Asciminib is a novel inhibitor of ABL1 and ABL2 gene fusions in ALL but requires the ABL SH3 domain for efficacy.


Journal

Blood
ISSN: 1528-0020
Titre abrégé: Blood
Pays: United States
ID NLM: 7603509

Informations de publication

Date de publication:
07 Jun 2024
Historique:
accepted: 30 05 2024
received: 25 03 2024
revised: 24 05 2024
medline: 7 6 2024
pubmed: 7 6 2024
entrez: 7 6 2024
Statut: aheadofprint

Résumé

High-risk Ph-like ALL includes genomic rearrangement of the ABL1 and ABL2 genes (collectively ABL-rearranged, ABLr), and novel treatments are required. For the first time, we demonstrate asciminib efficacy in ABLr ALL, but only when the ABL SH3 domain is present.

Identifiants

pubmed: 38848536
pii: 516435
doi: 10.1182/blood.2024024776
pii:
doi:

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

Copyright © 2024 American Society of Hematology.

Auteurs

Laura N Eadie (LN)

South Australian Health and Medical Research Institute, Adelaide, Australia.

Elias Lagonik (E)

South Australian Health and Medical Research Institute, Adelaide, Australia.

Elyse C Page (EC)

South Australian Health and Medical Research Institute, Adelaide, Australia.

Caitlin E Schutz (CE)

South Australian Health and Medical Research Institute, Adelaide, Australia.

Susan L Heatley (SL)

South Australian Health & Medical Research Institute, Adelaide, Australia.

Barbara J McClure (BJ)

The University of Adelaide, Australia.

Michelle Olivia Forgione (MO)

South Australian Health and Medical Research Institute, Adelaide, Australia.

David T Yeung (DT)

South Australian Health and Medical Research Institute, Adelaide, Australia.

Timothy P Hughes (TP)

South Australian Health and Medical Research Institute, Adelaide, Australia.

Classifications MeSH