Molecular subtypes explain lupus epigenomic heterogeneity unveiling new regulatory genetic risk variants.


Journal

NPJ genomic medicine
ISSN: 2056-7944
Titre abrégé: NPJ Genom Med
Pays: England
ID NLM: 101685193

Informations de publication

Date de publication:
16 Jul 2024
Historique:
received: 03 04 2023
accepted: 17 05 2024
medline: 17 7 2024
pubmed: 17 7 2024
entrez: 16 7 2024
Statut: epublish

Résumé

The heterogeneity of systemic lupus erythematosus (SLE) can be explained by epigenetic alterations that disrupt transcriptional programs mediating environmental and genetic risk. This study evaluated the epigenetic contribution to SLE heterogeneity considering molecular and serological subtypes, genetics and transcriptional status, followed by drug target discovery. We performed a stratified epigenome-wide association studies of whole blood DNA methylation from 213 SLE patients and 221 controls. Methylation quantitative trait loci analyses, cytokine and transcription factor activity - epigenetic associations and methylation-expression correlations were conducted. New drug targets were searched for based on differentially methylated genes. In a stratified approach, a total of 974 differential methylation CpG sites with dependency on molecular subtypes and autoantibody profiles were found. Mediation analyses suggested that SLE-associated SNPs in the HLA region exert their risk through DNA methylation changes. Novel genetic variants regulating DNAm in disease or in specific molecular contexts were identified. The epigenetic landscapes showed strong association with transcription factor activity and cytokine levels, conditioned by the molecular context. Epigenetic signals were enriched in known and novel drug targets for SLE. This study reveals possible genetic drivers and consequences of epigenetic variability on SLE heterogeneity and disentangles the DNAm mediation role on SLE genetic risk and novel disease-specific meQTLs. Finally, novel targets for drug development were discovered.

Identifiants

pubmed: 39013887
doi: 10.1038/s41525-024-00420-0
pii: 10.1038/s41525-024-00420-0
doi:

Types de publication

Journal Article

Langues

eng

Pagination

38

Investigateurs

Lorenzo Beretta (L)
Barbara Vigone (B)
Jacques-Olivier Pers (JO)
Alain Saraux (A)
Valérie Devauchelle-Pensec (V)
Divi Cornec (D)
Sandrine Jousse-Joulin (S)
Bernard Lauwerys (B)
Julie Ducreux (J)
Anne-Lise Maudoux (AL)
Carlos Vasconcelos (C)
Ana Tavares (A)
Esmeralda Neves (E)
Raquel Faria (R)
Mariana Brandão (M)
Ana Campar (A)
António Marinho (A)
Fátima Farinha (F)
Isabel Almeida (I)
Miguel Angel Gonzalez-Gay Mantecón (MAG)
Ricardo Blanco Alonso (RB)
Alfonso Corrales Martínez (AC)
Ricard Cervera (R)
Ignasi Rodríguez-Pintó (I)
Gerard Espinosa (G)
Rik Lories (R)
Ellen De Langhe (E)
Nicolas Hunzelmann (N)
Doreen Belz (D)
Torsten Witte (T)
Niklas Baerlecken (N)
Georg Stummvoll (G)
Michael Zauner (M)
Michaela Lehner (M)
Eduardo Collantes (E)
Rafaela Ortega Castro (RO)
Ma Angeles Aguirre-Zamorano (MA)
Alejandro Escudero-Contreras (A)
Ma Carmen Castro-Villegas (MC)
Norberto Ortego (N)
María Concepción Fernández Roldán (MCF)
Enrique Raya (E)
Inmaculada Jiménez Moleón (IJ)
Enrique de Ramon (E)
Isabel Díaz Quintero (ID)
Pier Luigi Meroni (PL)
Maria Gerosa (M)
Tommaso Schioppo (T)
Carolina Artusi (C)
Carlo Chizzolini (C)
Aleksandra Zuber (A)
Donatienne Wynar (D)
Laszló Kovács (L)
Attila Balog (A)
Magdolna Deák (M)
Márta Bocskai (M)
Sonja Dulic (S)
Gabriella Kádár (G)
Falk Hiepe (F)
Velia Gerl (V)
Silvia Thiel (S)
Manuel Rodriguez Maresca (MR)
Antonio López-Berrio (A)
Rocío Aguilar-Quesada (R)
Héctor Navarro-Linares (H)
Montserrat Alvarez (M)
Damiana Alvarez-Errico (D)
Nancy Azevedo (N)
Nuria Barbarroja (N)
Anne Buttgereit (A)
Qingyu Cheng (Q)
Carlo Chizzolini (C)
Jonathan Cremer (J)
Aurélie De Groof (A)
Ellen De Langhe (E)
Julie Ducreux (J)
Aleksandra Dufour (A)
Velia Gerl (V)
Maria Hernandez-Fuentes (M)
Laleh Khodadadi (L)
Katja Kniesch (K)
Tianlu Li (T)
Chary Lopez-Pedrera (C)
Zuzanna Makowska (Z)
Concepción Marañón (C)
Brian Muchmore (B)
Esmeralda Neves (E)
Bénédicte Rouvière (B)
Quentin Simon (Q)
Elena Trombetta (E)
Nieves Varela (N)
Torsten Witte (T)

