Mixed responses to targeted therapy driven by chromosomal instability through p53 dysfunction and genome doubling.


Journal

Nature communications
ISSN: 2041-1723
Titre abrégé: Nat Commun
Pays: England
ID NLM: 101528555

Informations de publication

Date de publication:
13 Jun 2024
Historique:
received: 12 09 2023
accepted: 28 03 2024
medline: 14 6 2024
pubmed: 14 6 2024
entrez: 13 6 2024
Statut: epublish

Résumé

The phenomenon of mixed/heterogenous treatment responses to cancer therapies within an individual patient presents a challenging clinical scenario. Furthermore, the molecular basis of mixed intra-patient tumor responses remains unclear. Here, we show that patients with metastatic lung adenocarcinoma harbouring co-mutations of EGFR and TP53, are more likely to have mixed intra-patient tumor responses to EGFR tyrosine kinase inhibition (TKI), compared to those with an EGFR mutation alone. The combined presence of whole genome doubling (WGD) and TP53 co-mutations leads to increased genome instability and genomic copy number aberrations in genes implicated in EGFR TKI resistance. Using mouse models and an in vitro isogenic p53-mutant model system, we provide evidence that WGD provides diverse routes to drug resistance by increasing the probability of acquiring copy-number gains or losses relative to non-WGD cells. These data provide a molecular basis for mixed tumor responses to targeted therapy, within an individual patient, with implications for therapeutic strategies.

Identifiants

pubmed: 38871738
doi: 10.1038/s41467-024-47606-9
pii: 10.1038/s41467-024-47606-9
doi:

Substances chimiques

Tumor Suppressor Protein p53 0
ErbB Receptors EC 2.7.10.1
TP53 protein, human 0
Protein Kinase Inhibitors 0
EGFR protein, human EC 2.7.10.1

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

4871

Subventions

Organisme : Wellcome Trust
ID : FC001169
Pays : United Kingdom
Organisme : Cancer Research UK (CRUK)
ID : C416/A21999
Organisme : Cancer Research UK (CRUK)
ID : C11496/A30025
Organisme : Wellcome Trust
ID : FC001169
Pays : United Kingdom
Organisme : Wellcome Trust
ID : FC001169
Pays : United Kingdom
Organisme : Royal Society
ID : RSRP\R\210001
Organisme : Novo Nordisk Fonden (Novo Nordisk Foundation)
ID : ID16584
Organisme : EC | EC Seventh Framework Programm | FP7 Ideas: European Research Council (FP7-IDEAS-ERC - Specific Programme: "Ideas" Implementing the Seventh Framework Programme of the European Community for Research, Technological Development and Demonstration Activities (2007 to 2013))
ID : 617844
Organisme : EC | EC Seventh Framework Programm | FP7 Ideas: European Research Council (FP7-IDEAS-ERC - Specific Programme: "Ideas" Implementing the Seventh Framework Programme of the European Community for Research, Technological Development and Demonstration Activities (2007 to 2013))
ID : 617844
Organisme : EC | Horizon 2020 Framework Programme (EU Framework Programme for Research and Innovation H2020)
ID : 835297
Organisme : EC | Horizon 2020 Framework Programme (EU Framework Programme for Research and Innovation H2020)
ID : 835297
Organisme : EC | Horizon 2020 Framework Programme (EU Framework Programme for Research and Innovation H2020)
ID : 835297

