RNAseq Analysis of Novel 1,3,4-Oxadiazole Chalcogen Analogues Reveals Anti-Tubulin Properties on Cancer Cell Lines.


Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
09 Jul 2023
Historique:
received: 16 05 2023
revised: 30 06 2023
accepted: 04 07 2023
medline: 31 7 2023
pubmed: 29 7 2023
entrez: 29 7 2023
Statut: epublish

Résumé

1,3,4-Oxadiazole derivatives are among the most studied anticancer drugs. Previous studies have analyzed the action of different 1,3,4-oxadiazole derivatives and their effects on cancer cells. This study investigated the characterization of two new compounds named

Identifiants

pubmed: 37511023
pii: ijms241411263
doi: 10.3390/ijms241411263
pmc: PMC10379353
pii:
doi:

Substances chimiques

Tubulin 0
1,3,4-oxadiazole 20O2F20OUR
Antineoplastic Agents 0
Tubulin Modulators 0
Chalcogens 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Références

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Auteurs

Stefano Zoroddu (S)

Department of Biomedical Sciences, University of Sassari, Viale San Pietro 43/b, 07100 Sassari, Italy.

Luca Sanna (L)

Department of Biomedical Sciences, University of Sassari, Viale San Pietro 43/b, 07100 Sassari, Italy.

Valentina Bordoni (V)

Department of Biomedical Sciences, University of Sassari, Viale San Pietro 43/b, 07100 Sassari, Italy.

Weidong Lyu (W)

Division of Immunology, International Institute of Infection and Immunity, Shantou University Medical College, Shantou 515031, China.

Gabriele Murineddu (G)

Department of Medicine, Surgery and Pharmacy, University of Sassari, 07100 Sassari, Italy.

Gerard A Pinna (GA)

Department of Medicine, Surgery and Pharmacy, University of Sassari, 07100 Sassari, Italy.

Sonia Vanina Forcales (SV)

Department of Pathology and Experimental Therapeutics, School of Medicine, Health Science Campus of Bellvitge, University of Barcelona, Carrer de la Feixa Llarga, s/n, Hospitalet de Llobregat, 08907 Barcelona, Spain.

Arturo Sala (A)

Centre for Inflammation Research and Translational Medicine (CIRTM), Department of Life Sciences, Brunel University, London UB8 3PH, UK.

David J Kelvin (DJ)

Division of Immunology, International Institute of Infection and Immunity, Shantou University Medical College, Shantou 515031, China.
Department of Microbiology and Immunology, Dalhousie University, 6299 South St, Halifax, NS B3H 4R2, Canada.

Luigi Bagella (L)

Department of Biomedical Sciences, University of Sassari, Viale San Pietro 43/b, 07100 Sassari, Italy.
Sbarro Institute for Cancer Research and Molecular Medicine, Centre for Biotechnology, College of Science and Technology, Temple University, Philadelphia, PA 19122, USA.

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Classifications MeSH