International Union of Basic and Clinical Pharmacology CXIII: Nuclear Receptor Superfamily-Update 2023.
Journal
Pharmacological reviews
ISSN: 1521-0081
Titre abrégé: Pharmacol Rev
Pays: United States
ID NLM: 0421737
Informations de publication
Date de publication:
Nov 2023
Nov 2023
Historique:
received:
05
07
2021
revised:
07
08
2023
accepted:
10
08
2023
medline:
23
10
2023
pubmed:
17
8
2023
entrez:
16
8
2023
Statut:
ppublish
Résumé
The NR superfamily comprises 48 transcription factors in humans that control a plethora of gene network programs involved in a wide range of physiologic processes. This review will summarize and discuss recent progress in NR biology and drug development derived from integrating various approaches, including biophysical techniques, structural studies, and translational investigation. We also highlight how defective NR signaling results in various diseases and disorders and how NRs can be targeted for therapeutic intervention via modulation via binding to synthetic lipophilic ligands. Furthermore, we also review recent studies that improved our understanding of NR structure and signaling. SIGNIFICANCE STATEMENT: Nuclear receptors (NRs) are ligand-regulated transcription factors that are critical regulators of myriad physiological processes. NRs serve as receptors for an array of drugs, and in this review, we provide an update on recent research into the roles of these drug targets.
Identifiants
pubmed: 37586884
pii: pharmrev.121.000436
doi: 10.1124/pharmrev.121.000436
pmc: PMC10595025
doi:
Substances chimiques
Receptors, Cytoplasmic and Nuclear
0
Transcription Factors
0
Carrier Proteins
0
Ligands
0
Types de publication
Review
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Pagination
1233-1318Subventions
Organisme : NIAMS NIH HHS
ID : R01 AR069280
Pays : United States
Organisme : NIA NIH HHS
ID : RF1 AG077160
Pays : United States
Organisme : BLRD VA
ID : I01 BX002773
Pays : United States
Organisme : NIA NIH HHS
ID : RF1 AG060769
Pays : United States
Organisme : NIDDK NIH HHS
ID : F32 DK105845
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK056123
Pays : United States
Organisme : Intramural NIH HHS
ID : Z01 ES090057
Pays : United States
Organisme : NIGMS NIH HHS
ID : P20 GM103546
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK129646
Pays : United States
Organisme : NINDS NIH HHS
ID : R01 NS126204
Pays : United States
Organisme : NIMH NIH HHS
ID : R01 MH093429
Pays : United States
Organisme : NIMH NIH HHS
ID : R01 MH092769
Pays : United States
Organisme : NIDDK NIH HHS
ID : R56 DK056123
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK061935
Pays : United States
Organisme : NIDDK NIH HHS
ID : R01 DK117940
Pays : United States
Organisme : Intramural NIH HHS
ID : Z01 ES070065
Pays : United States
Organisme : BLRD VA
ID : I01 BX005466
Pays : United States
Organisme : Intramural NIH HHS
ID : Z01 ES101586
Pays : United States
Organisme : NIDDK NIH HHS
ID : R55 DK061935
Pays : United States
Informations de copyright
U.S. Government work not protected by U.S. copyright.
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