Novel insights into the dependence of adsorption-desorption kinetics on particle geometry in chiral chromatography.

Adsorption-desorption kinetics Chiral chromatography Sub 2-m fully porous particles Superficially porous particles

Journal

Analytical and bioanalytical chemistry
ISSN: 1618-2650
Titre abrégé: Anal Bioanal Chem
Pays: Germany
ID NLM: 101134327

Informations de publication

Date de publication:
15 Feb 2024
Historique:
received: 13 11 2023
accepted: 29 01 2024
revised: 25 01 2024
medline: 15 2 2024
pubmed: 15 2 2024
entrez: 15 2 2024
Statut: aheadofprint

Résumé

The existence of slow adsorption-desorption kinetics in chiral liquid chromatography is common knowledge. This may significantly contribute to worsening the efficiency and kinetic performance of a chromatographic run, especially when high flow rates are employed. Many attempts and protocols have been proposed to access this term, the so-called [Formula: see text], but they are based on different (theoretical) assumptions. As a consequence, no official method is available for the estimation of the adsorption-desorption kinetics term. In this work, a novel approach to access [Formula: see text] is presented. This procedure combines experimental results obtained with kinetic and thermodynamic measurements. The investigations have been performed on two zwitterionic teicoplanin chiral stationary phases (CSPs) based on 1.9 [Formula: see text]m fully porous and 2.0 [Formula: see text]m superficially porous particles (FPPs and SPPs), using Z-D,L-Methionine as probe molecule. Kinetic studies have been performed through the combination of both stop-flow and dynamic measurements, while adsorption isotherms have been calculated through Inverse Method. This study has confirmed that, on both particle formats, analyte diffusion on the surface of the particle is negligible, meaning that adsorption is localized, and it has been demonstrated that adsorption-desorption kinetics is strongly dependent on particle geometry and, in particular, on the loading of chiral selector. These findings are fundamental not only to unravel novel aspects of the complex enantiorecognition mechanism but also to optimize the employment of CSPs for ultra-fast and preparative applications.

Identifiants

pubmed: 38358532
doi: 10.1007/s00216-024-05186-z
pii: 10.1007/s00216-024-05186-z
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Ministero dell'Universitá e della Ricerca
ID : 0001052

Informations de copyright

© 2024. The Author(s).