Investigateurs

Jason F Lester (JF)
Amrita Bajaj (A)
Apostolos Nakas (A)
Azmina Sodha-Ramdeen (A)
Mohamad Tufail (M)
Molly Scotland (M)
Rebecca Boyles (R)
Sridhar Rathinam (S)
Claire Wilson (C)
Domenic Marrone (D)
Sean Dulloo (S)
Dean A Fennell (DA)
Gurdeep Matharu (G)
Jacqui A Shaw (JA)
Ekaterini Boleti (E)
Heather Cheyne (H)
Mohammed Khalil (M)
Shirley Richardson (S)
Tracey Cruickshank (T)
Gillian Price (G)
Keith M Kerr (KM)
Sarah Benafif (S)
Jack French (J)
Kayleigh Gilbert (K)
Babu Naidu (B)
Akshay J Patel (AJ)
Aya Osman (A)
Carol Enstone (C)
Gerald Langman (G)
Helen Shackleford (H)
Madava Djearaman (M)
Salma Kadiri (S)
Gary Middleton (G)
Angela Leek (A)
Jack Davies Hodgkinson (JD)
Nicola Totton (N)
Angeles Montero (A)
Elaine Smith (E)
Eustace Fontaine (E)
Felice Granato (F)
Antonio Paiva-Correia (A)
Juliette Novasio (J)
Kendadai Rammohan (K)
Leena Joseph (L)
Paul Bishop (P)
Rajesh Shah (R)
Stuart Moss (S)
Vijay Joshi (V)
Philip A J Crosbie (PAJ)
Katherine D Brown (KD)
Mathew Carter (M)
Anshuman Chaturvedi (A)
Pedro Oliveira (P)
Colin R Lindsay (CR)
Fiona H Blackhall (FH)
Matthew G Krebs (MG)
Yvonne Summers (Y)
Alexandra Clipson (A)
Jonathan Tugwood (J)
Alastair Kerr (A)
Dominic G Rothwell (DG)
Caroline Dive (C)
Hugo J W L Aerts (HJWL)
Roland F Schwarz (RF)
Tom L Kaufmann (TL)
Gareth A Wilson (GA)
Rachel Rosenthal (R)
Peter Van Loo (P)
Nicolai J Birkbak (NJ)
Zoltan Szallasi (Z)
Judit Kisistok (J)
Mateo Sokac (M)
Roberto Salgado (R)
Miklos Diossy (M)
Jonas Demeulemeester (J)
Abigail Bunkum (A)
Angela Dwornik (A)
Alastair Magness (A)
Andrew J Rowan (AJ)
Angeliki Karamani (A)
Antonia Toncheva (A)
Benny Chain (B)
Carla Castignani (C)
Chris Bailey (C)
Christopher Abbosh (C)
Clare Puttick (C)
Clare E Weeden (CE)
Claudia Lee (C)
Corentin Richard (C)
Cristina Naceur-Lombardelli (C)
David R Pearce (DR)
Despoina Karagianni (D)
Dhruva Biswas (D)
Dina Levi (D)
Elizabeth Larose Cadieux (E)
Emilia L Lim (EL)
Emma Colliver (E)
Emma Nye (E)
Felip Gálvez-Cancino (F)
Francisco Gimeno-Valiente (F)
George Kassiotis (G)
Georgia Stavrou (G)
Gerasimos-Theodoros Mastrokalos (GT)
Helen L Lowe (HL)
Ignacio Garcia Matos (IG)
Imran Noorani (I)
Jacki Goldman (J)
James L Reading (JL)
Jayant K Rane (JK)
Jerome Nicod (J)
John A Hartley (JA)
Karl S Peggs (KS)
Katey S S Enfield (KSS)
Kayalvizhi Selvaraju (K)
Kerstin Thol (K)
Kevin W Ng (KW)
Kezhong Chen (K)
Krijn Dijkstra (K)
Kristiana Grigoriadis (K)
Krupa Thakkar (K)
Leah Ensell (L)
Mansi Shah (M)
Maria Litovchenko (M)
Mariam Jamal-Hanjani (M)
Mariana Werner Sunderland (M)
Matthew R Huska (MR)
Mark S Hill (MS)
Michelle Dietzen (M)
Michelle M Leung (MM)
Mickael Escudero (M)
Miljana Tanić (M)
Monica Sivakumar (M)
Olga Chervova (O)
Olivia Lucas (O)
Oriol Pich (O)
Othman Al-Sawaf (O)
Paulina Prymas (P)
Philip Hobson (P)
Piotr Pawlik (P)
Richard Kevin Stone (RK)
Robert Bentham (R)
Roberto Vendramin (R)
Sadegh Saghafinia (S)
Samuel Gamble (S)
Selvaraju Veeriah (S)
Seng Kuong Anakin Ung (SKA)
Sergio A Quezada (SA)
Sharon Vanloo (S)
Sonya Hessey (S)
Sophia Ward (S)
Sian Harries (S)
Stefan Boeing (S)
Stephan Beck (S)
Supreet Kaur Bola (SK)
Takahiro Karasaki (T)
Tamara Denner (T)
Teresa Marafioti (T)
Thomas Patrick Jones (TP)
Victoria Spanswick (V)
Vittorio Barbè (V)
Wei-Ting Lu (WT)
Wing Kin Liu (WK)
Yin Wu (Y)
Yutaka Naito (Y)
Zoe Ramsden (Z)
Catarina Veiga (C)
Gary Royle (G)
Charles-Antoine Collins-Fekete (CA)
Francesco Fraioli (F)
Paul Ashford (P)
Martin D Forster (MD)
Siow Ming Lee (SM)
Elaine Borg (E)
Mary Falzon (M)
Dionysis Papadatos-Pastos (D)
James Wilson (J)
Tanya Ahmad (T)
Alexander James Procter (AJ)
Asia Ahmed (A)
Magali N Taylor (MN)
Arjun Nair (A)
David Lawrence (D)
Davide Patrini (D)
Neal Navani (N)
Ricky M Thakrar (RM)
Sam M Janes (SM)
Emilie Martinoni Hoogenboom (E)
Fleur Monk (F)
James W Holding (JW)
Junaid Choudhary (J)
Kunal Bhakhri (K)
Marco Scarci (M)
Pat Gorman (P)
Reena Khiroya (R)
Robert C M Stephens (RCM)
Yien Ning Sophia Wong (YNS)
Zoltan Kaplar (Z)
Steve Bandula (S)
Allan Hackshaw (A)
Anne-Marie Hacker (AM)
Abigail Sharp (A)
Sean Smith (S)
Harjot Kaur Dhanda (H)
Camilla Pilotti (C)
Rachel Leslie (R)
Anca Grapa (A)
Hanyun Zhang (H)
Khalid AbdulJabbar (K)
Xiaoxi Pan (X)
Yinyin Yuan (Y)
David Chuter (D)
Mairead MacKenzie (M)
Serena Chee (S)
Aiman Alzetani (A)
Judith Cave (J)
Jennifer Richards (J)
Eric Lim (E)
Paulo De Sousa (P)
Simon Jordan (S)
Alexandra Rice (A)
Hilgardt Raubenheimer (H)
Harshil Bhayani (H)
Lyn Ambrose (L)
Anand Devaraj (A)
Hema Chavan (H)
Sofina Begum (S)
Silviu I Buderi (SI)
Daniel Kaniu (D)
Mpho Malima (M)
Sarah Booth (S)
Andrew G Nicholson (AG)
Nadia Fernandes (N)
Pratibha Shah (P)
Chiara Proli (C)
Madeleine Hewish (M)
Sarah Danson (S)
Michael J Shackcloth (MJ)
Lily Robinson (L)
Peter Russell (P)
Kevin G Blyth (KG)
Andrew Kidd (A)
Craig Dick (C)
John Le Quesne (J)
Alan Kirk (A)
Mo Asif (M)
Rocco Bilancia (R)
Nikos Kostoulas (N)
Mathew Thomas (M)