Informations de copyright

© 2024. The Author(s).

Références

Rider, V. et al. Gender bias in human systemic lupus erythematosus: a problem of steroid receptor action? Front. Immunol. 9, 611 (2018).
pubmed: 29643853 pmcid: 5882779 doi: 10.3389/fimmu.2018.00611
Nehar-Belaid, D. et al. Mapping systemic lupus erythematosus heterogeneity at the single-cell level. Nat. Immunol. 21, 1094–1106 (2020).
pubmed: 32747814 pmcid: 7442743 doi: 10.1038/s41590-020-0743-0
Bentham, J. et al. Genetic association analyses implicate aberrant regulation of innate and adaptive immunity genes in the pathogenesis of systemic lupus erythematosus. Nat. Genet. 47, 1457–1464 (2015).
pubmed: 26502338 pmcid: 4668589 doi: 10.1038/ng.3434
Wang, Y.-F. et al. Identification of 38 novel loci for systemic lupus erythematosus and genetic heterogeneity between ancestral groups. Nat. Commun. 12, 772 (2021).
pubmed: 33536424 pmcid: 7858632 doi: 10.1038/s41467-021-21049-y
Kariuki, S. N. et al. Trait-stratified genome-wide association study identifies novel and diverse genetic associations with serologic and cytokine phenotypes in systemic lupus erythematosus. Arthritis Res. Ther. 12, R151 (2010).
pubmed: 20659327 pmcid: 2945049 doi: 10.1186/ar3101
Chung, S. A. et al. Differential genetic associations for systemic lupus erythematosus based on anti–dsDNA autoantibody production. PLoS Genet. 7, e1001323 (2011).
pubmed: 21408207 pmcid: 3048371 doi: 10.1371/journal.pgen.1001323
Teruel, M. & Sawalha, A. H. Epigenetic variability in systemic lupus erythematosus: what we learned from genome-wide DNA methylation studies. Curr. Rheumatol. Rep. 19, 32 (2017).
pubmed: 28470479 pmcid: 5819620 doi: 10.1007/s11926-017-0657-5
Barturen, G. et al. Integrative analysis reveals a molecular stratification of systemic autoimmune diseases. Arthritis Rheumatol. https://doi.org/10.1002/art.41610 (2020).
Teruel, M. et al. Integrative epigenomics in Sjögren´s syndrome reveals novel pathways and a strong interaction between the HLA, autoantibodies and the interferon signature. Sci. Rep. 11, 23292 (2021).
pubmed: 34857786 pmcid: 8640069 doi: 10.1038/s41598-021-01324-0
Gateva, V. et al. A large-scale replication study identifies TNIP1, PRDM1, JAZF1, UHRF1BP1 and IL10 as risk loci for systemic lupus erythematosus. Nat. Genet. 41, 1228–1233 (2009).
pubmed: 19838195 pmcid: 2925843 doi: 10.1038/ng.468
Guerra, S. G., Vyse, T. J. & Cunninghame Graham, D. S. The genetics of lupus: a functional perspective. Arthritis Res. Ther. 14, 211 (2012).
pubmed: 22640752 pmcid: 3446495 doi: 10.1186/ar3844
Teruel, M. & Alarcón-Riquelme, M. E. The genetic basis of systemic lupus erythematosus: What are the risk factors and what have we learned. J. Autoimmun. 74, 161–175 (2016).
pubmed: 27522116 doi: 10.1016/j.jaut.2016.08.001
Ulff-Møller, C. J., Svendsen, A. J., Viemose, L. N. & Jacobsen, S. Concordance of autoimmune disease in a nationwide Danish systemic lupus erythematosus twin cohort. Semin. Arthritis Rheum. 47, 538–544 (2018).
pubmed: 28755788 doi: 10.1016/j.semarthrit.2017.06.007
Dupont, C., Armant, D. R. & Brenner, C. A. Epigenetics: definition, mechanisms and clinical perspective. Semin. Reprod. Med. 27, 351–357 (2009).
pubmed: 19711245 pmcid: 2791696 doi: 10.1055/s-0029-1237423