Références

De Luca C, Felletti S, Franchina FA, Bozza D, Compagnin G, Nosengo C, Pasti L, Cavazzini A, Catani M. Recent developments in the high-throughput separation of biologically active chiral compounds via high performance liquid chromatography. J Pharm Biomed Anal. 2024;238: 115794. https://doi.org/10.1016/j.jpba.2023.115794 .
doi: 10.1016/j.jpba.2023.115794 pubmed: 37890321
Catani M, Ismail OH, Gasparrini F, Antonelli M, Pasti L, Marchetti N, Felletti S, Cavazzini A. Recent advancements and future directions of superficially porous chiral stationary phases for ultrafast high-performance enantioseparations. Analyst. 2017;142:555–66.
doi: 10.1039/C6AN02530G pubmed: 28091634
Ismail OH, Pasti L, Ciogli A, Villani C, Kocergin J, Anderson S, Gasparrini F, Cavazzini A, Catani M. Pirkle-type chiral stationary phase on core-shell and fully porous particles: are superficially porous particles always the better choice toward ultrafast high-performance enantioseparations? J Chromatogr A. 2016;1466:96–104.
Ismail OH, Ciogli A, Villani C, Martino MD, Pierini M, Cavazzini A, Bell DS, Gasparrini F. Ultra-fast high-efficiency enantioseparations by means of a teicoplanin-based chiral stationary phase made on sub-2 [Formula: see text]m totally porous silica particles of narrow size distribution. J Chromatogr A. 2016;1427:55–68.
doi: 10.1016/j.chroma.2015.11.071 pubmed: 26687167
Ismail OH, Antonelli M, Ciogli A, Villani C, Cavazzini A, Catani M, Felletti S, Bell DS, Gasparrini F. Future perspectives in high efficient and ultrafast chiral liquid chromatography through zwitterionic teicoplanin-based 2[Formula: see text]m superficially porous particles. J Chromatogr A. 2017;1520:91–102.
doi: 10.1016/j.chroma.2017.09.008 pubmed: 28911942
Felletti S, De Luca C, Lievore G, Chenet T, Chankvetadze B, Farkas T, Cavazzini A, Catani M. Mass transfer kinetics on modern Whelk-O1 chiral stationary phases made on fully- and superficially-porous particles. J Chromatogr A. 2021;1637: 461854.
doi: 10.1016/j.chroma.2020.461854 pubmed: 33387912
Felletti S, De Luca C, Mazzoccanti G, Gasparrini F, Manetto S, Franchina FA, Chenet T, Pasti L, Cavazzini A, Catani M. Understanding the transition from high-selective to high-efficient chiral separations by changing the organic modifier with zwitterionic-teicoplanin chiral stationary phase. Anal Chem. 2023;95:9630–7.
doi: 10.1021/acs.analchem.3c01344 pubmed: 37294639
Gritti F, Guiochon G. Mass transfer kinetics, band broadening and column efficiency. J Chromatogr A. 2012;1221:2–40.
doi: 10.1016/j.chroma.2011.04.058 pubmed: 21664619
Catani M, Felletti S, Ismail OH, Gasparrini F, Pasti L, Marchetti N, De Luca C, Costa V, Cavazzini A. New frontiers and cutting edge applications in ultra high performance liquid chromatography through latest generation superficially porous particles with particular emphasis to the field of chiral separations. Anal Bioanal Chem. 2018;410:2457–65.
doi: 10.1007/s00216-017-0842-4 pubmed: 29340722
Felletti S, Catani M, Mazzoccanti G, De Luca C, Lievore G, Buratti A, Pasti L, Gasparrini F, Cavazzini A. Shedding light on mechanisms leading to convex-upward van deemter curves on a cellulose tris(4-chloro-3-methylphenylcarbamate)-based chiral stationary phase. J Chromatogr A. 2020;1630: 461532.
doi: 10.1016/j.chroma.2020.461532 pubmed: 32950816
Schmitt K, Woiwode U, Kohout M, Zhang T, Lindner W, Lämmerhofer M. Comparison of small size fully porous particles and superficially porous particles of chiral anion-exchange type stationary phases in ultra-high performance liquid chromatography: effect of particle and pore size on chromatographic efficiency and kinetic performance. J Chromatogr A. 2018;1569:149–59.
doi: 10.1016/j.chroma.2018.07.056 pubmed: 30041874
Gritti F, Guiochon G. Possible resolution gain in enantioseparations afforded by core-shell particle technology. J Chromatogr A. 2014;1348:87–96.
doi: 10.1016/j.chroma.2014.04.041 pubmed: 24835764
Gritti F, Guiochon G. Mass transfer mechanism in chiral reversed phase liquid chromatography. J Chromatogr A. 2014;1332:35–45.
doi: 10.1016/j.chroma.2014.01.040 pubmed: 24529955
Neue UD. HPLC Columns: Theory, Technology and Practice (Wiley-VCH, 1997)
Gritti F, Guiochon G. General HETP equation for the study of mass-transfer mechanisms in RPLC. Anal Chem. 2006;78(15):5329–47.
doi: 10.1021/ac060203r pubmed: 16878867
Miyabe K, Matsumoto Y, Guiochon G. Peak parking-moment analysis. A strategy for the study of the mass-transfer kinetics in the stationary phase. Anal Chem. 2007;79:1970–1982.
Miyabe K, Ando N, Guiochon G. Peak parking method for measurement of molecular diffusivity in liquid phase systems. J Chromatogr A. 2009;1216:4377–82.
doi: 10.1016/j.chroma.2009.02.058 pubmed: 19345369
Desmet G, Broeckhoven K, Deridder S, Cabooter D. Review of recent insights in the measurement and modelling of the b-term dispersion and related mass transfer properties in liquid chromatography. Anal Chim Acta. 2022;1214: 339955.
doi: 10.1016/j.aca.2022.339955 pubmed: 35649640
Song H, Sadriaj D, Desmet G, Cabooter D. Methodologies to determine b-term coefficients revisited. J Chromatogr A. 2018;1532:124–35.
doi: 10.1016/j.chroma.2017.11.070 pubmed: 29221865
Knox JH, Scott HP. B and C terms in the van Deemter equation for liquid chromatography. J Chromatogr. 1983;282:297–313.
doi: 10.1016/S0021-9673(00)91609-1
Spudeit DA, Dolzan MD, Breitbach ZS, Barber WE, Micke GA, Armstrong DW. Superficially porous particles vs. fully porous particles for bonded high performance liquid chromatographic chiral stationary phases: Isopropyl cyclofructan 6. J Chromatogr A. 2014;1363:89–95.