Informations de copyright

© 2024. The Author(s).

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Auteurs

Sebastijan Hobor (S)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Maise Al Bakir (M)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Crispin T Hiley (CT)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Department of Medical Oncology, University College London Hospitals, 235 Euston Rd, Fitzrovia, London, NW1 2BU, UK.

Marcin Skrzypski (M)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Department of Medical Oncology, University College London Hospitals, 235 Euston Rd, Fitzrovia, London, NW1 2BU, UK.
Department of Oncology and Radiotherapy, Medical University of Gdańsk, ul. Mariana Smoluchowskiego 17, 80-214, Gdańsk, Poland.

Alexander M Frankell (AM)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.

Bjorn Bakker (B)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
European Research Institute for the Biology of Ageing, University of Groningen, University Medical Center Groningen, A. Deusinglaan 1, Groningen, 9713, the Netherlands.

Thomas B K Watkins (TBK)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Aleksandra Markovets (A)

Oncology Data Science, Oncology R&D, AstraZeneca, Boston, MA, USA.

Jonathan R Dry (JR)

Late Development, Oncology R&D, AstraZeneca, Boston, MA, USA.

Andrew P Brown (AP)

Late Development, Oncology R&D, AstraZeneca, Boston, MA, USA.

Jasper van der Aart (J)

Research and Early Development, Oncology R&D, AstraZeneca, Cambridge, UK.