Joseph, S. et al. Epigenome-wide association study of peripheral blood mononuclear cells in systemic lupus erythematosus: Identifying DNA methylation signatures associated with interferon-related genes based on ethnicity and SLEDAI. J. Autoimmun. 96, 147–157 (2019).
pubmed: 30301579 doi: 10.1016/j.jaut.2018.09.007
Rask-Andersen, M. et al. Epigenome-wide association study reveals differential DNA methylation in individuals with a history of myocardial infarction. Hum. Mol. Genet. 25, 4739–4748 (2016).
pubmed: 28172975
Imgenberg-Kreuz, J. et al. DNA methylation mapping identifies gene regulatory effects in patients with systemic lupus erythematosus. Ann. Rheum. Dis. 77, 736–743 (2018).
pubmed: 29437559 doi: 10.1136/annrheumdis-2017-212379
Min, J. L. et al. Genomic and phenotypic insights from an atlas of genetic effects on DNA methylation. Nat. Genet. 53, 1311–1321 (2021).
pubmed: 34493871 pmcid: 7612069 doi: 10.1038/s41588-021-00923-x
Bonder, M. J. et al. Disease variants alter transcription factor levels and methylation of their binding sites. Nat. Genet. 49, 131–138 (2017).
pubmed: 27918535 doi: 10.1038/ng.3721
Rönnblom, L. & Leonard, D. Interferon pathway in SLE: one key to unlocking the mystery of the disease. Lupus Sci. Med. 6, e000270 (2019).
pubmed: 31497305 pmcid: 6703304 doi: 10.1136/lupus-2018-000270
Liu, W., Li, M., Wang, Z. & Wang, J. IFN-γ Mediates the development of systemic lupus erythematosus. Biomed. Res. Int. 2020, 7176515 (2020).
Zhu, H., Wang, G. & Qian, J. Transcription factors as readers and effectors of DNA methylation. Nat. Rev. Genet. 17, 551–565 (2016).
pubmed: 27479905 pmcid: 5559737 doi: 10.1038/nrg.2016.83
Jones, E. L., Laidlaw, S. M. & Dustin, L. B. TRIM21/Ro52 - roles in innate immunity and autoimmune disease. Front. Immunol. 12, 738473 (2021).
pubmed: 34552597 pmcid: 8450407 doi: 10.3389/fimmu.2021.738473
Lopez-Dominguez, R. et al. Transcription factor activity inference in systemic lupus erythematosus. Life 11, 299 (2021).
pubmed: 33915751 pmcid: 8065841 doi: 10.3390/life11040299
Kerick, M. et al. Expression quantitative trait locus analysis in systemic sclerosis identifies new candidate genes associated with multiple aspects of disease pathology. Arthritis Rheumatol. 73, 1288–1300 (2021).
pubmed: 33455083 doi: 10.1002/art.41657
Castell, S. D., Harman, M. F., Morón, G., Maletto, B. A. & Pistoresi-Palencia, M. C. Neutrophils which migrate to lymph nodes modulate CD4 + T cell response by a PD-L1 dependent mechanism. Front. Immunol. 10, 105 (2019).
pubmed: 30761151 pmcid: 6362305 doi: 10.3389/fimmu.2019.00105
Peng, D. et al. Common variants in or near ZNRF1, COLEC12, SCYL1BP1 and API5 are associated with diabetic retinopathy in Chinese patients with type 2 diabetes. Diabetologia 58, 1231–1238 (2015).
pubmed: 25819896 doi: 10.1007/s00125-015-3569-9
Bethunaickan, R., Berthier, C. C., Zhang, W., Kretzler, M. & Davidson, A. Comparative transcriptional profiling of 3 murine models of SLE nephritis reveals both unique and shared regulatory networks. PLoS ONE 8, e77489 (2013).
pubmed: 24167575 pmcid: 3805607 doi: 10.1371/journal.pone.0077489
Osthoff, A.-K. R. et al. 2018 EULAR recommendations for physical activity in people with inflammatory arthritis and osteoarthritis. Ann. Rheum. Dis. 77, 1251–1260 (2018).
