Astemizole, a Second-Generation Histamine H1-Receptor Antagonist, Did Not Attenuate the Aggregation Process of α-Synuclein In Vitro.

Parkinson’s disease amyloid astemizole synuclein

Journal

Biomedicines
ISSN: 2227-9059
Titre abrégé: Biomedicines
Pays: Switzerland
ID NLM: 101691304

Informations de publication

Date de publication:
08 Mar 2024
Historique:
received: 30 12 2023
revised: 03 03 2024
accepted: 05 03 2024
medline: 28 3 2024
pubmed: 28 3 2024
entrez: 28 3 2024
Statut: epublish

Résumé

The antihistamine astemizole has shown disease-modifying effects in several preclinical disease models of Parkinson's disease (PD). Astemizole also interacts with an anomalous aggregation of Alzheimer's disease-related amyloid-β (Aβ) peptide and has inhibitory activity on the human prion protein PrP

Identifiants

pubmed: 38540224
pii: biomedicines12030611
doi: 10.3390/biomedicines12030611
pii:
doi:

Types de publication

Journal Article

Langues

eng

Subventions

Organisme : Ulsan University Hospital Research Grant
ID : UUH-2017-03
Organisme : National Research Foundation of Korea
ID : 2021R1F1A1062478

Auteurs

Jung Il Choi (JI)

Basic-Clinical Convergence Research Institute, University of Ulsan, Ulsan 44033, Republic of Korea.

Hyunjo Lee (H)

Department of Neurology, Ulsan University Hospital, University of Ulsan College of Medicine, Ulsan 44033, Republic of Korea.

Dong Jun Kim (DJ)

Basic-Clinical Convergence Research Institute, University of Ulsan, Ulsan 44033, Republic of Korea.

Eun Suk Park (ES)

Department of Neurosurgery, Wonkwang University Hospital, Wonkwang University School of Medicine, Iksan 54538, Republic of Korea.

Kyung Yeon Lee (KY)

Department of Pediatrics, Ulsan University Hospital, University of Ulsan College of Medicine, Ulsan 44033, Republic of Korea.

Hui-Jun Yang (HJ)

Basic-Clinical Convergence Research Institute, University of Ulsan, Ulsan 44033, Republic of Korea.
Department of Neurology, Ulsan University Hospital, University of Ulsan College of Medicine, Ulsan 44033, Republic of Korea.

Classifications MeSH