Hilda van den Bos (H)

European Research Institute for the Biology of Ageing, University of Groningen, University Medical Center Groningen, A. Deusinglaan 1, Groningen, 9713, the Netherlands.

Diana Spierings (D)

European Research Institute for the Biology of Ageing, University of Groningen, University Medical Center Groningen, A. Deusinglaan 1, Groningen, 9713, the Netherlands.

Dahmane Oukrif (D)

Research Department of Pathology, University College London Medical School, University Street, London, WC1E 6JJ, UK.

Marco Novelli (M)

Research Department of Pathology, University College London Medical School, University Street, London, WC1E 6JJ, UK.

Turja Chakrabarti (T)

Department of Medicine, University of California, San Francisco, CA, 94158, USA.

Adam H Rabinowitz (AH)

Furlong Laboratory, EMBL Meyerhofstraße 1, 69117, Heidelberg, Germany.

Laila Ait Hassou (L)

European Organization for Research and Treatment of Cancer, Brussels, Belgium.

Saskia Litière (S)

Bioinformatics & Biostatistics; Francis Crick Institute, London, UK.

D Lucas Kerr (DL)

Department of Medicine, University of California, San Francisco, CA, 94158, USA.

Lisa Tan (L)

Department of Medicine, University of California, San Francisco, CA, 94158, USA.

Gavin Kelly (G)

Bioinformatics & Biostatistics; Francis Crick Institute, London, UK.

David A Moore (DA)

Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Department of Cellular Pathology, University College London Hospitals, London, UK.

Matthew J Renshaw (MJ)

Advanced Light Microscopy, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Subramanian Venkatesan (S)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

William Hill (W)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Ariana Huebner (A)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Cancer Genome Evolution Research Group, Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, London, UK.

Carlos Martínez-Ruiz (C)

Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Cancer Genome Evolution Research Group, Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, London, UK.

James R M Black (JRM)

Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Cancer Genome Evolution Research Group, Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, London, UK.

Wei Wu (W)

Department of Medicine, University of California, San Francisco, CA, 94158, USA.

Mihaela Angelova (M)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Nicholas McGranahan (N)

Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.
Cancer Genome Evolution Research Group, Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, London, UK.

Julian Downward (J)

Oncogene Biology Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Juliann Chmielecki (J)

Late Development, Oncology R&D, AstraZeneca, Boston, MA, USA.

Carl Barrett (C)

Late Development, Oncology R&D, AstraZeneca, Boston, MA, USA.

Kevin Litchfield (K)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Su Kit Chew (SK)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.

Collin M Blakely (CM)

Department of Medicine, University of California, San Francisco, CA, 94158, USA.

Elza C de Bruin (EC)

Research and Early Development, Oncology R&D, AstraZeneca, Cambridge, UK.

Floris Foijer (F)

European Research Institute for the Biology of Ageing, University of Groningen, University Medical Center Groningen, A. Deusinglaan 1, Groningen, 9713, the Netherlands.

Karen H Vousden (KH)

p53 and Metabolism Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.

Trever G Bivona (TG)

Department of Medicine, University of California, San Francisco, CA, 94158, USA.
Chan-Zuckerberg Biohub, San Francisco, USA.

Robert E Hynds (RE)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK.

Nnennaya Kanu (N)

Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK. n.kanu@ucl.ac.uk.

Simone Zaccaria (S)

Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK. s.zaccaria@ucl.ac.uk.
Computational Cancer Genomics Research Group, University College London Cancer Institute, London, UK. s.zaccaria@ucl.ac.uk.

Eva Grönroos (E)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK. Eva.Gronroos@crick.ac.uk.

Charles Swanton (C)

Cancer Evolution and Genome Instability Laboratory, The Francis Crick Institute, 1 Midland Rd, London, NW1 1AT, UK. Charles.Swanton@crick.ac.uk.
Cancer Research UK Lung Cancer Centre of Excellence, University College London Cancer Institute, Paul O'Gorman Building, 72 Huntley Street, London, WC1E 6BT, UK. Charles.Swanton@crick.ac.uk.
Department of Medical Oncology, University College London Hospitals, 235 Euston Rd, Fitzrovia, London, NW1 2BU, UK. Charles.Swanton@crick.ac.uk.

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