doi: 10.1136/annrheumdis-2018-213585
Gutierrez-Arcelus, M. et al. Allele-specific expression changes dynamically during T cell activation in HLA and other autoimmune loci. Nat. Genet. 52, 247–253 (2020).
pubmed: 32066938 pmcid: 7135372 doi: 10.1038/s41588-020-0579-4
Carmona, F. D. et al. Novel identification of the IRF7 region as an anticentromere autoantibody propensity locus in systemic sclerosis. Ann. Rheum. Dis. 71, 114–119 (2012).
pubmed: 21926187 doi: 10.1136/annrheumdis-2011-200275
European Scleroderma Group†. et al. GWAS for systemic sclerosis identifies multiple risk loci and highlights fibrotic and vasculopathy pathways. Nat. Commun. 10, 4955 (2019).
doi: 10.1038/s41467-019-12760-y
Rinne, S. J. et al. Candidate predisposition variants in kaposi sarcoma as detected by whole-genome sequencing. Open Forum Infect. Dis. 6, ofz337 (2019).
pubmed: 31660331 pmcid: 6778425 doi: 10.1093/ofid/ofz337
Gutierrez-Arcelus, M., Rich, S. S. & Raychaudhuri, S. Autoimmune diseases — connecting risk alleles with molecular traits of the immune system. Nat. Rev. Genet. 17, 160–174 (2016).
pubmed: 26907721 pmcid: 4896831 doi: 10.1038/nrg.2015.33
Wang, W. et al. RUNX3 gene polymorphisms are associated with clinical features of systemic lupus erythematosus in Chinese Han population. J. Dermatol. Sci. 80, 69–71 (2015).
pubmed: 26233263 doi: 10.1016/j.jdermsci.2015.07.005
O’Reilly, S. Epigenetic regulation of RUNX3 in systemic sclerosis pathogenesis: time to target? Ann. Rheum. Dis. 78, 1149–1150 (2019).
pubmed: 31142477 doi: 10.1136/annrheumdis-2019-215648
Steegenga, W. T. et al. Genome-wide age-related changes in DNA methylation and gene expression in human PBMCs. Age (Dordr.) 36, 9648 (2014).
pubmed: 24789080 doi: 10.1007/s11357-014-9648-x
Verschoor, C. P. et al. The relation between DNA methylation patterns and serum cytokine levels in community-dwelling adults: a preliminary study. BMC Genet. 18, 57 (2017).
pubmed: 28637423 pmcid: 5480116 doi: 10.1186/s12863-017-0525-3
Hagberg, N. et al. The STAT4 SLE risk allele rs7574865[T] is associated with increased IL-12-induced IFN-γ production in T cells from patients with SLE. Ann. Rheum. Dis. 77, 1070–1077 (2018).
pubmed: 29475858 doi: 10.1136/annrheumdis-2017-212794
Liang, Y., Pan, H.-F. & Ye, D.-Q. Therapeutic potential of STAT4 in autoimmunity. Expert Opin. Ther. Targets 18, 945–960 (2014).
pubmed: 24844303 doi: 10.1517/14728222.2014.920325
Menke, J. et al. Targeting transcription factor Stat4 uncovers a role for interleukin-18 in the pathogenesis of severe lupus nephritis in mice. Kidney Int 79, 452–463 (2011).
pubmed: 20980973 doi: 10.1038/ki.2010.438
Remmers, E. F. et al. STAT4 and the risk of rheumatoid arthritis and systemic lupus erythematosus. N. Engl. J. Med. 357, 977–986 (2007).
pubmed: 17804842 pmcid: 2630215 doi: 10.1056/NEJMoa073003
Sigurdsson, S. et al. A risk haplotype of STAT4 for systemic lupus erythematosus is over-expressed, correlates with anti-dsDNA and shows additive effects with two risk alleles of IRF5. Hum. Mol. Genet. 17, 2868–2876 (2008).
pubmed: 18579578 pmcid: 2525501 doi: 10.1093/hmg/ddn184
Taylor, K. E. et al. Specificity of the STAT4 genetic association for severe disease manifestations of systemic lupus erythematosus. PLoS Genet. 4, e1000084 (2008).
