Candidate Tracers for Imaging Colony-Stimulating Factor 1 Receptor in Neuroinflammation with Positron Emission Tomography: Issues and Progress.
Journal
ACS pharmacology & translational science
ISSN: 2575-9108
Titre abrégé: ACS Pharmacol Transl Sci
Pays: United States
ID NLM: 101721411
Informations de publication
Date de publication:
10 Nov 2023
10 Nov 2023
Historique:
received:
31
08
2023
pmc-release:
18
10
2024
medline:
17
11
2023
pubmed:
17
11
2023
entrez:
17
11
2023
Statut:
epublish
Résumé
The tyrosine kinase, colony-stimulating factor 1 receptor (CSF1R), has attracted attention as a potential biomarker of neuroinflammation for imaging studies with positron emission tomography (PET), especially because of its location on microglia and its role in microglia proliferation. The development of an effective radiotracer for specifically imaging and quantifying brain CSF1R is highly challenging. Here we review the progress that has been made on PET tracer development and discuss issues that have arisen and which remain to be addressed and resolved.
Identifiants
pubmed: 37974622
doi: 10.1021/acsptsci.3c00213
pmc: PMC10644394
doi:
Types de publication
Journal Article
Review
Langues
eng
Pagination
1632-1650Informations de copyright
Not subject to U.S. Copyright. Published 2023 by American Chemical Society.
Déclaration de conflit d'intérêts
The authors declare no competing financial interest.
Références
Pharmaceuticals (Basel). 2018 Dec 13;11(4):
pubmed: 30551596
Front Cell Neurosci. 2021 Jul 02;15:691067
pubmed: 34276311
Nat Biotechnol. 2011 Oct 30;29(11):1046-51
pubmed: 22037378
Front Aging Neurosci. 2017 Aug 09;9:244
pubmed: 28848420
Front Neurosci. 2021 Sep 24;15:742065
pubmed: 34630027
J Cereb Blood Flow Metab. 2021 Sep;41(9):2410-2422
pubmed: 33757319
Drug Des Devel Ther. 2020 May 04;14:1693-1704
pubmed: 32440095
J Exp Med. 2013 Jan 14;210(1):157-72
pubmed: 23296467
Pharmaceuticals (Basel). 2022 Feb 23;15(3):
pubmed: 35337075
Cancer Res. 1993 Oct 1;53(19):4595-602
pubmed: 8402633
Curr Drug Metab. 2007 May;8(4):341-63
pubmed: 17504223
Bioorg Med Chem Lett. 2017 May 15;27(10):2153-2160
pubmed: 28377059
Science. 2015 Jan 23;347(6220):1260419
pubmed: 25613900
Front Aging Neurosci. 2021 Nov 15;13:789834
pubmed: 34867307
Bioorg Med Chem. 2021 Jul 15;42:116245
pubmed: 34119698
AIDS. 2023 Jul 15;37(9):1419-1424
pubmed: 37070549
Curr Med Chem. 2022 Aug 6;29(28):4862-4890
pubmed: 35352645
Semin Nucl Med. 2023 Mar;53(2):213-229
pubmed: 36270830
Curr Top Med Chem. 2009;9(7):599-610
pubmed: 19689368
Cytokine. 2012 Dec;60(3):793-805
pubmed: 22974529
Biochem Soc Trans. 2015 Aug;43(4):586-92
pubmed: 26551697
J Neurol. 2016 Sep;263(9):1864-5
pubmed: 27314966
Bioorg Med Chem Lett. 2022 Jun 1;65:128704
pubmed: 35351586
Pharmacol Res. 2016 Jan;103:26-48
pubmed: 26529477
J Virol. 2016 Jun 24;90(14):6255-6262
pubmed: 27122585
Eur J Med Chem. 2023 Jul 5;255:115344
pubmed: 37141705
Drug Metab Dispos. 2013 Apr;41(4):754-62
pubmed: 23305710
Trends Neurosci. 2016 Jun;39(6):378-393
pubmed: 27083478
Cancer Lett. 1999 Nov 15;146(2):117-26
pubmed: 10656616
Development. 1996 Sep;122(9):2661-72
pubmed: 8787741
EJNMMI Res. 2022 Sep 30;12(1):64
pubmed: 36175737
Nucleic Acids Res. 2000 Jan 1;28(1):235-42
pubmed: 10592235
Acta Pharm Sin B. 2021 Feb;11(2):373-393
pubmed: 33643818
Proc Natl Acad Sci U S A. 2005 Nov 1;102(44):16078-83
pubmed: 16249345
Neuron. 2014 Apr 16;82(2):380-97
pubmed: 24742461
