pubmed: 10399029
Clin Nucl Med. 2022 Feb 1;47(2):e156-e157
pubmed: 34284478
Appl Radiat Isot. 2016 Dec;118:366-374
pubmed: 27776333
J Am Chem Soc. 2019 Dec 11;141(49):19404-19414
pubmed: 31794205
Clin Nucl Med. 2022 Feb 1;47(2):e184-e186
pubmed: 34507333
Appl Radiat Isot. 2020 Oct;164:109262
pubmed: 32819503
Cancers (Basel). 2022 Sep 29;14(19):
pubmed: 36230691
Endocr Relat Cancer. 2016 Aug;23(8):587-94
pubmed: 27492634