Synthon Approach in Crystal Engineering to Modulate Physicochemical Properties in Organic Salts of Chlorpropamide.

bioavailability cocrystal salt cocrystal salt hydrate conformational adjustment and conformational changes crystal packing dissolution hydrogen bonding pharmacokinetics salt solubility

Journal

Molecular pharmaceutics
ISSN: 1543-8392
Titre abrégé: Mol Pharm
Pays: United States
ID NLM: 101197791

Informations de publication

Date de publication:
30 Apr 2024
Historique:
medline: 30 4 2024
pubmed: 30 4 2024
entrez: 30 4 2024
Statut: aheadofprint

Résumé

The formulation of drug with improved bioavailability is always challenging and indispensable in the field of pharmaceutics. The control of intermolecular interactions via crystal engineering approach and solid-state molecular recognition results in the formation of active drug molecules with modulated pharmacological benefits. Therefore, with the aim to improve the solubility and dissolution rate of the drug chlorpropamide (

Identifiants

pubmed: 38688017
doi: 10.1021/acs.molpharmaceut.4c00043
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Auteurs

Anila M Menon (AM)

Department of Chemistry, IISER Bhopal, Bhopal Bypass Road, Bhopal, Madhya Pradesh 462066, India.

Nagamalli Naga Sidhartha (NN)

Department of Pharmaceutical Analysis, NIPER Hyderabad, Balanagar, Hyderabad, Telangana 500037, India.

Ipsha Shruti (I)

Department of Chemistry, IISER Bhopal, Bhopal Bypass Road, Bhopal, Madhya Pradesh 462066, India.

Ajay Suresh (A)

Department of Chemistry, IISER Bhopal, Bhopal Bypass Road, Bhopal, Madhya Pradesh 462066, India.

Ravindra Meena (R)

Department of Chemistry, IISER Bhopal, Bhopal Bypass Road, Bhopal, Madhya Pradesh 462066, India.

Amol G Dikundwar (AG)

Department of Pharmaceutical Analysis, NIPER Hyderabad, Balanagar, Hyderabad, Telangana 500037, India.

Deepak Chopra (D)

Department of Chemistry, IISER Bhopal, Bhopal Bypass Road, Bhopal, Madhya Pradesh 462066, India.

Classifications MeSH