Discovery and development of macrocyclic peptide modulators of the cannabinoid 2 receptor.

G protein-coupled receptor allosteric modulator cannabinoid type 2 receptor peptide plant

Journal

The Journal of biological chemistry
ISSN: 1083-351X
Titre abrégé: J Biol Chem
Pays: United States
ID NLM: 2985121R

Informations de publication

Date de publication:
26 Apr 2024
Historique:
received: 21 02 2024
revised: 15 04 2024
accepted: 23 04 2024
medline: 29 4 2024
pubmed: 29 4 2024
entrez: 28 4 2024
Statut: aheadofprint

Résumé

The cannabinoid-type 2 receptor (CB

Identifiants

pubmed: 38679329
pii: S0021-9258(24)01831-3
doi: 10.1016/j.jbc.2024.107330
pii:
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

107330

Informations de copyright

Copyright © 2024 The Authors. Published by Elsevier Inc. All rights reserved.

Auteurs

Nataša Tomašević (N)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.

Fabiola Susanna Emser (FS)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.

Edin Muratspahić (E)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.

Jasmin Gattringer (J)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.

Simon Hasinger (S)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.

Roland Hellinger (R)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria.

Peter Keov (P)

Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, 3052, Australia; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville 3052, VIC, Australia.

Manuel Felkl (M)

Institute of Biological Chemistry, Faculty of Chemistry, University of Vienna, 1090 Vienna, Austria.

Jürg Gertsch (J)

Institute of Biochemistry and Molecular Medicine, University of Bern, 3012 Bern, Switzerland.

Christian F W Becker (CFW)

Institute of Biological Chemistry, Faculty of Chemistry, University of Vienna, 1090 Vienna, Austria.

Christian W Gruber (CW)

Center for Physiology and Pharmacology, Institute of Pharmacology, Medical University of Vienna, 1090 Vienna, Austria. Electronic address: christian.w.gruber@meduniwien.ac.at.

Classifications MeSH