Synthesis and Enzymatic Evaluation of a Small Library of Substituted Phenylsulfonamido-Alkyl Sulfamates towards Carbonic Anhydrase II.

Carbonic Anhydrase II / antagonists & inhibitors Carbonic Anhydrase Inhibitors / chemistry Sulfonic Acids / chemistry Animals Cattle Structure-Activity Relationship Sulfonamides / chemistry Small Molecule Libraries / chemistry Molecular Structure
carbonic anhydrase II inhibitor sulfamates

Journal

Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009

Informations de publication

Date de publication:
25 Jun 2024
Historique:
received: 13 05 2024
revised: 19 06 2024
accepted: 20 06 2024
medline: 13 7 2024
pubmed: 13 7 2024
entrez: 13 7 2024
Statut: epublish

Résumé

A small library of 79 substituted phenylsulfonamidoalkyl sulfamates,

Identifiants

DOI: 10.3390/molecules29133015 PMID: 38998967
pubmed: 38998967
pii: molecules29133015
doi: 10.3390/molecules29133015
pii:
doi:

Substances chimiques

Carbonic Anhydrase II EC 4.2.1.-
Carbonic Anhydrase Inhibitors 0
Sulfonic Acids 0
Sulfonamides 0
sulfamic acid 9NFU33906Q
Small Molecule Libraries 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Auteurs

Toni C Denner (TC)

Organic Chemistry, Martin-Luther University Halle-Wittenberg, Kurt-Mothes, Str. 2, D-06120 Halle (Saale), Germany.
ORCID: 0000-0003-0191-5651

Niels V Heise (NV)

Organic Chemistry, Martin-Luther University Halle-Wittenberg, Kurt-Mothes, Str. 2, D-06120 Halle (Saale), Germany.
ORCID: 0000-0002-6540-6357

Ahmed Al-Harrasi (A)

Natural & Medical Sciences Research Center, University of Nizwa, Nizwa 616, Oman.
ORCID: 0000-0002-0815-5942

René Csuk (R)

Organic Chemistry, Martin-Luther University Halle-Wittenberg, Kurt-Mothes, Str. 2, D-06120 Halle (Saale), Germany.
ORCID: 0000-0001-7911-290X

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Classifications MeSH

questionsmedicales.fr › Enzymes et coenzymes › Enzymes › Lyases › Carbon-oxygen lyases › Hydro-lyases › Carbonic anhydrases › Carbonic anhydrase II › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Actions chimiques et utilisations › Actions pharmacologiques › Mécanismes moléculaires de l'action pharmacologique › Antienzymes › Inhibiteurs de l'anhydrase carbonique › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Composés chimiques organiques › Composés du soufre › Acides du soufre › Acides sulfoniques › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Eucaryotes › Animaux › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Eucaryotes › Animaux › Chordés › Vertébrés › Mammifères › Eutheria › Artiodactyla › Ruminants › Bovins › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Phénomènes physiologiques › Phénomènes pharmacologiques et toxicologiques › Phénomènes pharmacologiques › Relation structure-activité › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Composés chimiques organiques › Composés du soufre › Sulfones › Sulfonamides › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Bibliothèques de petites molécules › Synthesis and Enzymatic Evaluation of a Small...
questionsmedicales.fr › Phénomènes chimiques › Structure moléculaire › Synthesis and Enzymatic Evaluation of a Small...