Nucl Med Biol. 2021 Sep-Oct;100-101:44-51
pubmed: 34174546
Brain. 2009 Apr;132(Pt 4):1078-92
pubmed: 19151372
Bioorg Med Chem Lett. 2008 Mar 1;18(5):1642-8
pubmed: 18242992
J Med Chem. 2021 Dec 23;64(24):17656-17689
pubmed: 34905377
Front Immunol. 2022 Sep 23;13:1010946
pubmed: 36211392
J Pharmacol Exp Ther. 2012 Dec;343(3):650-60
pubmed: 22942241
Curr Oncol Rep. 2017 Sep 5;19(11):70
pubmed: 28875266
Nucl Med Biol. 2022 Nov-Dec;114-115:99-107
pubmed: 36371938
Front Neurol. 2022 Apr 29;13:874388
pubmed: 35572921
Chem Rev. 2008 May;108(5):1501-16
pubmed: 18426240
EJNMMI Radiopharm Chem. 2022 May 8;7(1):11
pubmed: 35526184
Expert Opin Drug Discov. 2008 Jun;3(6):607-621
pubmed: 19662101
Cancer Discov. 2011 Jun;1(1):54-67
pubmed: 22039576
J Immunol. 1993 Jan 15;150(2):594-604
pubmed: 8419491
Bioorg Med Chem. 2023 Apr 1;83:117233
pubmed: 36933438
Lancet Neurol. 2015 Apr;14(4):388-405
pubmed: 25792098
Nat Med. 2013 Oct;19(10):1264-72
pubmed: 24056773
J Nucl Med. 2008 Aug;49(8):1328-35
pubmed: 18632828
Nat Commun. 2019 Aug 21;10(1):3758
pubmed: 31434879
Drug Dev Res. 2023 May;84(3):484-513
pubmed: 36779375
Front Neurosci. 2022 May 24;16:872509
pubmed: 35685772
Curr Med Chem. 2016;23(18):1818-69
pubmed: 27087244
ACS Chem Neurosci. 2021 Mar 17;12(6):998-1006
pubmed: 33667059
J Nucl Med. 2020 Aug;61(8):1107-1112
pubmed: 32620705
Am J Pathol. 2000 Sep;157(3):895-904
pubmed: 10980129
Nat Biotechnol. 2008 Jan;26(1):127-32
pubmed: 18183025
ACS Chem Neurosci. 2022 Dec 21;13(24):3641-3660
pubmed: 36473177
J Comp Neurol. 1998 Jun 8;395(3):342-58
pubmed: 9596528
Nature. 1997 Oct 16;389(6652):689-95
pubmed: 9338779
Proc Natl Acad Sci U S A. 2019 Jan 29;116(5):1686-1691
pubmed: 30635412
Trends Pharmacol Sci. 2009 Aug;30(8):431-40
pubmed: 19616318
Nat Rev Cancer. 2012 Nov;12(11):753-66
pubmed: 23076159
Acta Neuropathol. 2001 Mar;101(3):249-55
pubmed: 11307625
N Engl J Med. 2015 Jul 30;373(5):428-37
pubmed: 26222558
Bioorg Med Chem Lett. 2019 Jan 1;29(1):115-118
pubmed: 30442420
Xenobiotica. 2015 Feb;45(2):107-23
pubmed: 25180976
J Med Chem. 2020 Feb 13;63(3):1397-1414
pubmed: 31934767
Lancet Psychiatry. 2020 Dec;7(12):1064-1074
pubmed: 33098761
Front Immunol. 2021 Sep 16;12:739130
pubmed: 34603323
J Labelled Comp Radiopharm. 2019 Nov;62(13):903-908
pubmed: 31524293
Bioorg Med Chem Lett. 2010 Mar 1;20(5):1543-7
pubmed: 20137931
Eur J Neurosci. 2021 Jan;53(1):151-171
pubmed: 32150310
Dev Biol. 2012 Jul 15;367(2):100-13
pubmed: 22542597
Clin Cancer Res. 2005 Mar 15;11(6):2320-6
pubmed: 15788683
Int Immunopharmacol. 2008 Oct;8(10):1354-76
pubmed: 18687298
Blood. 2010 Feb 18;115(7):1461-71
pubmed: 20008303
Cell Rep. 2018 Jul 31;24(5):1203-1217.e6
pubmed: 30067976
Brain Res. 1994 Mar 7;639(1):171-4
pubmed: 7514086
Int J Mol Sci. 2019 Jun 28;20(13):
pubmed: 31261683
Science. 2020 Mar 6;367(6482):
pubmed: 32139519
Bioorg Med Chem Lett. 2009 Feb 1;19(3):701-5
pubmed: 19114305
Eur J Nucl Med Mol Imaging. 2019 Dec;46(13):2831-2847
pubmed: 31396666
Bioorg Med Chem Lett. 2014 Oct 15;24(20):4784-90
pubmed: 25257201
Biomedicines. 2021 Oct 12;9(10):
pubmed: 34680566
Glia. 2001 Jul;35(1):72-9
pubmed: 11424194
Prog Mol Biol Transl Sci. 2019;165:371-399
pubmed: 31481170
J Pharmacol Exp Ther. 2008 Jul;326(1):41-50
pubmed: 18434589
J Cereb Blood Flow Metab. 2007 Sep;27(9):1533-9
pubmed: 17519979
ACS Pharmacol Transl Sci. 2023 Mar 10;6(4):614-632
pubmed: 37082755
J Med Chem. 1988 Mar;31(3):656-71
pubmed: 2894467