Optimization of a medium composition for the heterologous production of Alcaligenes faecalis penicillin G acylase in Bacillus megaterium.

Alcaligenes faecalis Bacillus megaterium Design of experiments Expression Penicillin acylase

Journal

Protein expression and purification
ISSN: 1096-0279
Titre abrégé: Protein Expr Purif
Pays: United States
ID NLM: 9101496

Informations de publication

Date de publication:
10 2023
Historique:
received: 23 02 2023
revised: 06 06 2023
accepted: 20 06 2023
medline: 5 7 2023
pubmed: 23 6 2023
entrez: 22 6 2023
Statut: ppublish

Résumé

Penicillin G acylase (PGA) is a strategic enzyme in the production processes of beta-lactam antibiotics. High demand for β-lactam semisynthetic antibiotics explain the genetic and biochemical engineering strategies devoted towards novel ways for PGA production and application. This work presents a fermentation process for the heterologous production of PGA from Alcaligenes faecalis in Bacillus megaterium with optimization. The thermal stability from A. faecalis PGA is considerably higher than other described PGA and the recombinant enzyme is secreted to the culture medium by B. megaterium, which facilitates the separation and purification steps. Media optimization using fractional factorial design experiments was used to identify factors related to PGA activity detection in supernatant and cell lysates. The optimized medium resulted in almost 6-fold increased activity in the supernatant samples when compared with the basal medium. Maximum enzyme activity in optimized medium composition achieves values between 135 and 140 IU/ml. The results suggest a promising model for recombinant production of PGA in B. megaterium with possible extracellular expression of the active enzyme.

Identifiants

pubmed: 37348663
pii: S1046-5928(23)00098-0
doi: 10.1016/j.pep.2023.106327
pii:
doi:

Substances chimiques

Penicillin Amidase EC 3.5.1.11
Anti-Bacterial Agents 0
beta-Lactams 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

106327

Informations de copyright

Copyright © 2023 Elsevier Inc. All rights reserved.

Auteurs

Wagner Lopes (W)

Institute of Drug Technology, Oswaldo Cruz Foundation, Rio de Janeiro, RJ, Brazil.

Poliana Deolindo (P)

Institute of Drug Technology, Oswaldo Cruz Foundation, Rio de Janeiro, RJ, Brazil.

Alexandre Andrade de Souza Costa (AA)

Institute of Drug Technology, Oswaldo Cruz Foundation, Rio de Janeiro, RJ, Brazil.

Melissa Teixeira Gomes da Silva (MT)

Institute of Drug Technology, Oswaldo Cruz Foundation, Rio de Janeiro, RJ, Brazil.

Otavio Padula de Miranda (OP)

Institute of Drug Technology, Oswaldo Cruz Foundation, Rio de Janeiro, RJ, Brazil.

Graziela Jardim Pacheco (GJ)

Institute of Drug Technology, Oswaldo Cruz Foundation, Rio de Janeiro, RJ, Brazil. Electronic address: graziela.pacheco@fiocruz.br.

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Classifications MeSH