Serotonin-2 Receptor Agonists Produce Anti-inflammatory Effects through Functionally Selective Mechanisms That Involve the Suppression of Disease-Induced Arginase 1 Expression.


Journal

ACS pharmacology & translational science
ISSN: 2575-9108
Titre abrégé: ACS Pharmacol Transl Sci
Pays: United States
ID NLM: 101721411

Informations de publication

Date de publication:
09 Feb 2024
Historique:
received: 24 10 2023
revised: 11 01 2024
accepted: 12 01 2024
pmc-release: 25 01 2025
medline: 15 2 2024
pubmed: 15 2 2024
entrez: 15 2 2024
Statut: epublish

Résumé

Functional selectivity in the context of serotonin 2A (5-HT

Identifiants

pubmed: 38357283
doi: 10.1021/acsptsci.3c00297
pmc: PMC10863441
doi:

Types de publication

Journal Article

Langues

eng

Pagination

478-492

Informations de copyright

© 2024 American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare the following competing financial interest(s): CDN, TPF and ALH had a sponsored research contract with Eleusis Therapeutics and CDN and TPF were members of its scientific advisory board when portions of this study were performed. CDN and TPF are founders of 2A Biosciences and receive sponsored research funding from 2A Biosciences.

Auteurs

Thomas W Flanagan (TW)

Department of Pharmacology and Experimental TherapeuticsLouisiana State University Health Sciences CenterNew Orleans, Louisiana70112, United States.

Timothy P Foster (TP)

Department of Microbiology, Immunology, and ParasitologyLouisiana State University Health Sciences CenterNew Orleans, Louisiana70112, United States.

Thomas E Galbato (TE)

Department of Microbiology, Immunology, and ParasitologyLouisiana State University Health Sciences CenterNew Orleans, Louisiana70112, United States.

Pek Yee Lum (PY)

Auransa Inc.Palo Alto, California94301, United States.

Brent Louie (B)

Auransa Inc.Palo Alto, California94301, United States.

Gavin Song (G)

Auransa Inc.Palo Alto, California94301, United States.

Adam L Halberstadt (AL)

Department of PsychiatryUniversity of San Diego, California, San Diego, California92093, United States.

Gerald B Billac (GB)

Department of Pharmacology and Experimental TherapeuticsLouisiana State University Health Sciences CenterNew Orleans, Louisiana70112, United States.

Charles D Nichols (CD)

Department of Pharmacology and Experimental TherapeuticsLouisiana State University Health Sciences CenterNew Orleans, Louisiana70112, United States.

Classifications MeSH