Tacrolimus Exposure Before and After a Switch From Twice-Daily Immediate-Release to Once-Daily Prolonged Release Tacrolimus: The ENVARSWITCH Study.

AUC monitoring LCP-tacrolimus conversion dose individualization dried blood spots kidney transplantation liver transplantation therapeutic drug monitoring

Journal

Transplant international : official journal of the European Society for Organ Transplantation
ISSN: 1432-2277
Titre abrégé: Transpl Int
Pays: Switzerland
ID NLM: 8908516

Informations de publication

Date de publication:
2023
Historique:
received: 15 03 2023
accepted: 06 07 2023
medline: 18 8 2023
pubmed: 17 8 2023
entrez: 17 8 2023
Statut: epublish

Résumé

LCP-tacrolimus displays enhanced oral bioavailability compared to immediate-release (IR-) tacrolimus. The ENVARSWITCH study aimed to compare tacrolimus AUC

Identifiants

pubmed: 37588007
doi: 10.3389/ti.2023.11366
pii: 11366
pmc: PMC10425592
doi:

Substances chimiques

Tacrolimus WM0HAQ4WNM

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

11366

Informations de copyright

Copyright © 2023 Monchaud, Woillard, Crépin, Tafzi, Micallef, Rerolle, Dharancy, Conti, Choukroun, Thierry, Buchler, Salamé, Garrouste, Duvoux, Colosio, Merville, Anglicheau, Etienne, Saliba, Mariat, Debette-Gratien and Marquet.

Déclaration de conflit d'intérêts

CMo reports receiving lecture fees and support for participation in International Congress from Astellas. SD reports receiving lecture fees from Chiesi, Novartis, Sandoz, Intercept, Astellas, Roche, Ipsen and Abbvie and serving as a board member of Novartis and Biotest. AT reports a research grant from Astellas. MB reports financial support from Chiesi for participation in International Congress. CG has received consulting fees from Chiesi and speaker’s honoraria from Astellas. DA has received travel grant and honoraria for lectures from Chiesi. FS has received speaker’s honoraria and/or research grants from Chiesi, Novartis, Astellas, Gilead, Neovii, Merck Sharp & Dohme, Pfizer and Baxter. CMa reports research grants, financial support for participation in congresses and expertise fees from Chiesi and Astellas. PMa has received speaker and consultant honoraria and/or research grants from Chiesi, Sandoz, Astellas and BMS. The remaining authors declare that the research was conducted in the absence of any commercial or financial relationships that could be construed as a potential conflict of interest.

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Auteurs

Caroline Monchaud (C)

Department of Pharmacology, Toxicology and Pharmacovigilance, Centre Hospitalier Universitaire de Limoges, Limoges, France.
INSERM1248 Pharmacolgy and Transplantation, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.

Jean-Baptiste Woillard (JB)

Department of Pharmacology, Toxicology and Pharmacovigilance, Centre Hospitalier Universitaire de Limoges, Limoges, France.
INSERM1248 Pharmacolgy and Transplantation, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.

Sabrina Crépin (S)

Department of Pharmacology, Toxicology and Pharmacovigilance, Centre Hospitalier Universitaire de Limoges, Limoges, France.
INSERM1248 Pharmacolgy and Transplantation, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.
Unité de Vigilance des Essais Cliniques, Centre Hospitalier Universitaire de Limoges, Limoges, France.

Naïma Tafzi (N)

Department of Pharmacology, Toxicology and Pharmacovigilance, Centre Hospitalier Universitaire de Limoges, Limoges, France.

Ludovic Micallef (L)

Department of Pharmacology, Toxicology and Pharmacovigilance, Centre Hospitalier Universitaire de Limoges, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.

Jean-Philippe Rerolle (JP)

INSERM1248 Pharmacolgy and Transplantation, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.
Department of Nephrology, Dialysis and Transplantation, Centre Hospitalier Universitaire de Limoges, Limoges, France.

Sébastien Dharancy (S)

Department of Hepatology-Transplantation, CHU Lille, Lille, France.

Filomena Conti (F)

Department of Hepato-Gastro-Enterology, Hôpital Pitié-Salpêtrière, Paris, France.

Gabriel Choukroun (G)

Department of Nephrology, Internal Medicine, Transplantation, Centre Hospitalier Universitaire (CHU) d'Amiens, Amiens, France.

Antoine Thierry (A)

Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Poitiers, France.
Department of Nephrology, Hemodialysis and Renal Transplantation, Centre Hospitalier Universitaire (CHU) de Poitiers, Poitiers, France.

Matthias Buchler (M)

Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Tours, France.
Department of Nephrology-Arterial Hypertension, Dialyses, Renal Transplantation, Centre Hospitalier Universitaire de Tours, Tours, France.

Ephrem Salamé (E)

Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Tours, France.
Center for Hepatobiliary and Pancreatic Surgery, Hepatic Transplantation, Centre Hospitalier Universitaire de Tours, Tours, France.

Cyril Garrouste (C)

Department of Nephrology-Hemodialyses, Centre Hospitalier Universitaire de Clermont-Ferrand, Clermont-Ferrand, France.

Christophe Duvoux (C)

Department of Hepatology, Hôpital Henri-Mondor, Assistance Publique Hôpitaux de Paris, Créteil, France.

Charlotte Colosio (C)

Department of Nephrology, Centre Hospitalier Universitaire de Reims, Reims, France.

Pierre Merville (P)

Department of Nephrology, Transplantation, Dialysis and Aphereses, Centre Hospitalier Universitaire de Bordeaux, Bordeaux, France.

Dany Anglicheau (D)

Department of Kidney and Metabolism Diseases, Transplantation and Clinical Immunology, Hôpital Necker-Enfants Malades, Paris, France.

Isabelle Etienne (I)

Department of Nephrology, Hemodialysis, Transplantation, Centre Hospitalier Universitaire (CHU) de Rouen, Rouen, France.

Faouzi Saliba (F)

Hôpital Paul Brousse, Villejuif, France.

Christophe Mariat (C)

Department of Nephrology, Dialysis and Renal Transplantation, Centre Hospitalier Universitaire (CHU) de Saint-Étienne, Saint-Etienne, France.

Marilyne Debette-Gratien (M)

INSERM1248 Pharmacolgy and Transplantation, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.
Department of Hepato-Gastro-Enterology and Nutrition, Centre Hospitalier Universitaire de Limoges, Limoges, France.

Pierre Marquet (P)

Department of Pharmacology, Toxicology and Pharmacovigilance, Centre Hospitalier Universitaire de Limoges, Limoges, France.
INSERM1248 Pharmacolgy and Transplantation, Limoges, France.
Fédération Hospitalo-Universitaire Survival Optimization in Organ Transplantation (FHU SUPORT), Limoges, France.

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