Guanidines: Synthesis of Novel Histamine H

antagonist breast cancer guanidines histamine H3 receptor multi-target directed ligand

Journal

Pharmaceuticals (Basel, Switzerland)
ISSN: 1424-8247
Titre abrégé: Pharmaceuticals (Basel)
Pays: Switzerland
ID NLM: 101238453

Informations de publication

Date de publication:
30 Apr 2023
Historique:
received: 10 04 2023
revised: 27 04 2023
accepted: 28 04 2023
medline: 27 5 2023
pubmed: 27 5 2023
entrez: 27 5 2023
Statut: epublish

Résumé

This study examines the properties of novel guanidines, designed and synthesized as histamine H

Identifiants

pubmed: 37242458
pii: ph16050675
doi: 10.3390/ph16050675
pmc: PMC10223552
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Medical Univeristy of Lodz
ID : 503/3-016-01/503-31-001-19-00
Organisme : Medical University of Lublin
ID : DS37
Organisme : Polish Smart Growth Operational Programme POIR 4.2
ID : POIR.04.02.00-00-D023/20

Références

Bioorg Med Chem Lett. 2001 Apr 9;11(7):951-4
pubmed: 11294398
Cancer Biol Ther. 2008 Jan;7(1):28-35
pubmed: 17932461
PLoS One. 2017 Oct 5;12(10):e0186108
pubmed: 28982153
ACS Chem Neurosci. 2018 May 16;9(5):1195-1214
pubmed: 29384656
Int J Mol Sci. 2018 Apr 19;19(4):
pubmed: 29671795
Bioorg Med Chem Lett. 2013 Dec 1;23(23):6415-20
pubmed: 24140447
J Pharmacol Sci. 2005 Jan;97(1):116-23
pubmed: 15655289
Inflamm Res. 2001 Apr;50 Suppl 2:S102-3
pubmed: 11411574
Curr Med Chem. 2015;22(3):373-404
pubmed: 25386820
Biochem Pharmacol. 1973 Dec 1;22(23):3099-108
pubmed: 4202581
Naunyn Schmiedebergs Arch Pharmacol. 1999 Nov;360(5):552-7
pubmed: 10598794
Molecules. 2019 Dec 06;24(24):
pubmed: 31817628
Arch Pharm (Weinheim). 2012 Aug;345(8):591-7
pubmed: 22549828
Neurology. 2010 Oct 19;75(16):1472-9
pubmed: 20956793
ACS Chem Neurosci. 2014 Mar 19;5(3):225-42
pubmed: 24422467
ACS Chem Neurosci. 2021 Jul 7;12(13):2503-2519
pubmed: 34100603
J Med Chem. 2011 Jan 13;54(1):26-53
pubmed: 21062081
Front Neurosci. 2016 May 30;10:201
pubmed: 27303254
Inflamm Allergy Drug Targets. 2010 Jul;9(3):146-57
pubmed: 20632959
Methods Find Exp Clin Pharmacol. 1992 Dec;14(10):747-51
pubmed: 1338472
Cancer Biol Ther. 2006 Nov;5(11):1462-71
pubmed: 17012845
Semin Cancer Biol. 2000 Feb;10(1):15-23
pubmed: 10888267
Arch Pharm (Weinheim). 2012 Jun;345(6):431-43
pubmed: 22415744
Leuk Lymphoma. 2000 Jan;36(3-4):367-73
pubmed: 10674909
Bioorg Med Chem Lett. 2020 Nov 15;30(22):127522
pubmed: 32871268
Biochem Pharmacol. 1961 Jul;7:88-95
pubmed: 13726518
ACS Chem Neurosci. 2015 Mar 18;6(3):438-45
pubmed: 25588572
Nat Commun. 2022 Oct 15;13(1):6105
pubmed: 36243875
Eur J Pharmacol. 2011 Mar 11;654(3):200-8
pubmed: 21237145
J Chem Inf Model. 2015 Jan 26;55(1):149-64
pubmed: 25531792
J Pharmacol Exp Ther. 2008 Aug;326(2):406-13
pubmed: 18474684
Oncotarget. 2015 Jul 10;6(19):17107-20
pubmed: 25940798
Biochem Biophys Res Commun. 2016 Nov 18;480(3):479-485
pubmed: 27773822
Br J Pharmacol Chemother. 1959 Mar;14(1):48-58
pubmed: 13651579
J Cell Biol. 1990 Apr;110(4):1211-5
pubmed: 2182646
Inflamm Res. 2009 Apr;58 Suppl 1:55-6
pubmed: 19274436
Cancer Res. 1984 Feb;44(2):639-45
pubmed: 6692368

Auteurs

Marek Staszewski (M)

Department of Synthesis and Technology of Drugs, Medical University of Lodz, Muszyńskiego 1, 90-151 Łódź, Poland.

Magdalena Iwan (M)

Department of Toxicology, Medical University of Lublin, Chodźki 8, 20-093 Lublin, Poland.

Tobias Werner (T)

Institute of Pharmaceutical and Medicinal Chemistry, Heinrich Heine University Düsseldorf, Universitaetsstr. 1, 40225 Duesseldorf, Germany.

Marek Bajda (M)

Department of Physicochemical Drug Analysis, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.

Justyna Godyń (J)

Department of Physicochemical Drug Analysis, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.

Gniewomir Latacz (G)

Department of Technology and Biotechnology of Drugs, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.

Agnieszka Korga-Plewko (A)

Independent Medical Biology Unit, Medical University of Lublin, Jaczewskiego 8b, 20-090 Lublin, Poland.

Joanna Kubik (J)

Independent Medical Biology Unit, Medical University of Lublin, Jaczewskiego 8b, 20-090 Lublin, Poland.

Natalia Szałaj (N)

Department of Physicochemical Drug Analysis, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.

Holger Stark (H)

Institute of Pharmaceutical and Medicinal Chemistry, Heinrich Heine University Düsseldorf, Universitaetsstr. 1, 40225 Duesseldorf, Germany.

Barbara Malawska (B)

Department of Physicochemical Drug Analysis, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.

Anna Więckowska (A)

Department of Physicochemical Drug Analysis, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.

Krzysztof Walczyński (K)

Department of Synthesis and Technology of Drugs, Medical University of Lodz, Muszyńskiego 1, 90-151 Łódź, Poland.

Classifications MeSH