Preparation, characterisation, pharmacokinetics and distribution of esculin microspheres administered via intravitreal injection into rabbit brain.

Esculin Parkinson’s disease brain targeting intravitreal injection microspheres

Journal

Xenobiotica; the fate of foreign compounds in biological systems
ISSN: 1366-5928
Titre abrégé: Xenobiotica
Pays: England
ID NLM: 1306665

Informations de publication

Date de publication:
19 Apr 2024
Historique:
medline: 19 4 2024
pubmed: 19 4 2024
entrez: 19 4 2024
Statut: aheadofprint

Résumé

This study explored the distribution of esculin microspheres in rabbit brain tissue following intravitreal injection and investigated the possibility of direct entry of the drug into the brain through the eye, to develop a formulation with enhanced therapeutic efficacy against Parkinson's disease.Chitosan microspheres of esculin were prepared

Identifiants

pubmed: 38638108
doi: 10.1080/00498254.2024.2341402
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

1-15

Auteurs

Danqing Wu (D)

Department of Pharmaceutics, College of Pharmacy, Anhui University of Chinese Medicine, Hefei, China.

Rui Luo (R)

Department of Pharmaceutics, College of Pharmacy, Anhui University of Chinese Medicine, Hefei, China.

Yangnan Chen (Y)

Department of Pharmaceutics, College of Pharmacy, Anhui University of Chinese Medicine, Hefei, China.

Zhiyun Zheng (Z)

Department of Pharmaceutics, College of Pharmacy, Anhui University of Chinese Medicine, Hefei, China.
Institute of Pharmaceutics, Anhui Academy of Chinese Medical Sciences, Hefei, China.
Anhui Province Key Laboratory of Pharmaceutical Preparation Technology and Application, Hefei, China.

Shuangying Gui (S)

Department of Pharmaceutics, College of Pharmacy, Anhui University of Chinese Medicine, Hefei, China.
Institute of Pharmaceutics, Anhui Academy of Chinese Medical Sciences, Hefei, China.
Anhui Province Key Laboratory of Pharmaceutical Preparation Technology and Application, Hefei, China.

Ning He (N)

Department of Pharmaceutics, College of Pharmacy, Anhui University of Chinese Medicine, Hefei, China.
Institute of Pharmaceutics, Anhui Academy of Chinese Medical Sciences, Hefei, China.
Anhui Province Key Laboratory of Pharmaceutical Preparation Technology and Application, Hefei, China.

Classifications MeSH