Innate immune pathway modulator screen identifies STING pathway activation as a strategy to inhibit multiple families of arbo and respiratory viruses.

Chikungunya virus SARS-CoV-2 West Nile virus Zika virus cAIMP cGAS-STING pathway enterovirus-D68 pattern-recognition receptors respiratory syncytial virus scleroglucan

Journal

Cell reports. Medicine
ISSN: 2666-3791
Titre abrégé: Cell Rep Med
Pays: United States
ID NLM: 101766894

Informations de publication

Date de publication:
16 05 2023
Historique:
received: 28 01 2023
revised: 17 03 2023
accepted: 07 04 2023
medline: 19 5 2023
pubmed: 30 4 2023
entrez: 29 4 2023
Statut: ppublish

Résumé

RNA viruses continue to remain a threat for potential pandemics due to their rapid evolution. Potentiating host antiviral pathways to prevent or limit viral infections is a promising strategy. Thus, by testing a library of innate immune agonists targeting pathogen recognition receptors, we observe that Toll-like receptor 3 (TLR3), stimulator of interferon genes (STING), TLR8, and Dectin-1 ligands inhibit arboviruses, Chikungunya virus (CHIKV), West Nile virus, and Zika virus to varying degrees. STING agonists (cAIMP, diABZI, and 2',3'-cGAMP) and Dectin-1 agonist scleroglucan demonstrate the most potent, broad-spectrum antiviral function. Furthermore, STING agonists inhibit severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) and enterovirus-D68 (EV-D68) infection in cardiomyocytes. Transcriptome analysis reveals that cAIMP treatment rescue cells from CHIKV-induced dysregulation of cell repair, immune, and metabolic pathways. In addition, cAIMP provides protection against CHIKV in a chronic CHIKV-arthritis mouse model. Our study describes innate immune signaling circuits crucial for RNA virus replication and identifies broad-spectrum antivirals effective against multiple families of pandemic potential RNA viruses.

Identifiants

pubmed: 37119814
pii: S2666-3791(23)00134-9
doi: 10.1016/j.xcrm.2023.101024
pmc: PMC10213809
pii:
doi:

Substances chimiques

Antiviral Agents 0

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

101024

Subventions

Organisme : NIAID NIH HHS
ID : R01 AI163216
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK132735
Pays : United States
Organisme : NEI NIH HHS
ID : R01 EY032149
Pays : United States

Commentaires et corrections

Type : UpdateOf

Informations de copyright

Copyright © 2023 The Authors. Published by Elsevier Inc. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of interests The authors declare no competing interests.

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Auteurs

Gustavo Garcia (G)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Joseph Ignatius Irudayam (JI)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Arjit Vijey Jeyachandran (AV)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Swati Dubey (S)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Christina Chang (C)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Sebastian Castillo Cario (S)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Nate Price (N)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Sathya Arumugam (S)

Department of Mathematics, Government College Daman, Daman, Dadra and Nagar Haveli and Daman and Diu 396210, India.

Angelica L Marquez (AL)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Aayushi Shah (A)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Amir Fanaei (A)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA.

Nikhil Chakravarty (N)

Department of Epidemiology, University of California, Los Angeles, Los Angeles, CA, USA.

Shantanu Joshi (S)

Department of Neurology, University of California, Los Angeles, Los Angeles, CA, USA; Department of Bioengineering, University of California, Los Angeles, Los Angeles, CA, USA.

Sanjeev Sinha (S)

All India Institute of Medical Sciences, New Delhi, India.

Samuel W French (SW)

Department of Pathology and Laboratory Medicine, University of California, Los Angeles, Los Angeles, CA, USA; Jonsson Comprehensive Cancer Center, University of California, Los Angeles, Los Angeles, CA 90095, USA.

Mark S Parcells (MS)

Department of Animal and Food Sciences, Department of Biological Sciences, University of Delaware, Newark, DE 19716, USA.

Arunachalam Ramaiah (A)

Tata Institute for Genetics and Society, Center at inStem, Bangalore 560065, India; City of Milwaukee Health Department, Milwaukee, WI 53202, USA. Electronic address: arama@milwaukee.gov.

Vaithilingaraja Arumugaswami (V)

Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA, USA; Eli and Edythe Broad Center of Regenerative Medicine and Stem Cell Research, University of California, Los Angeles, Los Angeles, CA, USA; California NanoSystems Institute, University of California, Los Angeles, Los Angeles, CA, USA. Electronic address: varumugaswami@mednet.ucla.edu.

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