Influence of Molecular Design on the Tumor Targeting and Biodistribution of PSMA-Binding Tracers Labeled with Technetium-99m.

BQ0411 BQ0412 PSMA coupling linker prostate cancer prostate-specific membrane antigen single-photon emission computed tomography technetium-99m

Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
23 Mar 2024
Historique:
received: 29 02 2024
revised: 21 03 2024
accepted: 22 03 2024
medline: 13 4 2024
pubmed: 13 4 2024
entrez: 13 4 2024
Statut: epublish

Résumé

Previously, we designed the EuK-based PSMA ligand BQ0413 with an maE

Identifiants

pubmed: 38612427
pii: ijms25073615
doi: 10.3390/ijms25073615
pii:
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Swedish Cancer Society
ID : 20 0815 Pj
Organisme : Swedish Cancer Society
ID : 21 1485 Pj
Organisme : Swedish Research Council
ID : 2022-00556

Auteurs

Ekaterina Bezverkhniaia (E)

Department of Medicinal Chemistry, Uppsala University, 751 23 Uppsala, Sweden.

Panagiotis Kanellopoulos (P)

Department of Medicinal Chemistry, Uppsala University, 751 23 Uppsala, Sweden.

Ulrika Rosenström (U)

Department of Medicinal Chemistry, Uppsala University, 751 23 Uppsala, Sweden.

Vladimir Tolmachev (V)

Department of Immunology, Genetics and Pathology, Uppsala University, 752 37 Uppsala, Sweden.

Anna Orlova (A)

Department of Medicinal Chemistry, Uppsala University, 751 23 Uppsala, Sweden.
Science for Life Laboratory, Uppsala University, 752 37 Uppsala, Sweden.

Classifications MeSH