Patel DC, Breitbach ZS, Yu J, Nguyen KA, Armstrong DW. Quinine bonded to superficially porous particles for high-efficiency and ultrafast liquid and supercritical fluid chromatography. Anal Chim Acta. 2017;963:164–74.
doi: 10.1016/j.aca.2017.02.005 pubmed: 28335970
Cavazzini A, Gritti F, Kaczmarski K, Marchetti N, Guiochon G. Mass-transfer kinetics in a shell packing material for chromatography. Anal Chem. 2007;79:5972–9.
doi: 10.1021/ac070571a pubmed: 17580955
Guiochon G, Gritti F. Shell particles, trials, tribulations and triumphs. J Chromatogr A. 2011;1218:1915–38.
doi: 10.1016/j.chroma.2011.01.080 pubmed: 21353228
Gritti F, Cavazzini A, Marchetti N, Guiochon G. Comparison between the efficiencies of columns packed with fully and partially porous C[Formula: see text]-bonded silica materials. J Chromatogr A. 2007;1157:289–303.
doi: 10.1016/j.chroma.2007.05.030 pubmed: 17543317
Felletti S, De Luca C, Lievore G, Pasti L, Chenet T, Mazzoccanti G, Gasparrini F, Cavazzini A, Catani M. Investigation of mass transfer properties and kinetic performance of high-efficiency columns packed with c18 sub-2 [Formula: see text]m fully and superficially porous particles. J Sep Sci. 2020;43:1737–45.
doi: 10.1002/jssc.202000041 pubmed: 32125067
Giddings JC. Dynamics of Chromatography. New York: Marcel Dekker; 1965.
Cavazzini A, Remelli M, Dondi F, Felinger A. Stochastic theory of multiple-site linear adsorption chromatography. Anal Chem. 1999;71:3453–62.
doi: 10.1021/ac990282p
Felinger A, Cavazzini A, Remelli M, Dondi F. Stochastic-dispersive theory of chromatography. Anal Chem. 1999;71:4472–9.
doi: 10.1021/ac990412u
Cavazzini A, Remelli M, Dondi F. Stochastic theory of two-site adsorption chromatography by the characteristic function method. J Microcol Sep. 1997;9:295–302.
doi: 10.1002/(SICI)1520-667X(1997)9:4<295::AID-MCS7>3.0.CO;2-X
Guiochon G, Felinger A, Katti A, Shirazi D. Fundamentals of Preparative and Nonlinear Chromatography. 2nd ed. Boston: Academic Press; 2006.
Felinger A, Zhou DM, Guiochon G. Determination of the single component and competitive adsorption isotherms of the 1-indanol enantiomers by the inverse method. J Chromatogr A. 2003;1005:35–49.
doi: 10.1016/S0021-9673(03)00889-6 pubmed: 12924781
Vajda P, Cavazzini A, Felinger A. Adsorption equilibria of proline in hydrophilic interaction chromatography. J Chromatogr A. 2010;1217:5965–70.
doi: 10.1016/j.chroma.2010.07.058 pubmed: 20719320
Felletti S, De Luca C, Ismail OH, Pasti L, Costa V, Gasparrini F, Cavazzini A, Catani M. On the effect of chiral selector loading and mobile phase composition on adsorption properties of latest generation fully- and superficially-porous whelk-o1 particles for high-efficient ultrafast enantioseparations. J Chromatogr A. 2018;1579:41–8.
Al-Bokari M, Cherrak D, Guiochon G. Determination of the porosities of monolithic columns by inverse size-exclusion chromatography. J Chromatogr A. 2002;975:275–84.
doi: 10.1016/S0021-9673(02)01271-2 pubmed: 12456082
Guan H, Guiochon G. Study of physico-chemical properties of some packing materials: I. Measurements of the external porosity of packed columns by inverse size-exclusion chromatography. J Chromatogr A. 1996;731:27–40.
Barhate CL, Breitbach ZS, Pinto EC, Regalado EL, Welch CJ, Amstrong DW. Ultrafast separation of fluorinated and desfluorinated pharmaceuticals using highly efficient and selective chiral selectors bonded to superficially porous particles. J Chromatogr A. 2015;1426:241–7.
doi: 10.1016/j.chroma.2015.11.056 pubmed: 26643720
Gritti F, Guiochon G. Mass transfer mechanism in hydrophilic interaction chromatography. J Chromatogr A. 2013;1302:55–64.
doi: 10.1016/j.chroma.2013.06.001 pubmed: 23827468
Berthod A, Chen XH, Kullman JP, Armstrong DW, Gasparrini F, D’Acquarica I, Villani C, Carotti A. Role of the carbohydrate moities in chiral recognition on teicoplanin-based lc stationary phases. Anal Chem. 2000;72:1767–80.
doi: 10.1021/ac991004t pubmed: 10784140
D’Acquarica I, Gasparrini F, Misiti D, Pierini M, Villani C. HPLC chiral stationary phases containing macrocyclic antibiotics: practical aspects and recognition mechanism. Adv Chromatogr. 2008;46:109–73.
pubmed: 19013947
Cavazzini A, Nadalini G, Dondi F, Gasparrini F, Ciogli A, Villani C. Study of mechanisms of chiral discrimination of amino acids and their derivatives on a teicoplanin-based chiral stationary phase. J Chromatogr A. 2004;1031:143–58.
doi: 10.1016/j.chroma.2003.10.090 pubmed: 15058578
Economou N, Zentner I, Lazo E, Jakoncic J, Stojanoff V, Weeks S, Grasty K, Cocklin S, Loll P. Structure of the complex between teicoplanin and a bacterial cell-wall peptide: use of a carrier-protein approach. Acta Crystallogr. 2013;D69:520–33.
Han S, Le B, Hajare H, Baxter R, Miller S. X-ray crystal structure of teicoplanin A-2 bound to a catalytic peptide sequence via the carrier protein strategy. J Org Chem. 2014;79:8550–6.
doi: 10.1021/jo501625f pubmed: 25147913 pmcid: 4168787
Gritti F, Guiochon G. Comparison between the intra-particle diffusivity in the hydrophilic interaction chromatography and reversed phase liquid chromatography modes. impact on the column efficiency. J Chromatogr A. 2013;1297:85–95.
Ludlum D, Warner R, Smith H. The diffusion of thiourea in water at 25[Formula: see text]C. J Phys Chem. 1962;66:1540–2.
doi: 10.1021/j100814a506
Kaczmarski K, Guiochon G. Modeling of the mass-transfer kinetics in chromatographic columns packed with shell and pellicular particles. Anal Chem. 2007;79:4648–56.
doi: 10.1021/ac070209w pubmed: 17492836

