Conformational analysis and spectroscopic properties of antichagasic nifurtimox.

Conformational analysis Density functional theory Mid-infrared spectroscopy Nifurtimox UV–VIS spectroscopy

Journal

Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy
ISSN: 1873-3557
Titre abrégé: Spectrochim Acta A Mol Biomol Spectrosc
Pays: England
ID NLM: 9602533

Informations de publication

Date de publication:
26 Apr 2024
Historique:
received: 09 09 2023
revised: 27 03 2024
accepted: 23 04 2024
medline: 2 5 2024
pubmed: 2 5 2024
entrez: 1 5 2024
Statut: aheadofprint

Résumé

Considering the health relevance of Chagas' disease, recent research efforts have focused on developing more efficient drug delivery systems containing nifurtimox (NFX). This paper comprehensively investigates NFX through conformational analysis and spectroscopic characterization. Using a conformer-rotamer ensemble sampling tool (CREST-xtb), five distinct conformers of NFX were sampled within a 3.0 kcal mol

Identifiants

pubmed: 38692105
pii: S1386-1425(24)00512-2
doi: 10.1016/j.saa.2024.124346
pii:
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

124346

Informations de copyright

Copyright © 2024. Published by Elsevier B.V.

Déclaration de conflit d'intérêts

Declaration of competing interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Idejan P Gross (IP)

Laboratory of Food, Drug, and Cosmetics (LTMAC), School of Health Sciences, University of Brasilia, 70.910-900 Brasília, DF, Brazil. Electronic address: gross.idejan@gmail.com.

Ana Luiza Lima (AL)

Laboratory of Food, Drug, and Cosmetics (LTMAC), School of Health Sciences, University of Brasilia, 70.910-900 Brasília, DF, Brazil.

Giselle R Bedogni (GR)

Pharmaceutical Technical Area, Department of Pharmacy, Faculty of Biochemical and Pharmaceutical Sciences, National University of Rosario, Rosario, Argentina; National Council for Scientific and Technical Research, Godoy Cruz, Argentina.

Livia Sa-Barreto (L)

Laboratory of Food, Drug, and Cosmetics (LTMAC), School of Health Sciences, University of Brasilia, 70.910-900 Brasília, DF, Brazil.

Tais Gratieri (T)

Laboratory of Food, Drug, and Cosmetics (LTMAC), School of Health Sciences, University of Brasilia, 70.910-900 Brasília, DF, Brazil.

Guilherme M Gelfuso (GM)

Laboratory of Food, Drug, and Cosmetics (LTMAC), School of Health Sciences, University of Brasilia, 70.910-900 Brasília, DF, Brazil.

Claudio J Salomon (CJ)

Pharmaceutical Technical Area, Department of Pharmacy, Faculty of Biochemical and Pharmaceutical Sciences, National University of Rosario, Rosario, Argentina; National Council for Scientific and Technical Research, Godoy Cruz, Argentina. Electronic address: csalomon@fbioyf.unr.edu.ar.

Marcílio Cunha-Filho (M)

Laboratory of Food, Drug, and Cosmetics (LTMAC), School of Health Sciences, University of Brasilia, 70.910-900 Brasília, DF, Brazil.

Classifications MeSH