Structure-Based Identification of Kelch-like ECH-Associated Protein 1 as a Pharmacological Target of Electrophile-Containing Catechol-


Journal

ACS pharmacology & translational science
ISSN: 2575-9108
Titre abrégé: ACS Pharmacol Transl Sci
Pays: United States
ID NLM: 101721411

Informations de publication

Date de publication:
08 Mar 2024
Historique:
received: 13 10 2023
revised: 26 01 2024
accepted: 29 01 2024
pmc-release: 13 02 2025
medline: 14 3 2024
pubmed: 14 3 2024
entrez: 14 3 2024
Statut: epublish

Résumé

Entacapone and nitecapone are electrophile-containing catechol-

Identifiants

pubmed: 38481699
doi: 10.1021/acsptsci.3c00281
pmc: PMC10928886
doi:

Types de publication

Journal Article

Langues

eng

Pagination

693-706

Informations de copyright

© 2024 American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

Auteurs

Ping Wang (P)

College of Life Sciences, Beijing Normal University, No. 19 Xinjiekouwai Street, Beijing 100875, China.
National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Yang Li (Y)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Jinyi Yang (J)

Academy for Advanced Interdisciplinary Studies, Peking University, Beijing 102206, China.
National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Ziwen Li (Z)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Xintong Ren (X)

College of Life Sciences, Beijing Normal University, No. 19 Xinjiekouwai Street, Beijing 100875, China.
National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Qingshi Meng (Q)

State Key Laboratory of Animal Nutrition and Feeding, Institute of Animal Science, Chinese Academy of Agricultural Sciences, Beijing 100193, China.

Pengfei Li (P)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Luzhe Qin (L)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.
School of Life Sciences, Tsinghua University, Beijing 100084, China.

Wei Li (W)

RPXDs (Suzhou) Co., Ltd., Suzhou 215028, China.

Yuting Xie (Y)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Nannan Hou (N)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.

Niu Huang (N)

National Institute of Biological Sciences, No. 7 Science Park Road, Zhongguancun Life Science Park, Beijing 102206, China.
Tsinghua Institute of Multidisciplinary Biomedical Research, Tsinghua University, Beijing 102206, China.

Classifications MeSH