Ozanimod Therapy in Patients With COVID-19 Requiring Oxygen Support: A Randomized, Open-Label, Pilot Trial.

COVID-19 bradycardia immunomodulators new therapeutic class pneumonia sphingosine-1-phosphate receptor ligands

Journal

Chest
ISSN: 1931-3543
Titre abrégé: Chest
Pays: United States
ID NLM: 0231335

Informations de publication

Date de publication:
28 Oct 2023
Historique:
received: 04 05 2023
revised: 26 09 2023
accepted: 20 10 2023
pubmed: 29 10 2023
medline: 29 10 2023
entrez: 28 10 2023
Statut: aheadofprint

Résumé

Sphingosine-1-phosphate receptor ligands (SRLs) dampen immunopathologic damages in models of viral pneumonia. Is it feasible to administer an SRL therapy, here ozanimod (OZA), to acutely ill patients infected with SARS-CoV-2? The prospective, randomized, open-label, COVID-19 Ozanimod Intervention (COZI) pilot trial was conducted in three Canadian hospitals. Patients admitted for COVID-19 requiring oxygen were eligible. Randomization was stratified for risk factors of poor outcome and oxygen needs at inclusion. Participants were allocated to standard of care (SOC) or to SOC plus OZA. OZA (oral, once daily, incremental dosage) was administered for a maximum of 14 days. Primary end point investigated for size effect and variance over time was the assessment of safety and efficacy, evaluated by the daily score on the World Health Organization-adapted six-point ordinal scale for clinical improvement analyzed under the intention-to-treat principle. Twenty-three patients were randomized to the SOC arm, and 20 were randomized to the OZA arm from September 2020 to February 2022. Evaluation of efficacy showed nonsignificant reductions of median duration of respiratory support (6 [range, 3-10] vs 9 [range, 4-12] days; P = .34), median duration of hospitalization (9 [range, 6-12] vs 10 [range, 6-18] days; P = .20), and median time to clinical improvement (4 [range, 3-7] vs 7 [range, 3-11] days; P = .12) for OZA compared with SOC, respectively. Heart rate was significantly lower with OZA (65 [range, 63-67] vs 71 [range, 69-72] beats/min; P < .0001). However, QT and PR intervals were not affected. No severe adverse drug reaction was reported. To our knowledge, SRL utility in severe pneumonia has never been tested in patients. We show for the first time that this new pharmacologic agent can safely be administered to patients hospitalized for viral pneumonia, with potential clinical benefits. Bradycardia was frequent but well tolerated. ClinicalTrials.gov; No.: NCT04405102; URL: www. gov.

Sections du résumé

BACKGROUND BACKGROUND
Sphingosine-1-phosphate receptor ligands (SRLs) dampen immunopathologic damages in models of viral pneumonia.
RESEARCH QUESTION OBJECTIVE
Is it feasible to administer an SRL therapy, here ozanimod (OZA), to acutely ill patients infected with SARS-CoV-2?
STUDY DESIGN AND METHODS METHODS
The prospective, randomized, open-label, COVID-19 Ozanimod Intervention (COZI) pilot trial was conducted in three Canadian hospitals. Patients admitted for COVID-19 requiring oxygen were eligible. Randomization was stratified for risk factors of poor outcome and oxygen needs at inclusion. Participants were allocated to standard of care (SOC) or to SOC plus OZA. OZA (oral, once daily, incremental dosage) was administered for a maximum of 14 days. Primary end point investigated for size effect and variance over time was the assessment of safety and efficacy, evaluated by the daily score on the World Health Organization-adapted six-point ordinal scale for clinical improvement analyzed under the intention-to-treat principle.
RESULTS RESULTS
Twenty-three patients were randomized to the SOC arm, and 20 were randomized to the OZA arm from September 2020 to February 2022. Evaluation of efficacy showed nonsignificant reductions of median duration of respiratory support (6 [range, 3-10] vs 9 [range, 4-12] days; P = .34), median duration of hospitalization (9 [range, 6-12] vs 10 [range, 6-18] days; P = .20), and median time to clinical improvement (4 [range, 3-7] vs 7 [range, 3-11] days; P = .12) for OZA compared with SOC, respectively. Heart rate was significantly lower with OZA (65 [range, 63-67] vs 71 [range, 69-72] beats/min; P < .0001). However, QT and PR intervals were not affected. No severe adverse drug reaction was reported.
INTERPRETATION CONCLUSIONS
To our knowledge, SRL utility in severe pneumonia has never been tested in patients. We show for the first time that this new pharmacologic agent can safely be administered to patients hospitalized for viral pneumonia, with potential clinical benefits. Bradycardia was frequent but well tolerated.
CLINICAL TRIAL REGISTRATION BACKGROUND
ClinicalTrials.gov; No.: NCT04405102; URL: www.
CLINICALTRIALS RESULTS
gov.

Identifiants

pubmed: 37898184
pii: S0012-3692(23)05668-4
doi: 10.1016/j.chest.2023.10.023
pii:
doi:

Banques de données

ClinicalTrials.gov
['NCT04405102']

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

Copyright © 2023 American College of Chest Physicians. Published by Elsevier Inc. All rights reserved.

Déclaration de conflit d'intérêts

Financial/Nonfinancial Disclosures The authors have reported to CHEST the following: F. L. is a shareholder and administrator of the board of directors of OxyNov for the FreeO(2) device used in a few participants in this study. F. M. has financial participation in this company. None declared (P. B.-L., J.-F. S., P. R., T. N., N. C., D. M.).

Auteurs

François Lellouche (F)

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval, Quebec City, Canada; Department of Medicine, Université Laval, Quebec City, Canada. Electronic address: francois.lellouche@criucpq.ulaval.ca.

Pascale Blais-Lecours (P)

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval, Quebec City, Canada.

François Maltais (F)

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval, Quebec City, Canada; Department of Medicine, Université Laval, Quebec City, Canada.

Jean-François Sarrazin (JF)

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval, Quebec City, Canada; Department of Medicine, Université Laval, Quebec City, Canada.

Philippe Rola (P)

CIUSSS EMTL, Santa Cabrini Hospital, Montreal, Canada.

Tuyen Nguyen (T)

CISSS Laval, Cité-de-la-Santé Hospital, Laval, QC, Canada.

Nathalie Châteauvert (N)

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval, Quebec City, Canada.

David Marsolais (D)

Institut universitaire de cardiologie et de pneumologie de Québec-Université Laval, Quebec City, Canada; Department of Medicine, Université Laval, Quebec City, Canada.

Classifications MeSH