Insight into the molecular interaction between the anticancer drug, enzalutamide and human alpha-2-macroglobulin: Biochemical and biophysical approach.

Alpha-2-macroglobulin Circular dichroism Enzalutamide Fluorescence spectroscopy Isothermal titration calorimetry

Journal

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy
ISSN: 1873-3557
Titre abrégé: Spectrochim Acta A Mol Biomol Spectrosc
Pays: England
ID NLM: 9602533

Informations de publication

Date de publication:
26 Jan 2024
Historique:
received: 19 10 2023
revised: 21 01 2024
accepted: 22 01 2024
medline: 5 2 2024
pubmed: 5 2 2024
entrez: 4 2 2024
Statut: aheadofprint

Résumé

The drug pharmacokinetics is affected upon binding with proteins, thus making drug-protein interactions crucial. This study investigated the interaction between enzalutamide and human major antiproteinase alpha-2-macroglobulin (α

Identifiants

pubmed: 38310741
pii: S1386-1425(24)00123-9
doi: 10.1016/j.saa.2024.123957
pii:
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

123957

Informations de copyright

Copyright © 2024 Elsevier B.V. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of Competing Interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Mohammad Khalid Zia (M)

Department of Biochemistry, Faculty of Life Sciences, Aligarh Muslim University, Aligarh 202002, India.

Tooba Siddiqui (T)

Department of Biochemistry, Faculty of Life Sciences, Aligarh Muslim University, Aligarh 202002, India.

Sana Ansari (S)

Department of Biochemistry, Faculty of Life Sciences, Aligarh Muslim University, Aligarh 202002, India.

Mohammad Muaz (M)

Interdisciplinary Nanotechnology Centre, Aligarh Muslim University, Aligarh 202002, India.

Haseeb Ahsan (H)

Department of Biochemistry, Faculty of Dentistry, Jamia Millia Islamia, New Delhi 110025, India.

Fahim Halim Khan (F)

Department of Biochemistry, Faculty of Life Sciences, Aligarh Muslim University, Aligarh 202002, India. Electronic address: fahimhkhan@rediffmail.com.

Classifications MeSH