Auteurs

Chiara De Luca (C)

Department of Chemical, Pharmaceutical and Agricultural Sciences, University of Ferrara, via L. Borsari 46, Ferrara, 44121, Italy.

Greta Compagnin (G)

Department of Chemical, Pharmaceutical and Agricultural Sciences, University of Ferrara, via L. Borsari 46, Ferrara, 44121, Italy.

Chiara Nosengo (C)

Department of Chemical, Pharmaceutical and Agricultural Sciences, University of Ferrara, via L. Borsari 46, Ferrara, 44121, Italy.

Giulia Mazzoccanti (G)

Department of Drug Chemistry and Technology, "Sapienza" Università di Roma, P.le A. Moro 5, Rome, 00185, Italy.

Francesco Gasparrini (F)

Department of Drug Chemistry and Technology, "Sapienza" Università di Roma, P.le A. Moro 5, Rome, 00185, Italy.

Alberto Cavazzini (A)

Department of Chemical, Pharmaceutical and Agricultural Sciences, University of Ferrara, via L. Borsari 46, Ferrara, 44121, Italy.
Council for Agricultural Research and Economics, CREA, via della Navicella 2/4, Rome, 00184, Italy.

Martina Catani (M)

Department of Chemical, Pharmaceutical and Agricultural Sciences, University of Ferrara, via L. Borsari 46, Ferrara, 44121, Italy. ctnmtn@unife.it.

Simona Felletti (S)

Department of Environmental and Prevention Sciences, University of Ferrara, via L. Borsari 46, Ferrara, 44121, Italy. fllsmn1@unife.it.

Classifications MeSH