Muscarinic Receptor Activators as Novel Treatments for Schizophrenia.

KarXT acetylcholine and xanomeline antipsychotic muscarinic schizophrenia

Journal

Biological psychiatry
ISSN: 1873-2402
Titre abrégé: Biol Psychiatry
Pays: United States
ID NLM: 0213264

Informations de publication

Date de publication:
25 Mar 2024
Historique:
received: 17 11 2023
revised: 08 03 2024
accepted: 17 03 2024
medline: 28 3 2024
pubmed: 28 3 2024
entrez: 27 3 2024
Statut: aheadofprint

Résumé

Achieving optimal treatment outcomes for individuals living with schizophrenia remains challenging, despite 70 years of drug development efforts. Many chemically distinct antipsychotics have been developed over the past seven decades with improved safety and tolerability but with only slight variation in efficacy. All currently prescribed antipsychotics act as antagonists or partial agonists at the dopamine D

Identifiants

pubmed: 38537670
pii: S0006-3223(24)01173-9
doi: 10.1016/j.biopsych.2024.03.014
pii:
doi:

Types de publication

Journal Article Review

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

Copyright © 2024. Published by Elsevier Inc.

Auteurs

Steven M Paul (SM)

Karuna Therapeutics, Boston, MA, USA; Department of Psychiatry and Neurology, Washington University of St. Louis, St. Louis, MO, USA. Electronic address: spaul@karunatx.com.

Samantha E Yohn (SE)

Karuna Therapeutics, Boston, MA, USA.

Stephen K Brannan (SK)

Karuna Therapeutics, Boston, MA, USA.

Nichole M Neugebauer (NM)

Karuna Therapeutics, Boston, MA, USA.

Alan Breier (A)

Department of Psychiatry, Indiana University School of Medicine, Indianapolis, IN, USA.

Classifications MeSH