Structural analysis of the peptidoglycan DL-endopeptidase CwlO complexed with its inhibitory protein IseA.

hydrophobic pocket for IseA binding inhibition of DL‐endopeptidase peptidoglycan degradation

Journal

The FEBS journal
ISSN: 1742-4658
Titre abrégé: FEBS J
Pays: England
ID NLM: 101229646

Informations de publication

Date de publication:
05 Jun 2024
Historique:
revised: 08 03 2024
received: 04 09 2023
accepted: 28 05 2024
medline: 6 6 2024
pubmed: 6 6 2024
entrez: 6 6 2024
Statut: aheadofprint

Résumé

Peptidoglycan DL-endopeptidases locally cleave the peptide stem of peptidoglycan in the bacterial cell wall. This process facilitates bacterial growth and division by loosening the rigid peptidoglycan layer. IseA binds to the active site of multiple DL-endopeptidases and inhibits excessive peptidoglycan degradation that leads to cell lysis. To better understand how IseA inhibits DL-endopeptidase activity, we determined the crystal structure of the peptidoglycan DL-endopeptidase CwlO/IseA complex and compared it with that of the peptidoglycan DL-endopeptidase LytE/IseA complex. Structural analyses showed significant differences between the hydrophobic pocket-binding residues of the DL-endopeptidases (F361 of CwlO and W237 of LytE). Additionally, binding assays showed that the F361 mutation of CwlO to the bulkier hydrophobic residue, tryptophan, increased its binding affinity for IseA, whereas mutation to alanine reduced the affinity. These analyses revealed that the hydrophobic pocket-binding residue of DL-endopeptidases determines IseA-binding affinity and is required for substrate-mimetic inhibition by IseA.

Identifiants

pubmed: 38840475
doi: 10.1111/febs.17197
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : National Research Foundation of Korea
ID : 2022R1A5A1031361
Organisme : National Research Foundation of Korea
ID : RS-2023-00301974
Organisme : National Research Foundation of Korea
ID : RS-2024-00334946

Informations de copyright

© 2024 Federation of European Biochemical Societies.

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Auteurs

Sudarshan Tandukar (S)

College of Pharmacy, Yeungnam University, Gyeongsan, Korea.

Eunju Kwon (E)

Division of Life Science, Gyeongsang National University, Jinju, Korea.
Research Institute of Molecular Alchemy, Gyeongsang National University, Jinju, Korea.

Dong Young Kim (DY)

College of Pharmacy, Yeungnam University, Gyeongsan, Korea.

Classifications MeSH