In vitro evaluation of PET radiotracers for imaging synaptic density, the acetylcholine transporter, AMPA-tarp-γ8 and muscarinic M4 receptors in Alzheimer's disease.

Alzheimer’s disease Autoradiography PET SV2A SynVesT-1 cholinergic fluorine-18 glutamatergic synaptic density tritium

Journal

American journal of nuclear medicine and molecular imaging
ISSN: 2160-8407
Titre abrégé: Am J Nucl Med Mol Imaging
Pays: United States
ID NLM: 101564121

Informations de publication

Date de publication:
2024
Historique:
received: 18 10 2023
accepted: 04 02 2024
medline: 19 3 2024
pubmed: 19 3 2024
entrez: 19 3 2024
Statut: epublish

Résumé

Several therapeutics and biomarkers that target Alzheimer's disease (AD) are under development. Our clinical positron emission tomography (PET) research programs are interested in six radiopharmaceuticals to image patients with AD and related dementias, specifically [

Identifiants

pubmed: 38500748
pmc: PMC10944377

Types de publication

Journal Article

Langues

eng

Pagination

1-12

Informations de copyright

AJNMMI Copyright © 2024.

Déclaration de conflit d'intérêts

N.V. is a co-founder of MedChem Imaging, Inc., S.K. was an employee of Eisai Inc. when the work was undertaken, and A.C. and P.S. are currently employees of Eisai Inc.

Auteurs

Faustine d'Orchymont (F)

Azrieli Centre for Neuro-Radiochemistry, Brain Health Imaging Centre, Centre for Addiction and Mental Health (CAMH) Toronto, ON, Canada.

Andrea Narvaez (A)

Azrieli Centre for Neuro-Radiochemistry, Brain Health Imaging Centre, Centre for Addiction and Mental Health (CAMH) Toronto, ON, Canada.
Enigma Biomedical Group, Inc. Toronto, ON, Canada.

Roger Raymond (R)

Azrieli Centre for Neuro-Radiochemistry, Brain Health Imaging Centre, Centre for Addiction and Mental Health (CAMH) Toronto, ON, Canada.

Pallavi Sachdev (P)

Eisai, Inc. Nutley, NJ, USA.

Arnaud Charil (A)

Eisai, Inc. Nutley, NJ, USA.

Stephen Krause (S)

Eisai, Inc. Nutley, NJ, USA.

Neil Vasdev (N)

Azrieli Centre for Neuro-Radiochemistry, Brain Health Imaging Centre, Centre for Addiction and Mental Health (CAMH) Toronto, ON, Canada.
Department of Psychiatry, University of Toronto Toronto, ON, Canada.

Classifications MeSH