pubmed: 18516230 pmcid: 2377340 doi: 10.1371/journal.pgen.1000084
Yang, W. et al. Genome-wide association study in asian populations identifies variants in ETS1 and WDFY4 associated with systemic lupus erythematosus. PLoS Genet. 6, e1000841 (2010).
pubmed: 20169177 pmcid: 2820522 doi: 10.1371/journal.pgen.1000841
Garrett-Sinha, L. A., Kearly, A. & Satterthwaite, A. B. The role of the transcription factor Ets1 in lupus and other autoimmune diseases. Crit. Rev. Immunol. 36, 485–510 (2016).
pubmed: 28845756 pmcid: 5695541 doi: 10.1615/CritRevImmunol.2017020284
Kim, C. J. et al. The transcription factor Ets1 suppresses T follicular helper type 2 cell differentiation to halt the onset of systemic lupus erythematosus. Immunity 49, 1034–1048.e8 (2018).
pubmed: 30566881 doi: 10.1016/j.immuni.2018.10.012
Shao, W.-H. & Cohen, P. L. The role of tyrosine kinases in systemic lupus erythematosus and their potential as therapeutic targets. Expert Rev. Clin. Immunol. 10, 573–582 (2014).
pubmed: 24678775 pmcid: 4249585 doi: 10.1586/1744666X.2014.893827
L, L. L. et al. Standardization procedure for flow cytometry data harmonization in prospective multicenter studies. Sci. Rep. 10, 11567–11567 (2020).
doi: 10.1038/s41598-020-68468-3
Teruel, M. et al. An integrative multi-omics approach in Sjögren’s Syndrome identifies novel genetic drivers with regulatory function and disease-specificity. medRxiv https://doi.org/10.1101/2020.09.14.20192211 (2020).
Das, S. et al. Next-generation genotype imputation service and methods. Nat. Genet. 48, 1284–1287 (2016).
pubmed: 27571263 pmcid: 5157836 doi: 10.1038/ng.3656
Loh, P.-R. et al. Reference-based phasing using the Haplotype Reference Consortium panel. Nat. Genet. 48, 1443–1448 (2016).
pubmed: 27694958 pmcid: 5096458 doi: 10.1038/ng.3679
Purcell, S. et al. PLINK: a tool set for whole-genome association and population-based linkage analyses. Am. J. Hum. Genet. 81, 559–575 (2007).
pubmed: 17701901 pmcid: 1950838 doi: 10.1086/519795
Griss, J. et al. ReactomeGSA - efficient multi-omics comparative pathway analysis. Mol. Cell Proteom. 19, 2115–2124 (2020).
doi: 10.1074/mcp.TIR120.002155
Ulgen, E., Ozisik, O. & Sezerman, O. U. pathfindR: an R package for comprehensive identification of enriched pathways in omics data through active subnetworks. Front. Genet. 10, 858 (2019).
Shabalin, A. A. Matrix eQTL: ultra fast eQTL analysis via large matrix operations. Bioinformatics 28, 1353–1358 (2012).
pubmed: 22492648 pmcid: 3348564 doi: 10.1093/bioinformatics/bts163
Martínez-Bueno, M. & Alarcón-Riquelme, M. E. Exploring impact of rare variation in systemic lupus erythematosus by a genome wide imputation approach. Front. Immunol. 10, 258 (2019).
pubmed: 30863397 pmcid: 6399402 doi: 10.3389/fimmu.2019.00258
Imai, K., Keele, L. & Yamamoto, T. Identification, inference and sensitivity analysis for causal mediation effects. Stat. Sci. 25, 51–71 (2010).
doi: 10.1214/10-STS321
Garcia-Alonso, L., Holland, C. H., Ibrahim, M. M., Turei, D. & Saez-Rodriguez, J. Benchmark and integration of resources for the estimation of human transcription factor activities. Genome Res. 29, 1363–1375 (2019).
pubmed: 31340985 pmcid: 6673718 doi: 10.1101/gr.240663.118

