Strat-M® positioning for skin permeation studies: A comparative study including EpiSkin® RHE, and human skin.

Excised human skin High-performance liquid chromatography Human skin models Lipid analysis Permeation assays Raman spectroscopy Reconstructed human skin Resorcinol Strat-M®

Journal

International journal of pharmaceutics
ISSN: 1873-3476
Titre abrégé: Int J Pharm
Pays: Netherlands
ID NLM: 7804127

Informations de publication

Date de publication:
25 Nov 2023
Historique:
received: 04 07 2023
revised: 25 09 2023
accepted: 04 10 2023
medline: 27 11 2023
pubmed: 8 10 2023
entrez: 7 10 2023
Statut: ppublish

Résumé

In the development and optimization of dermatological products, In Vitro Permeation Testing (IVPT) is pivotal for controlled study of skin penetration. To enhance standardization and replicate human skin properties reconstructed human skin and synthetic membranes are explored as alternatives. Strat-M® is a membrane designed to mimic the multi-layered structure of human skin for IVPT. For instance, in Strat-M®, the steady-state fluxes (J

Identifiants

pubmed: 37805151
pii: S0378-5173(23)00909-2
doi: 10.1016/j.ijpharm.2023.123488
pii:
doi:

Substances chimiques

Membranes, Artificial 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

123488

Informations de copyright

Copyright © 2023 Elsevier B.V. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of Competing Interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Hichem Kichou (H)

Université de Tours, EA 6295 Nanomédicaments et Nanosondes, Faculté de Pharmacie, 31 Avenue Monge, 37200 Tours, France.

Franck Bonnier (F)

LVMH Recherche, 185 Av. de Verdun, 45800 Saint-Jean-de-Braye, France.

Yuri Dancik (Y)

Certara UK Ltd., Simcyp Division, Level 2-Acero, 1 Concourse Way, Sheffield S1 2B1, UK.

Joudi Bakar (J)

Université Paris-Saclay, Faculté de Pharmacie, Lip(sys)(2) « Lipides, Systèmes Analytiques et Biologiques », 17 avenue des sciences, 91400 Orsay, France.

Rime Michael-Jubeli (R)

Université Paris-Saclay, Faculté de Pharmacie, Lip(sys)(2) « Lipides, Systèmes Analytiques et Biologiques », 17 avenue des sciences, 91400 Orsay, France.

Amanda C Caritá (AC)

Université de Tours, EA 6295 Nanomédicaments et Nanosondes, Faculté de Pharmacie, 31 Avenue Monge, 37200 Tours, France.

Xavier Perse (X)

Université de Tours, EA 6295 Nanomédicaments et Nanosondes, Faculté de Pharmacie, 31 Avenue Monge, 37200 Tours, France.

Martin Soucé (M)

Université de Tours, EA 6295 Nanomédicaments et Nanosondes, Faculté de Pharmacie, 31 Avenue Monge, 37200 Tours, France.

Laetitia Rapetti (L)

Alphenyx, 430 avenue du Maréchal Lattre de Tassigny, 13009 Marseille, France.

Ali Tfayli (A)

Université Paris-Saclay, Faculté de Pharmacie, Lip(sys)(2) « Lipides, Systèmes Analytiques et Biologiques », 17 avenue des sciences, 91400 Orsay, France.

Igor Chourpa (I)

Université de Tours, EA 6295 Nanomédicaments et Nanosondes, Faculté de Pharmacie, 31 Avenue Monge, 37200 Tours, France.

Emilie Munnier (E)

Université de Tours, EA 6295 Nanomédicaments et Nanosondes, Faculté de Pharmacie, 31 Avenue Monge, 37200 Tours, France. Electronic address: emilie.munnier@univ-tours.fr.

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Classifications MeSH