Auteurs

Olivia Castellini-Pérez (O)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain.
University of Granada, Granada, Spain.

Elena Povedano (E)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain.
Spanish National Research Council (CSIC), Institute of Economy, Geography and Demography, Madrid (IEGD), Madrid, Spain.
Autonomous University of Madrid, Madrid, Spain.

Guillermo Barturen (G)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain.
Department of Genetics, Faculty of Sciences, University of Granada, Granada, Spain.

Manuel Martínez-Bueno (M)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain.

Andrii Iakovliev (A)

Usher Institute of Population Health Sciences and Informatics. University of Edinburgh Medical School, EH8 9YL, Edinburgh, UK.

Martin Kerick (M)

IBPLN-CSIC, Instituto de Parasitología y Biomedicina López-Neyra, Consejo Superior de Investigaciones Científicas, Granada, 18016, Spain.

Raúl López-Domínguez (R)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain.

Concepción Marañón (C)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain.

Javier Martín (J)

IBPLN-CSIC, Instituto de Parasitología y Biomedicina López-Neyra, Consejo Superior de Investigaciones Científicas, Granada, 18016, Spain.

Esteban Ballestar (E)

Epigenetics and Immune Disease Group, Josep Carreras Research Institute (IJC), 08916, Badalona, Barcelona, Spain.

María Orietta Borghi (MO)

Università degli Studi di Milano and Istituto Auxologico Italiano, Milan, Italy.

Weiliang Qiu (W)

Sanofi, Early Development and Research, Cambridge, MA, USA.

Cheng Zhu (C)

Sanofi, Precision Medicine & Computational Biology (PMCB), R&D, Cambridge, MA, USA.

Srinivas Shankara (S)

Sanofi, Precision Medicine & Computational Biology (PMCB), R&D, Cambridge, MA, USA.

Athina Spiliopoulou (A)

Usher Institute of Population Health Sciences and Informatics. University of Edinburgh Medical School, EH8 9YL, Edinburgh, UK.

Emanuele de Rinaldis (E)

Sanofi, Precision Medicine & Computational Biology (PMCB), R&D, Cambridge, MA, USA.

Elena Carnero-Montoro (E)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain. elena.carnero@genyo.es.
University of Granada, Granada, Spain. elena.carnero@genyo.es.

Marta E Alarcón-Riquelme (ME)

GENYO. Center for Genomics and Oncological Research Pfizer/University of Granada/Andalusian Regional Government, 18016, Granada, Spain. marta.alarcon@genyo.es.
Institute for Environmental Medicine, Karolinska Institutet, 171 67, Solna, Sweden. marta.alarcon@genyo.es.

Classifications MeSH